日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting FOXM1 reshapes antitumor immunity to attenuate small cell lung cancer progression

靶向 FOXM1 可重塑抗肿瘤免疫,从而减缓小细胞肺癌的进展。

Khan, Md Arafat; Khan, Parvez; Fatima, Mahek; Rehman, Asad Ur; Anwar, Laiba; Alsafwani, Zahraa Wajih; Ahmad, Aatiya; Abbas Zaidi, Mohammad Ali; Cox, Jesse L; Zahid, Areem; Mohiuddin, Sameer; Kim, Sung Hoon; Santamaria-Barria, Juan A; Lakshmanan, Imayavaramban; Katzenellenbogen, Benita S; Katzenellenbogen, John A; Ganti, Apar K; Batra, Surinder K; Nasser, Mohd Wasim

JAK/STAT1-interferon-ISGylation networks in breast cancer resistance to inhibitors of FOXM1 and CDK4/6

JAK/STAT1-干扰素-ISGylation网络在乳腺癌对FOXM1和CDK4/6抑制剂的耐药性中发挥作用

Ziegler, Yvonne; Kumar, Sandeep; Saeh, Carlos M; Plotner, Blake N; Pento, Grace O; Kim, Sung Hoon; Raghavan, Alekya; Schiff, Rachel; Katzenellenbogen, John A; Katzenellenbogen, Benita S

Inhibition of FOXM1 Synergizes with BH3 Mimetics Venetoclax and Sonrotoclax in Killing Multiple Myeloma Cells through Repressing MYC Pathway

抑制FOXM1与BH3模拟物维奈托克和索罗托克协同作用,通过抑制MYC通路杀死多发性骨髓瘤细胞

Wen, Zhi; Wang, Yidan; Fox, Kathryn C; Bissonnette, Adam M; Moat, Luke F; Kitchner, Terrie E; Springstroh, Kelsey; Kim, Sung Hoon; Sheerar, Dagna S; Tanawattanacharoen, Patcharon; Leon, Chady A; Fagbemi, Seth O; Katzenellenbogen, John A; Hebbring, Scott J; Katzenellenbogen, Benita S; Janz, Siegfried; Onitilo, Adedayo A

OR04-08 Ligand Class Analysis Enables Predictive Models for Effective Antagonism of Endocrine Resistant Breast Cancer

OR04-08 配体类别分析可构建预测模型,有效拮抗内分泌耐药性乳腺癌

Ravani, Victoria Lis; Bagheri, Zahra; Brufsky, Adam M; Michelon, Isabella; O'Regan, Ruth; Lustberg, Maryam; Han, Hyo; Wang, Ming; Wander, Seth A; Nwachukwu, Jerome C; Min, Charles K; Kobylski, Robin R; Kim, Tahchur J; Hou, Yingwei; Kim, Sung Hoon; Hancock, Govinda R; Izard, Tina; Fanning, Sean W; Katzenellenbogen, Benita S; Katzenellenbogen, John A; Nettles, Kendall W

Chloroindazole based estrogen receptor β ligands with favorable pharmacokinetics promote functional remyelination and visual recovery

具有良好药代动力学特性的氯吲唑类雌激素受体β配体可促进功能性髓鞘再生和视力恢复。

Feri, Micah; Kim, Sung Hoon; Cardenas, Flavio D; Anderson, Alyssa M; Poole, Brandon T; Deshpande, Devang; Desfor, Shane; Atkinson, Kelley C; Peterson, Stephanie R; Nettles, Kendall W; Nwachukwu, Jerome C; Ajayi, Moyinoluwa T; Beltran, Fernando; Martin, David E; Tapia, Julio; Curtis, Carol D; Garcia-Castro, Martin I; Katzenellenbogen, Benita S; Katzenellenbogen, John A; Tiwari-Woodruff, Seema K

Benzestrol Isomer Stereochemistry Determines the Distinct Estrogenic Activities and Conformations of the Eight Isomers When Bound to Estrogen Receptor α.

苯雌酚异构体的立体化学决定了八种异构体与雌激素受体α结合时不同的雌激素活性和构象

Hou Yingwei, Nwachukwu Jerome C, Carlson Kathryn, Kim Sung Hoon, Angle Samantha, Jacobsen Eric N, Woods Toby, Mateus Sofia L, Fanning Sean W, Ziegler Yvonne, Katzenellenbogen Benita S, Nettles Kendall W, Katzenellenbogen John A

Phthalates Impair Estrogenic Regulation of HIF2α and Extracellular Vesicle Secretion by Human Endometrial Stromal Cells.

邻苯二甲酸酯会损害雌激素对人子宫内膜间质细胞 HIF2α 和细胞外囊泡分泌的调节作用

Beal Jacob R, Bhurke Arpita, Carlson Kathryn E, Katzenellenbogen John A, Yu Jie, Flaws Jodi A, Bagchi Indrani C, Bagchi Milan K

Iterative Catalyst-Controlled Diastereoselective Matteson Homologations Enable the Selective Synthesis of Benzestrol Isomers

迭代催化剂控制的非对映选择性马特森同系化反应实现了苯并雌二醇异构体的选择性合成

Angle, Samantha R; Sharma, Hayden A; Choi, Christie K; Carlson, Kathryn E; Hou, Yingwei; Nwachukwu, Jerome C; Kim, Sung Hoon; Katzenellenbogen, Benita S; Nettles, Kendall W; Katzenellenbogen, John A; Jacobsen, Eric N

Reprogramming of endothelial gene expression by tamoxifen inhibits angiogenesis and ERα-negative tumor growth

他莫昔芬对内皮细胞基因表达的重编程抑制了血管生成和 ERα 阴性肿瘤的生长

Chanaëlle Fébrissy, Marine Adlanmerini, Christel Péqueux, Frédéric Boudou, Mélissa Buscato, Adrien Gargaros, Silveric Gilardi-Bresson, Khrystyna Boriak, Henrik Laurell, Coralie Fontaine, Benita S Katzenellenbogen, John A Katzenellenbogen, Julie Guillermet-Guibert, Jean-François Arnal, Raphaël Metivi

Asymmetric allostery in estrogen receptor-α homodimers drives responses to the ensemble of estrogens in the hormonal milieu

雌激素受体α同源二聚体的不对称变构作用驱动对激素环境中多种雌激素的反应。

Min, Charles K; Nwachukwu, Jerome C; Hou, Yingwei; Russo, Robin J; Papa, Alexandra; Min, Jian; Peng, Rouming; Kim, Sung Hoon; Ziegler, Yvonne; Rangarajan, Erumbi S; Izard, Tina; Katzenellenbogen, Benita S; Katzenellenbogen, John A; Nettles, Kendall W