日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Chemosensitization of cancer cells by KU-0060648, a dual inhibitor of DNA-PK and PI-3K

DNA-PK 和 PI-3K 双重抑制剂 KU-0060648 对癌细胞的化学增敏作用

Joanne M Munck, Michael A Batey, Yan Zhao, Helen Jenkins, Caroline J Richardson, Celine Cano, Michele Tavecchio, Jody Barbeau, Julia Bardos, Liam Cornell, Roger J Griffin, Keith Menear, Andrew Slade, Pia Thommes, Niall M B Martin, David R Newell, Graeme C M Smith, Nicola J Curtin

AZD8055 is a potent, selective, and orally bioavailable ATP-competitive mammalian target of rapamycin kinase inhibitor with in vitro and in vivo antitumor activity

AZD8055 是一种强效、选择性、口服生物利用度高的 ATP 竞争性哺乳动物雷帕霉素激酶抑制剂,具有体外和体内抗肿瘤活性

Christine M Chresta, Barry R Davies, Ian Hickson, Tom Harding, Sabina Cosulich, Susan E Critchlow, John P Vincent, Rebecca Ellston, Darren Jones, Patrizia Sini, Dominic James, Zoe Howard, Phillippa Dudley, Gareth Hughes, Lisa Smith, Sharon Maguire, Marc Hummersone, Karine Malagu, Keith Menear, Richa