日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

In vitro toxicokinetics and metabolic profiling of methoxycathinones and methylthiocathinones using human liver systems and hyphenated mass spectrometry

利用人肝系统和联用质谱法对甲氧基卡西酮和甲基硫代卡西酮进行体外毒代动力学和代谢分析

Kroesen, Matthias D; Gampfer, Tanja M; Wagmann, Lea; Kavanagh, Pierce V; Brandt, Simon D; Meyer, Markus R

Bioisostere-Driven Discovery of SePP: A Selenium-Containing Polypharmacological Agent Relevant to Fragile X Syndrome

生物等排体驱动的SePP发现:一种与脆性X综合征相关的含硒多药理学药物

Wallach, Jason; Cameron, Sean; Dybek, Michael; Stanley, Branden; Orme, Christopher; Riad, Nour; Kavanagh, Pierce; Brandt, Simon D; Knapp, Adam; Gamrat, James; Jauhola-Straight, Rebekah; Adejare, Adeboye; Rogier, Alexander J; Tyagi, Richa; Canal, Clinton E

A Comparative Study Using Reversed-Phase and Hydrophilic Interaction Liquid Chromatography to Investigate the In Vitro and In Vivo Metabolism of Five Selenium-Containing Cathinone Derivatives

采用反相和亲水相互作用液相色谱法对五种含硒卡西酮衍生物的体外和体内代谢进行比较研究

Wagmann, Lea; Schmitt, Jana H; Gampfer, Tanja M; Brandt, Simon D; Scott, Kenneth; Kavanagh, Pierce V; Meyer, Markus R

Bioisosteric analogs of MDMA: Improving the pharmacological profile?

MDMA的生物等排体类似物:能否改善其药理特性?

Alberto-Silva Ana Sofia, Hemmer Selina, Bock Hailey A, da Silva Leticia Alves, Scott Kenneth R, Kastner Nina, Bhatt Manan, Niello Marco, Jäntsch Kathrin, Kudlacek Oliver, Bossi Elena, Stockner Thomas, Meyer Markus R, McCorvy John D, Brandt Simon D, Kavanagh Pierce, Sitte Harald H

Bioisosteric analogs of MDMA with improved pharmacological profile

具有改进药理特性的MDMA生物等排体类似物

Alberto-Silva, Ana Sofia; Hemmer, Selina; Bock, Hailey A; Alves da Silva, Leticia; Scott, Kenneth R; Kastner, Nina; Bhatt, Manan; Niello, Marco; Jäntsch, Kathrin; Kudlacek, Oliver; Bossi, Elena; Stockner, Thomas; Meyer, Markus R; McCorvy, John D; Brandt, Simon D; Kavanagh, Pierce; Sitte, Harald H

(2-Aminopropyl)benzo[β]thiophenes (APBTs) are novel monoamine transporter ligands that lack stimulant effects but display psychedelic-like activity in mice

(2-氨丙基)苯并[β]噻吩 (APBTs) 是一类新型单胺转运体配体,它们不具有兴奋作用,但在小鼠体内却表现出类似迷幻剂的活性。

Rudin, Deborah; McCorvy, John D; Glatfelter, Grant C; Luethi, Dino; Szöllősi, Dániel; Ljubišić, Tea; Kavanagh, Pierce V; Dowling, Geraldine; Holy, Marion; Jaentsch, Kathrin; Walther, Donna; Brandt, Simon D; Stockner, Thomas; Baumann, Michael H; Halberstadt, Adam L; Sitte, Harald H

Analytical characterization of N,N-diallyltryptamine (DALT) and 16 ring-substituted derivatives

N,N-二烯丙基色胺(DALT)及其16种环取代衍生物的分析表征

Brandt, Simon D; Kavanagh, Pierce V; Dowling, Geraldine; Talbot, Brian; Westphal, Folker; Meyer, Markus R; Maurer, Hans H; Halberstadt, Adam L