日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural and dynamic features of cagrilintide binding to calcitonin and amylin receptors.

卡格里林肽与降钙素和胰淀素受体结合的结构和动力学特征

Cao Jianjun, Belousoff Matthew J, Johnson Rachel M, Keov Peter, Mariam Zamara, Deganutti Giuseppe, Christopoulos George, Hick Caroline A, Reedtz-Runge Steffen, Glendorf Tine, Ballarín-González Borja, Raun Kirsten, Bayly-Jones Charles, Wootten Denise, Sexton Patrick M

De novo design of miniprotein agonists and antagonists targeting G protein-coupled receptors.

从头设计靶向 G 蛋白偶联受体的微型蛋白激动剂和拮抗剂

Muratspahić Edin, Feldman David, Kim David E, Qu Xiangli, Bratovianu Ana-Maria, Rivera-Sánchez Paula, Dimitri Federica, Cao Jason, Cary Brian P, Belousoff Matthew J, Keov Peter, Chen Qingchao, Ren Yue, Fine Justyn, Sappington Isaac, Schlichthaerle Thomas, Zhang Jason Z, Pillai Arvind, Mihaljević Ljubica, Bauer Magnus, Torres Susana Vázquez, Motmaen Amir, Lee Gyu Rie, Tran Long, Wang Xinru, Goreshnik Inna, Vafeados Dionne K, Svendsen Justin E, Hosseinzadeh Parisa, Lindegaard Nicolai, Brandt Matthäus, Waltenspühl Yann, Deibler Kristine, Oostdyk Luke, Cao William, Anantharaman Lakshmi, Stewart Lance, Halloran Lauren, Spangler Jamie B, Sexton Patrick M, Roth Bryan L, Krumm Brian E, Wootten Denise, Tate Christopher G, Norn Christoffer, Baker David

Discovery and development of macrocyclic peptide modulators of the cannabinoid 2 receptor

大麻素2受体大环肽调节剂的发现与开发

Tomašević, Nataša; Emser, Fabiola Susanna; Muratspahić, Edin; Gattringer, Jasmin; Hasinger, Simon; Hellinger, Roland; Keov, Peter; Felkl, Manuel; Gertsch, Jürg; Becker, Christian F W; Gruber, Christian W

Orphan receptor GPR37L1 remains unliganded

孤儿受体GPR37L1仍未配体结合

Ngo, Tony; Wilkins, Brendan P; So, Sean S; Keov, Peter; Chahal, Kirti K; Finch, Angela M; Coleman, James L J; Kufareva, Irina; Smith, Nicola J

Nature-inspired dimerization as a strategy to modulate neuropeptide pharmacology exemplified with vasopressin and oxytocin

以血管加压素和催产素为例,利用自然界启发的二聚化策略来调节神经肽药理学

Dekan, Zoltan; Kremsmayr, Thomas; Keov, Peter; Godin, Mathilde; Teakle, Ngari; Dürrauer, Leopold; Xiang, Huang; Gharib, Dalia; Bergmayr, Christian; Hellinger, Roland; Gay, Marina; Vilaseca, Marta; Kurzbach, Dennis; Albericio, Fernando; Alewood, Paul F; Gruber, Christian W; Muttenthaler, Markus

The TRPV4 Agonist GSK1016790A Regulates the Membrane Expression of TRPV4 Channels

TRPV4激动剂GSK1016790A调节TRPV4通道的膜表达

Baratchi, Sara; Keov, Peter; Darby, William G; Lai, Austin; Khoshmanesh, Khashayar; Thurgood, Peter; Vahidi, Parisa; Ejendal, Karin; McIntyre, Peter

Discovery of peptide probes to modulate oxytocin-type receptors of insects

发现能够调节昆虫催产素型受体的肽探针

Keov, Peter; Liutkevičiūtė, Zita; Hellinger, Roland; Clark, Richard J; Gruber, Christian W

Molecular determinants of allosteric modulation at the M1 muscarinic acetylcholine receptor.

M1毒蕈碱乙酰胆碱受体变构调节的分子决定因素

Abdul-Ridha Alaa, López Laura, Keov Peter, Thal David M, Mistry Shailesh N, Sexton Patrick M, Lane J Robert, Canals Meritxell, Christopoulos Arthur