日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Development of Carborane-Based Benzothiazole Analogues as Cannabinoid Receptor Type 2 (CB(2)R) Ligands

开发基于碳硼烷的苯并噻唑类似物作为大麻素受体2型(CB(2)R)配体

Ueberham, Lea; Kazimir, Aleksandr; Deuther-Conrad, Winnie; Hey-Hawkins, Evamarie

Development of Carborane-Based Halogenated Naphthyridinone-Analogues as Cannabinoid Receptor Type 2 (CB(2)R) Ligands

开发基于碳硼烷的卤代萘啶酮类似物作为大麻素受体2型(CB(2)R)配体

Ueberham, Lea; Deuther-Conrad, Winnie; Lönnecke, Peter; Kazimir, Aleksandr; Hey-Hawkins, Evamarie

Advances in Diclofenac Derivatives: Exploring Carborane-Substituted N-Methyl and Nitrile Analogs for Anticancer Therapy.

双氯芬酸衍生物的研究进展:探索碳硼烷取代的N-甲基和腈类似物在抗癌治疗中的应用

Selg Christoph, Schuster Robert, Kazimir Aleksandr, Lönnecke Peter, Wolniewicz Mara, Schädlich Jonas, Laube Markus, Pietzsch Jens, Gordić Vuk, Krajnović Tamara, Mijatović Sanja, Maksimović-Ivanić Danijela, Hey-Hawkins Evamarie

Re-design and evaluation of diclofenac-based carborane-substituted prodrugs and their anti-cancer potential.

对基于双氯芬酸的碳硼烷取代前药进行重新设计和评价,并评估其抗癌潜力

Selg Christoph, Gordić Vuk, Krajnović Tamara, Buzharevski Antonio, Laube Markus, Kazimir Aleksandr, Lönnecke Peter, Wolniewicz Mara, Sárosi Menyhárt B, Schädlich Jonas, Pietzsch Jens, Mijatović Sanja, Maksimović-Ivanić Danijela, Hey-Hawkins Evamarie

Bipyraloxifene - a modified raloxifene vector against triple-negative breast cancer

双吡咯烷酮——一种针对三阴性乳腺癌的改良雷洛昔芬载体

Kazimir, Aleksandr; Götze, Tom; Murganić, Blagoje; Mijatović, Sanja; Maksimović-Ivanić, Danijela; Hey-Hawkins, Evamarie

Computer-guided design of Z domain peptides with improved inhibition of VEGF

计算机辅助设计Z结构域肽以提高对VEGF的抑制作用

Geist, Carsten; Useini, Abibe; Kazimir, Aleksandr; Kuempfel, Richy; Meiler, Jens; Lamers, Christina; Kalkhof, Stefan; Kuenze, Georg

Synthesis, Structure-Activity Relationships, Radiofluorination, and Biological Evaluation of [(18)F]RM365, a Novel Radioligand for Imaging the Human Cannabinoid Receptor Type 2 (CB2R) in the Brain with PET

本文研究了新型放射性配体[(18)F]RM365的合成、构效关系、放射性氟化及其在PET成像中对人脑内大麻素受体2型(CB2R)的生物学评价。

Teodoro, Rodrigo; Gündel, Daniel; Deuther-Conrad, Winnie; Kazimir, Aleksandr; Toussaint, Magali; Wenzel, Barbara; Bormans, Guy; Hey-Hawkins, Evamarie; Kopka, Klaus; Brust, Peter; Moldovan, Rareş-Petru

Development of the High-Affinity Carborane-Based Cannabinoid Receptor Type 2 PET Ligand [(18)F]LUZ5-d(8)

高亲和力碳硼烷基大麻素受体2型PET配体[(18)F]LUZ5-d(8)的开发

Ueberham, Lea; Gündel, Daniel; Kellert, Martin; Deuther-Conrad, Winnie; Ludwig, Friedrich-Alexander; Lönnecke, Peter; Kazimir, Aleksandr; Kopka, Klaus; Brust, Peter; Moldovan, Rareş-Petru; Hey-Hawkins, Evamarie

Correction: Kazimir et al. Metallodrugs against Breast Cancer: Combining the Tamoxifen Vector with Platinum(II) and Palladium(II) Complexes. Pharmaceutics 2023, 15, 682

更正:Kazimir 等人,《抗乳腺癌金属药物:他莫昔芬载体与铂(II)和钯(II)配合物的联合应用》,Pharmaceutics 2023, 15, 682

Kazimir, Aleksandr; Schwarze, Benedikt; Lönnecke, Peter; Jelača, Sanja; Mijatović, Sanja; Maksimović-Ivanić, Danijela; Hey-Hawkins, Evamarie

Exploring the potential of tamoxifen-based copper(ii) dichloride in breast cancer therapy.

探索基于他莫昔芬的二氯化铜(II)在乳腺癌治疗中的潜力

Kazimir Aleksandr, Schwarze Benedikt, Lönnecke Peter, Jelača Sanja, Mijatović Sanja, Maksimović-Ivanić Danijela, Hey-Hawkins Evamarie