日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

TLR3 forms a laterally aligned multimeric complex along double-stranded RNA for efficient signal transduction

TLR3 沿双链 RNA 形成横向排列的多聚体复合物,实现有效的信号转导

Kentaro Sakaniwa #, Akiko Fujimura #, Takuma Shibata #, Hideki Shigematsu, Toru Ekimoto, Masaki Yamamoto, Mitsunori Ikeguchi, Kensuke Miyake, Umeharu Ohto, Toshiyuki Shimizu

Tetrasubstituted imidazoles as incognito Toll-like receptor 8 a(nta)gonists

四取代咪唑作为隐性 Toll 样受体 8 激动剂

Yi Yang #, Adam Csakai #, Shuangshuang Jiang #, Christina Smith, Hiromi Tanji, Jian Huang, Torey Jones, Kentaro Sakaniwa, Lindsey Broadwell, Chengrui Shi, Subada Soti, Umeharu Ohto, Yaohui Fang, Shu Shen, Fei Deng, Toshiyuki Shimizu, Hang Yin

Small-molecule inhibition of TLR8 through stabilization of its resting state

通过稳定 TLR8 的静息状态来抑制 TLR8

Shuting Zhang, Zhenyi Hu, Hiromi Tanji, Shuangshuang Jiang, Nabanita Das, Jing Li, Kentaro Sakaniwa, Jin Jin, Yanyan Bian, Umeharu Ohto, Toshiyuki Shimizu, Hang Yin

Small-Molecule TLR8 Antagonists via Structure-Based Rational Design

基于结构的合理设计小分子 TLR8 拮抗剂

Zhenyi Hu, Hiromi Tanji, Shuangshuang Jiang, Shuting Zhang, Kyoin Koo, Jean Chan, Kentaro Sakaniwa, Umeharu Ohto, Albert Candia, Toshiyuki Shimizu, Hang Yin