日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-based design of an opioid receptor modulator for enhanced morphine analgesia

基于结构的阿片受体调节剂设计及其在增强吗啡镇痛中的应用

Wang, Yue; Luo, Ping; Xu, Haiyan; Zhan, Li; Sakamoto, Kensuke; Li, Mingyu; Wang, Jing; Huang, Xi-Ping; Zhou, Jianhui; Liu, Tao; Suo, Yanrui; Fan, Wenjia; He, Xinheng; Xu, Youwei; Cai, Yongjie; Wang, Chao; Zhao, Yuxi; Dai, Antao; Lai, Yali; Yuan, Qingning; Hu, Wen; Wu, Kai; Yang, Dehua; Cheng, Xi; Lu, Xiaojie; Krumm, Brian; Kenakin, Terry; Zhang, Jian; Roth, Bryan L; Gao, Zhaobing; Xu, H Eric; Zhuang, Youwen

Molecular mechanisms of inverse agonism via κ-opioid receptor-G protein complexes.

通过α-阿片受体-G蛋白复合物的反向激动作用的分子机制

Tyson Aaliyah S, Khan Saif, Motiwala Zenia, Han Gye Won, Zhang Zixin, Ranjbar Mohsen, Styrpejko Daniel, Ramos-Gonzalez Nokomis, Woo Stone, Villers Kelly, Landaker Delainey, Kenakin Terry, Shenvi Ryan, Majumdar Susruta, Gati Cornelius

Differential Effects of Sodium on Agonist-Induced Conformational Transitions and Signaling at μ and κ Opioid Receptors

钠对μ和κ阿片受体激动剂诱导的构象转变和信号传导的不同影响

Kuijer, Michael Bram; Fulton, Camryn J; Albert, Talia L; Knobloch, Paloma; Wang, Jing; Krumm, Brian E; Che, Tao; Varga, Balazs R; Majumdar, Susruta; Katritch, Vsevolod; Gumpper, Ryan H; Kenakin, Terry; Huang, Xi-Ping; Roth, Bryan L

Differential effects of sodium on agonist-induced conformational transitions and signaling at μ and κ opioid receptors

钠对μ和κ阿片受体激动剂诱导的构象转变和信号传导的不同影响

Kuijer, Bram; Fulton, Camryn J; Albert, Talia L; Knobloch, Paloma M; Wang, Jing; Krumm, Brian E; Che, Tao; Varga, Balazs R; Majumdar, Susruta; Katritch, Vsevolod; Gumpper, Ryan H; Kenakin, Terry; Huang, Xi-Ping; Roth, Bryan L

Intracellular Allosteric Antagonist of the Olfactory Receptor OR51E2

嗅觉受体 OR51E2 的细胞内变构拮抗剂

Tatjana Abaffy, Olivia Fu, Maira Harume-Nagai, Josh M Goldenberg, Victor Kenyon, Terry Kenakin

Structural insights into the human niacin receptor HCA2-Gi signalling complex

人类烟酸受体 HCA2-Gi 信号复合物的结构洞察

Yang Yang #, Hye Jin Kang #, Ruogu Gao #, Jingjing Wang, Gye Won Han, Jeffrey F DiBerto, Lijie Wu, Jiahui Tong, Lu Qu, Yiran Wu, Ryan Pileski, Xuemei Li, Xuejun Cai Zhang, Suwen Zhao, Terry Kenakin, Quan Wang, Raymond C Stevens, Wei Peng, Bryan L Roth, Zihe Rao, Zhi-Jie Liu

Community guidelines for GPCR ligand bias: IUPHAR review 32

GPCR配体偏向性社区指南:IUPHAR审查32

Kolb, Peter; Kenakin, Terry; Alexander, Stephen P H; Bermudez, Marcel; Bohn, Laura M; Breinholt, Christian S; Bouvier, Michel; Hill, Stephen J; Kostenis, Evi; Martemyanov, Kirill A; Neubig, Rick R; Onaran, H Ongun; Rajagopal, Sudarshan; Roth, Bryan L; Selent, Jana; Shukla, Arun K; Sommer, Martha E; Gloriam, David E

Virtual discovery of melatonin receptor ligands to modulate circadian rhythms

虚拟发现褪黑激素受体配体来调节昼夜节律

Reed M Stein #, Hye Jin Kang #, John D McCorvy #, Grant C Glatfelter #, Anthony J Jones, Tao Che, Samuel Slocum, Xi-Ping Huang, Olena Savych, Yurii S Moroz, Benjamin Stauch, Linda C Johansson, Vadim Cherezov, Terry Kenakin, John J Irwin, Brian K Shoichet, Bryan L Roth, Margarita L Dubocovich3

Differential Roles of Extracellular Histidine Residues of GPR68 for Proton-Sensing and Allosteric Modulation by Divalent Metal Ions

GPR68 胞外组氨酸残基对二价金属离子质子感应和变构调节的不同作用

Xi-Ping Huang, Terrence P Kenakin, Shuo Gu, Brian K Shoichet, Bryan L Roth

Design, Synthesis, and Characterization of Ogerin-Based Positive Allosteric Modulators for G Protein-Coupled Receptor 68 (GPR68)

基于 Ogerin 的 G 蛋白偶联受体 68 (GPR68) 正向变构调节剂的设计、合成和表征

Yu, Xufen; Huang, Xi-Ping; Kenakin, Terry P; Slocum, Samuel T; Chen, Xin; Martini, Michael L; Liu, Jing; Jin, Jian