日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Myelin Oligodendrocyte Glycoprotein (MOG)35-55 Mannan Conjugate Induces Human T-Cell Tolerance and Can Be Used as a Personalized Therapy for Multiple Sclerosis

髓鞘少突胶质细胞糖蛋白 (MOG)35-55 甘露聚糖缀合物可诱导人 T 细胞耐受,并可用作多发性硬化症的个体化治疗。

Rodi, Maria; de Lastic, Anne-Lise; Panagoulias, Ioannis; Aggeletopoulou, Ioanna; Kelaidonis, Kostas; Matsoukas, John; Apostolopoulos, Vasso; Mouzaki, Athanasia

Computational Evidence for Bisartan Arginine Blockers as Next-Generation Pan-Antiviral Therapeutics Targeting SARS-CoV-2, Influenza, and Respiratory Syncytial Viruses

比沙坦精氨酸阻滞剂作为下一代泛抗病毒疗法的计算证据,可靶向SARS-CoV-2、流感病毒和呼吸道合胞病毒

Ridgway, Harry; Apostolopoulos, Vasso; Moore, Graham J; Gadanec, Laura Kate; Zulli, Anthony; Swiderski, Jordan; Tsiodras, Sotirios; Kelaidonis, Konstantinos; Chasapis, Christos T; Matsoukas, John M

Structural Features Influencing the Bioactive Conformation of Angiotensin II and Angiotensin A: Relationship between Receptor Desensitization, Addiction, and the Blood-Brain Barrier

影响血管紧张素 II 和血管紧张素 A 生物活性构象的结构特征:受体脱敏、成瘾和血脑屏障之间的关系

Graham J Moore, Harry Ridway, Laura Kate Gadanec, Vasso Apostolopoulos, Anthony Zulli, Jordan Swiderski, Konstantinos Kelaidonis, Veroniki P Vidali, Minos-Timotheos Matsoukas, Christos T Chasapis, John M Matsoukas0

W254 in furin functions as a molecular gate promoting anti-viral drug binding: Elucidation of putative drug tunneling and docking by non-equilibrium molecular dynamics

弗林蛋白酶中的W254作为分子门控促进抗病毒药物结合:通过非平衡分子动力学阐明假定的药物隧道和对接机制

Ridgway, Harry; Orbell, John D; Matsoukas, Minos-Timotheos; Kelaidonis, Konstantinos; Moore, Graham J; Tsiodras, Sotiris; Gorgoulis, Vasilis G; Chasapis, Christos T; Apostolopoulos, Vasso; Matsoukas, John M

Network-Based Prediction of Side Effects of Repurposed Antihypertensive Sartans against COVID-19 via Proteome and Drug-Target Interactomes

基于蛋白质组和药物靶点相互作用组的抗高血压药物沙坦类药物再利用治疗COVID-19的副作用网络预测

Kiouri, Despoina P; Ntallis, Charalampos; Kelaidonis, Konstantinos; Peana, Massimiliano; Tsiodras, Sotirios; Mavromoustakos, Thomas; Giuliani, Alessandro; Ridgway, Harry; Moore, Graham J; Matsoukas, John M; Chasapis, Christos T

Computational and Enzymatic Studies of Sartans in SARS-CoV-2 Spike RBD-ACE2 Binding: The Role of Tetrazole and Perspectives as Antihypertensive and COVID-19 Therapeutics

沙坦类药物在 SARS-CoV-2 刺突 RBD-ACE2 结合中的计算和酶学研究:四唑的作用以及作为抗高血压和 COVID-19 治疗药物的前景

Konstantinos Kelaidonis, Irene Ligielli, Spiros Letsios, Veroniki P Vidali, Thomas Mavromoustakos, Niki Vassilaki, Graham J Moore, Weronika Hoffmann, Katarzyna Węgrzyn, Harry Ridgway, Christos T Chasapis, John M Matsoukas2

Existence of Quantum Pharmacology in Sartans: Evidence in Isolated Rabbit Iliac Arteries

沙坦类药物中存在量子药理学:来自兔离体髂动脉的证据

Laura Kate Gadanec, Jordan Swiderski, Vasso Apostolopoulos, Kostantinos Kelaidonis, Veroniki P Vidali, Aleksander Canko, Graham J Moore, John M Matsoukas, Anthony Zulli

Discovery of a new generation of angiotensin receptor blocking drugs: Receptor mechanisms and in silico binding to enzymes relevant to SARS-CoV-2

新一代血管紧张素受体阻滞剂的发现:受体机制及与SARS-CoV-2相关酶的计算机模拟结合

Ridgway, Harry; Moore, Graham J; Mavromoustakos, Thomas; Tsiodras, Sotirios; Ligielli, Irene; Kelaidonis, Konstantinos; Chasapis, Christos T; Gadanec, Laura Kate; Zulli, Anthony; Apostolopoulos, Vasso; Petty, Russell; Karakasiliotis, Ioannis; Gorgoulis, Vassilis G; Matsoukas, John M

Diminazene Aceturate Reduces Angiotensin II Constriction and Interacts with the Spike Protein of Severe Acute Respiratory Syndrome Coronavirus 2

乙酰脲酸二甲胺可降低血管紧张素 II 收缩并与严重急性呼吸综合征冠状病毒 2 的刺突蛋白相互作用

John M Matsoukas, Laura Kate Gadanec, Anthony Zulli, Vasso Apostolopoulos, Konstantinos Kelaidonis, Irene Ligielli, Kalliopi Moschovou, Nikitas Georgiou, Panagiotis Plotas, Christos T Chasapis, Graham Moore, Harry Ridgway, Thomas Mavromoustakos

The Human Myelin Proteome and Sub-Metalloproteome Interaction Map: Relevance to Myelin-Related Neurological Diseases

人类髓鞘蛋白质组和亚金属蛋白质组相互作用图谱:与髓鞘相关神经系统疾病的相关性

Chasapis, Christos T; Kelaidonis, Konstantinos; Ridgway, Harry; Apostolopoulos, Vasso; Matsoukas, John M