日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Use of new approach methodology for hepatic safety assessment of covalent inhibitor drug candidates.

采用新的方法对共价抑制剂候选药物进行肝脏安全性评价

Amberntsson Sara, Foster Alison J, Chouhan Bhavik, Wilkinson Stephen, Harlfinger Stephanie, Smith Graham, Kettle Jason G, Niedbala Michael, Kavanagh Stefan, Williams Dominic P

Discovery of a Novel Benzodiazepine Series of Cbl-b Inhibitors for the Enhancement of Antitumor Immunity

发现新型苯二氮卓类Cbl-b抑制剂可增强抗肿瘤免疫力

Boerth, Jeffrey A; Chinn, Alex J; Schimpl, Marianne; Bommakanti, Gayathri; Chan, Christina; Code, Erin L; Giblin, Kathryn A; Gohlke, Andrea; Hansel, Catherine S; Jin, Meizhong; Kavanagh, Stefan L; Lamb, Michelle L; Lane, Jordan S; Larner, Carrie J B; Mfuh, Adelphe M; Moore, Rachel K; Puri, Taranee; Quinn, Taylor R; Ye, Minwei; Robbins, Kevin J; Gancedo-Rodrigo, Miguel; Tang, Haoran; Walsh, Jarrod; Ware, Jamie; Wrigley, Gail L; Reddy, Iswarya Karapa; Zhang, Yun; Grimster, Neil P

Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate

三氨基嘧啶是一种速效且长效的抗疟疾候选药物。

Hameed P, Shahul; Solapure, Suresh; Patil, Vikas; Henrich, Philipp P; Magistrado, Pamela A; Bharath, Sowmya; Murugan, Kannan; Viswanath, Pavithra; Puttur, Jayashree; Srivastava, Abhishek; Bellale, Eknath; Panduga, Vijender; Shanbag, Gajanan; Awasthy, Disha; Landge, Sudhir; Morayya, Sapna; Koushik, Krishna; Saralaya, Ramanatha; Raichurkar, Anandkumar; Rautela, Nikhil; Roy Choudhury, Nilanjana; Ambady, Anisha; Nandishaiah, Radha; Reddy, Jitendar; Prabhakar, K R; Menasinakai, Sreenivasaiah; Rudrapatna, Suresh; Chatterji, Monalisa; Jiménez-Díaz, María Belén; Martínez, María Santos; Sanz, Laura María; Coburn-Flynn, Olivia; Fidock, David A; Lukens, Amanda K; Wirth, Dyann F; Bandodkar, Balachandra; Mukherjee, Kakoli; McLaughlin, Robert E; Waterson, David; Rosenbrier-Ribeiro, Lyn; Hickling, Kevin; Balasubramanian, V; Warner, Peter; Hosagrahara, Vinayak; Dudley, Adam; Iyer, Pravin S; Narayanan, Shridhar; Kavanagh, Stefan; Sambandamurthy, Vasan K