日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Monovalent pseudo-natural products supercharge degradation of IDO1 by its native E3 KLHDC3.

单价伪天然产物可加速 IDO1 的天然 E3 KLHDC3 的降解。

Hennes Elisabeth, Lucas Belén, Scholes Natalie S, Cheng Xiu-Fen, Scott Daniel C, Bischoff Matthias, Reich Katharina, Gasper Raphael, Lucas María, Xu Teng Teng, Rossini Sofia, Pulvermacher Lisa-Marie, Dötsch Lara, Imrichova Hana, Brause Alexandra, Führer Siska, Naredla Kesava Reddy, Sievers Sonja, Kumar Kamal, Janning Petra, Orabona Ciriana, Gersch Malte, Murray Peter J, Schulman Brenda A, Winter Georg E, Ziegler Slava, Waldmann Herbert

Design, Synthesis, and Structural Evolution of Pseudo-Natural Product IDO1 Inhibitors and Degraders

拟天然产物IDO1抑制剂和降解剂的设计、合成和结构演变

Cheng, Xiu-Fen; Lucas, Belén; Lampe, Philipp; Ugel, Stefano; Chen, Suyuan; Unger, Anke; Bischoff, Matthias; Adariani, Soheila Rezaei; Naredla, Kesava Reddy; Kumar, Kamal; Schmidt, Annika; Strohmann, Carsten; Janning, Petra; Gasper, Raphael; Lucas, María; Gersch, Malte; Sievers, Sonja; Bronte, Vincenzo; Ziegler, Slava; Waldmann, Herbert

Outcome measures used in the conservative management of people with non-specific thoracic spine pain (NTSP): a scoping review protocol

非特异性胸椎疼痛(NTSP)患者保守治疗中使用的结局指标:范围界定综述方案

Kovanur Sampath, Kesava; Fleischmann, Michael; Vaughan, Brett

Functional Ambidexterity of an Ancient Nucleic Acid-Binding Domain

古老核酸结合域的功能性双侧性

Weil-Ktorza, Orit; Naveh-Tassa, Segev; Fridmann-Sirkis, Yael; Despotović, Dragana; Cherukuri, Kesava Phaneendra; Corlett, Tatsuya; Levy, Yaakov; Metanis, Norman; Longo, Liam M

PP2A methylesterase, PME-1, and PP2A methyltransferase, LCMT-1, control sensitivity to impairments caused by injury-related oligomeric tau.

PP2A 甲基酯酶 PME-1 和 PP2A 甲基转移酶 LCMT-1 控制着对损伤相关寡聚 tau 引起的损伤的敏感性。

Sundaresh Sowmya N, Vogel Edward W 3rd, Hue Christopher D, Zhang Hong, Staniszewski Anna, Berman Hanna L, Gill Zafar, Asam Kesava, Liang Siqi, Shen Liwei, Gnanaprakash Madhumathi, Acquarone Erica, Masone Antonio, Fà Mauro, Kanaan Nicholas M, Morrison Barclay 3rd, Arancio Ottavio, Nicholls Russell E

Schwann cell Lrp1 deletion drives trigeminal neuron sensitization and orofacial pain by modulating mitochondrial function and TRPV1/TRPA1 activity.

雪旺细胞 Lrp1 缺失通过调节线粒体功能和 TRPV1/TRPA1 活性驱动三叉神经元敏化和口面部疼痛。

Gong Zhiting, Zhang Morgan, Liu Naijiang, Asam Kesava, Martellucci Stefano, Aouizerat Bradley, Campana Wendy, Ye Yi

Aberrant DNA methylation of genes regulating CD4+ T cell HIV-1 reservoir in women with HIV

感染艾滋病毒的女性体内,调控CD4+ T细胞HIV-1储存库的基因存在异常DNA甲基化。

Ke Xu ,Xinyu Zhang ,Kesava Asam ,Bryan C Quach ,Grier P Page ,Deborah Konkle-Parker ,Claudia Martinez ,Cecile D Lahiri ,Elizabeth F Topper ,Mardge H Cohen ,Seble G Kassaye ,Jack DeHovitz ,Mark H Kuniholm ,Nancie M Archin ,Amir Valizadeh ,Phyllis C Tien ,Vincent C Marconi ,Dana B Hancock ,Eric O Johnson ,Bradley E Aouizerat

Development of high-titer class-switched antibody responses to phosphorylated amino acids is prevalent in pancreatic ductal adenocarcinoma

胰腺导管腺癌中普遍存在针对磷酸化氨基酸的高滴度类别转换抗体反应。

Aguiar, Talita; Mashiko, Shunya; Asam, Kesava; Roy, Poulomi; Wang, Shikun; Frank, Katharina; Dietzel, Max; Schahadat, Luca G Z; Ausmeier, Mattea; Hertel, Andrea; Duan, Zhe Ran Susan; Aouizerat, Bradley; Genkinger, Jeanine M; Remotti, Helen; Zorn, Emmanuel

TNFR1 Suppression by XPro1595 Reduces Peripheral Neuropathies Associated with Perineural Invasion in Female Mice

XPro1595抑制TNFR1可减轻雌性小鼠神经周围侵袭相关的周围神经病变

Morgan Zhang ,Naijiang Liu ,Kesava Asam ,Charles Meng ,Bradley Aouizerat ,Yi Ye

Examination of aperture layout designs for an adaptive-stationary multi-pinhole brain-dedicated SPECT system

对自适应固定式多孔脑专用SPECT系统的孔径布局设计进行研究

Kalluri, Kesava S; Zeraatkar, Navid; Auer, Benjamin; Pells, Sophia; Pretorius, P Hendrik; Richards, Garrett R; May, Micaehla; Momsen, Neil; Doty, Kimberly; Gonzales, Maria Ruiz; Fromme, Timothy; Truong, Kevin; Kupinski, Matthew A; Kuo, Phillip H; Furenlid, Lars R; King, Michael A