Development of a Covalent Inhibitor of c-Jun N-Terminal Protein Kinase (JNK) 2/3 with Selectivity over JNK1
开发一种对 c-Jun N 端蛋白激酶 (JNK) 2/3 具有选择性而非 JNK1 的共价抑制剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.2c01834
Wenchao Lu ,Yao Liu ,Yang Gao ,Qixiang Geng ,Deepak Gurbani ,Lianbo Li ,Scott B Ficarro ,Cynthia J Meyer ,Dhiraj Sinha ,Inchul You ,Jason Tse ,Zhixiang He ,Wenzhi Ji ,Jianwei Che ,Audrey Y Kim ,Tengteng Yu ,Kenneth Wen ,Kenneth C Anderson ,Jarrod A Marto ,Kenneth D Westover ,Tinghu Zhang ,Nathanael S Gray