日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

CACHE Challenge #2: Targeting the RNA Site of the SARS-CoV-2 Helicase Nsp13

CACHE挑战#2:靶向SARS-CoV-2解旋酶Nsp13的RNA位点

Herasymenko, Oleksandra; Silva, Madhushika; Abu-Saleh, Abd Al-Aziz A; Ahmad, Ayaz; Alvarado-Huayhuaz, Jesus; Arce, Oscar E A; Armstrong, Roly J; Arrowsmith, Cheryl; Bachta, Kelly E; Beck, Hartmut; Berta, Denes; Bieniek, Mateusz K; Blay, Vincent; Bolotokova, Albina; Bourne, Philip E; Breznik, Marko; Brown, Peter J; Campbell, Aaron D G; Carosati, Emanuele; Chau, Irene; Cole, Daniel J; Cree, Ben; Dehaen, Wim; Denzinger, Katrin; Dos Santos Machado, Karina; Dunn, Ian; Durai, Prasannavenkatesh; Edfeldt, Kristina; Edwards, Aled; Fayne, Darren; Felfoldi, Daniel; Friston, Kallie; Ghiabi, Pegah; Gibson, Elisa; Günther, Judith; Gunnarsson, Anders; Hillisch, Alexander; Houston, Douglas R; Jensen, Jan Halborg; Harding, Rachel J; Harris, Kate S; Hoffer, Laurent; Hogner, Anders; Horton, Joshua T; Houliston, Scott; Hultquist, Judd F; Hutchinson, Ashley; Irwin, John J; Jukič, Marko; Kandwal, Shubhangi; Karlova, Andrea; Katis, Vittorio L; Kich, Ryan P; Kireev, Dmitri; Koes, David; Inniss, Nicole L; Lessel, Uta; Liu, Sijie; Loppnau, Peter; Lu, Wei; Martino, Sam; McGibbon, Miles; Meiler, Jens; Mettu, Akhila; Money-Kyrle, Sam; Moretti, Rocco; Moroz, Yurii S; Muvva, Charuvaka; Newman, Joseph A; Obendorf, Leon; Paige, Brooks; Pandit, Amit; Park, Keunwan; Perveen, Sumera; Pirie, Rachael; Poda, Gennady; Protopopov, Mykola; Pütter, Vera; Ricci, Federico; Roper, Natalie J; Rosta, Edina; Rzhetskaya, Margarita; Sabnis, Yogesh; Satchell, Karla J F; Schmitt Kremer, Frederico; Scott, Thomas; Seitova, Almagul; Steinmann, Casper; Talagayev, Valerij; Tarkhanova, Olga O; Tatum, Natalie J; Treleaven, Dakota; Velasque Werhli, Adriano; Walters, W Patrick; Wang, Xiaowen; Wells, Jude; Wells, Geoffrey; Westermaier, Yvonne; Wolber, Gerhard; Wortmann, Lars; Zhang, Jixian; Zhao, Zheng; Zheng, Shuangjia; Schapira, Matthieu

Safety and Efficacy of Busulphan Based on Dosing Patterns in the Real-World Management of Myeloproliferative Neoplasms

基于真实世界骨髓增生性肿瘤治疗中给药模式的白消安安全性和有效性

Mahdi, Ali; Rampotas, Alexandros; Roberts, Patrick; Stokes, Joanna; Mahdi, Eamon; Witherall, Ruth; Mannari, Deepak; Ibrahim, Naheed; Naylor, Georgina; Garg, Mamta; Manjra, Imran; Glancy, Paula; Katis, George; Bhagat, Sahil; Coppell, Jason; McGregor, Andrew; Frewin, Rebecca; Butt, Nauman M

Regulation of inositol 5-phosphatase activity by the C2 domain of SHIP1 and SHIP2.

SHIP1 和 SHIP2 的 C2 结构域对肌醇 5-磷酸酶活性的调节

Bradshaw William J, Kennedy Emma C, Moreira Tiago, Smith Luke A, Chalk Rod, Katis Vittorio L, Benesch Justin L P, Brennan Paul E, Murphy Emma J, Gileadi Opher

The mechanism of allosteric activation of SYK kinase derived from multiple phospho-ITAM-bound structures.

SYK激酶变构激活机制源于多个磷酸化ITAM结合结构

Bradshaw William J, Harris Gemma, Gileadi Opher, Katis Vittorio L

Evaluation of the RNA Silencing Suppression Activity of Three Cherry Virus F-Encoded Proteins

三种樱桃病毒F编码蛋白RNA沉默抑制活性的评价

Lotos, Leonidas; Katsiani, Asimina; Katis, Nikolaos I; Maliogka, Varvara I

Development of a time-resolved fluorescence resonance energy transfer ultra-high throughput screening assay targeting SYK and FCER1G interaction.

开发一种针对 SYK 和 FCER1G 相互作用的时间分辨荧光共振能量转移超高通量筛选检测方法

Du Yuhong, Wang Dongxue, Katis Vittorio L, Zoeller Elizabeth L, Qui Min, Levey Allan I, Gileadi Opher, Fu Haian

Characterizing left ventricular systolic dysfunction in sickle cell disease: three contrasting case reports

镰状细胞病左心室收缩功能障碍的特征:三个对比鲜明的病例报告

Katis, George; Srinivasan, Sridhar; Eleftheriou, Perla; Walker, Malcolm; Demetriades, Polyvios

Development of a Time-Resolved Fluorescence Resonance Energy Transfer ultra-high throughput screening assay for targeting SYK and FCER1G interaction

开发针对 SYK 和 FCER1G 相互作用的时间分辨荧光共振能量转移超高通量筛选检测方法

Yuhong Du, Dongxue Wang, Vittorio L Katis, Elizabeth L Zoeller, Min Qui, Allan I Levey, Opher Gileadi; Emory-SAGE-SGC TREAT-AD Center; Haian Fu

Development of SYK NanoBRET Cellular Target Engagement Assays for Gain-of-Function Variants

针对获得功能变体的 SYK NanoBRET 细胞靶标参与检测的开发

Jacob L Capener, James D Vasta, Vittorio L Katis, Ani Michaud, Michael T Beck, Sabrina C D Daglish, Sarit Cohen-Kedar, Efrat Shaham Barda, Stefanie Howell, Iris Dotan, Matthew B Robers, Alison D Axtman, Frances M Bashore

Development of SYK NanoBRET cellular target engagement assays for gain-of-function variants

开发用于功能获得性变异体的SYK NanoBRET细胞靶标结合分析方法

Capener, Jacob L; Vasta, James D; Katis, Vittorio L; Michaud, Ani; Beck, Michael T; Daglish, Sabrina C D; Cohen-Kedar, Sarit; Barda, Efrat Shaham; Howell, Stefanie; Dotan, Iris; Robers, Matthew B; Axtman, Alison D; Bashore, Frances M