日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural studies identify angiotensin II receptor blocker-like compounds as branched-chain ketoacid dehydrogenase kinase inhibitors

结构研究发现,血管紧张素II受体阻滞剂样化合物是支链酮酸脱氢酶激酶抑制剂。

Shenping Liu ,Bethany L Kormos ,John D Knafels ,Parag V Sahasrabudhe ,Amy Rosado ,Ruth F Sommese ,Allan R Reyes ,Jessica Ward ,Rachel J Roth Flach ,Xiaochun Wang ,Leanne M Buzon ,Matthew R Reese ,Samit K Bhattacharya ,Kiyoyuki Omoto ,Kevin J Filipski

BDK inhibition acts as a catabolic switch to mimic fasting and improve metabolism in mice

BDK抑制剂可作为一种分解代谢开关,模拟禁食状态,从而改善小鼠的新陈代谢。

Eliza Bollinger ,Matthew Peloquin ,Jenna Libera ,Bina Albuquerque ,Evanthia Pashos ,Arun Shipstone ,Angela Hadjipanayis ,Zhongyuan Sun ,Gang Xing ,Michelle Clasquin ,John C Stansfield ,Brendan Tierney ,Steven Gernhardt ,C Parker Siddall ,Timothy Greizer ,Frank J Geoly ,Sarah R Vargas ,Lily C Gao ,George Williams ,Mackenzie Marshall ,Amy Rosado ,Claire Steppan ,Kevin J Filipski ,Bei B Zhang ,Russell A Miller ,Rachel J Roth Flach

Selective pharmacological inhibition of the sodium-dependent phosphate cotransporter NPT2a promotes phosphate excretion

选择性药理抑制钠依赖性磷酸盐转运体 NPT2a 可促进磷酸盐排泄

Valerie Clerin, Hiroshi Saito, Kevin J Filipski, An Hai Nguyen, Jeonifer Garren, Janka Kisucka, Monica Reyes, Harald Jüppner