The curcumin analog HO-3867 selectively kills cancer cells by converting mutant p53 protein to transcriptionally active wildtype p53
姜黄素类似物 HO-3867 通过将突变 p53 蛋白转化为转录活性野生型 p53 来选择性杀死癌细胞
期刊:Journal of Biological Chemistry
影响因子:4
doi:10.1074/jbc.RA117.000950
Esha Madan, Taylor M Parker, Matthias R Bauer, Alisha Dhiman, Christopher J Pelham, Masaki Nagane, M Lakshmi Kuppusamy, Matti Holmes, Thomas R Holmes, Kranti Shaik, Kevin Shee, Salome Kiparoidze, Sean D Smith, Yu-Soon A Park, Jennifer J Gomm, Louise J Jones, Ana R Tomás, Ana C Cunha, Karuppaiyah Sel