日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery, preclinical safety, and efficacy characterization of SMAC mimetic S-016-1348 as a potential cancer therapeutic.

对 SMAC 模拟物 S-016-1348 作为潜在癌症治疗药物进行发现、临床前安全性和有效性表征。

Sinha Abhipsa, Nengroo Mushtaq Ahmad, Ali Rafat, Khan Afsar Ali, Dutta Himangsu Sekhar, Singh Akhilesh, Saini Krishan Kumar, Tripathi Kiran, Katekar Roshan, Rathaur Shivam, Vaishnav Jayanti, Singh Gajendra, Afsar Mohammad, Meena Sanjeev, Sahu Anjna, Shaw Abhishek Kumar, Singh Kulranjan, Ramachandran Ravishankar, Chourasia Manish Kumar, Barthwal Manoj, Yadav Prem Narayan, Kshatri Aravind Singh, Rangarajan Radha, Nazir Aamir, Ampapathi Ravi Sankar, Gayen Jiaur Rahaman, Koley Dipankar, Haq Wahajul, Datta Dipak

1-Hydroxy-1,8-napthyridinone (DHN) Analogs Potently Inhibit Monkeypox Virus Resolvase (Mpr)

1-羟基-1,8-萘啶酮 (DHN) 类似物可有效抑制猴痘病毒分解酶 (Mpr)

Offei, Samuel; Mahoney, Jacob P; Wang, Ziyue; Pant, Anil; Ryu, Won Hee; Katekar, Roshan; Xie, Jiashu; Yang, Zhilong; Wang, Zhengqiang

Discovery of Small-Molecule Orthopoxvirus Resolvase Inhibitors with Antiviral Activity

发现具有抗病毒活性的小分子正痘病毒分解酶抑制剂

Mahoney, Jacob P; Offei, Samuel; Pant, Anil; Wang, Ziyue; Weiner, Benjamin; Yin, Lulu; Ryu, Won Hee; Katekar, Roshan; Williams, Jessica M; Aihara, Hideki; Yang, Zhilong; Wang, Zhengqiang

Methylation Enables Sensitive LC-MS/MS Quantification of Ciclopirox in a Mouse Pharmacokinetics Study

甲基化作用使得在小鼠药代动力学研究中能够对环吡咯烷酮进行灵敏的LC-MS/MS定量分析。

Katekar, Roshan; Wang, Zhengqiang; Xie, Jiashu

Norditerpene Natural Products from Subterranean Fungi with Anti-Parasitic Activity

具有抗寄生虫活性的地下真菌来源的北二萜类天然产物

Kolas, Alexandra; Rusman, Yudi; Maia, Ana C R G; Williams, Jessica M; Xie, Jiashu; Katekar, Roshan; Fumuso, Fernanda G; Cotto-Rosario, Alexis; Onoh, Chidiebere N; Baggar, Hanen; Piaskowski, Mary L; Baigorria, Christian; Paes, Raphaella; Chakrabarti, Debopam; Weible, Lyssa J; Ojo, Kayode K; O'Connor, Roberta M; Salomon, Christine E

Design, synthesis and profiling of highly potent antivirals targeting emerging drug-resistant HIV-1 variants

针对新出现的耐药性HIV-1变异株的高效抗病毒药物的设计、合成和分析

Jamey, Nicolas; Udayanga, D M Nirosh; Zhang, Huanchun; Ravichandran, Shreya M; Cai, Xinyong; Lorson, Zachary C; McFadden, William M; Ryu, Won Hee; Katekar, Roshan; Xie, Jiashu; Kirby, Karen A; Sarafianos, Stefan G; Wang, Zhengqiang

Evaluation of the Pharmacokinetics of the Pancreastatin Inhibitor PSTi8 Peptide in Rats: Integration of In Vitro and In Vivo Findings

胰腺抑素抑制剂 PSTi8 肽在大鼠体内的药代动力学评估:体外和体内研究结果的整合

Guru R Valicherla, Roshan A Katekar, Shailesh Dadge, Mohammed Riyazuddin, Anees A Syed, Sandeep K Singh, Athar Husain, Muhammad Wahajuddin, Jiaur R Gayen

PSTi8 with metformin ameliorates perimenopause induced steatohepatitis associated ER stress by regulating SIRT-1/SREBP-1c axis

PSTi8 与二甲双胍联合作用可通过调节 SIRT-1/SREBP-1c 轴改善围绝经期引起的脂肪性肝炎相关 ER 应激

Pragati Singh, Mohammad Irshad Reza, Anees A Syed, Richa Garg, Athar Husain, Roshan Katekar, Umesh K Goand, Mohammed Riyazuddin, Anand P Gupta, Jiaur R Gayen

Efficacy of manual therapy treatments for people with cervicogenic dizziness and pain: protocol of a randomised controlled trial

手法治疗对颈源性眩晕和疼痛患者的疗效:一项随机对照试验方案

Reid, Susan A; Rivett, Darren A; Katekar, Michael G; Callister, Robin

Phytotropins: III. NAPHTHYLPHTHALAMIC ACID BINDING SITES ON MAIZE COLEOPTILE MEMBRANES AS POSSIBLE RECEPTOR SITES FOR PHYTOTROPIN ACTION

植物促生素:III. 玉米胚芽鞘膜上的萘酞胺酸结合位点作为植物促生素作用的可能受体位点

Katekar, G F; Navé, J F; Geissler, A E