日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Site-Specific Quadruple-Functionalised Antibodies

位点特异性四功能抗体

Journeaux, Toby; Geeson, Michael B; Murray, Thomas V; Papworth, Monika A; Gothard, Matt; Kettle, Jason G; Vasco, Aldrin V; Bernardes, Gonçalo J L

Focused Structure-Based Virtual Screening Identifies Novel Inhibitors of SOS1

基于结构的虚拟筛选鉴定出SOS1的新型抑制剂

Bonomo, Silvia; Gibault, Floriane; Bagal, Sharan K; Blackwell, J Henry; Breed, Jason; Collie, Gavin W; Couturier, Maxime; Diène, Coura; Di Fruscia, Paolo; Gray, Sean; Hughes, Craig; Jeyaharan, Dhadchayini; Kettle, Jason G; Milbradt, Alexander G; Northall, Sarah; Peters, Katherine; Stubbs, Christopher J; Underwood, Elizabeth; Chen, Yunhua; Hao, Haie; Lainchbury, Michael D

Use of new approach methodology for hepatic safety assessment of covalent inhibitor drug candidates.

采用新的方法对共价抑制剂候选药物进行肝脏安全性评价

Amberntsson Sara, Foster Alison J, Chouhan Bhavik, Wilkinson Stephen, Harlfinger Stephanie, Smith Graham, Kettle Jason G, Niedbala Michael, Kavanagh Stefan, Williams Dominic P

Vinylpyridine as a Tunable Covalent Warhead Targeting C797 in EGFR.

乙烯基吡啶作为可调控共价弹头靶向 EGFR 中的 C797

Pemberton Nils, Compagne Nina, Argyrou Argyrides, Evertsson Emma, Gunnarsson Anders, Kettle Jason G, Orme Jonathan P, Ward Richard A

Drugging the undruggable: a computational chemist's view of KRAS(G12C)

药物治疗:计算化学家眼中的 KRAS(G12C)

Bodnarchuk, Michael S; Cassar, Doyle J; Kettle, Jason G; Robb, Graeme; Ward, Richard A