日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Proteomic characterization and cytotoxic potential of proteins from Cuscuta (Cuscuta epithymum (L.) crude herbal product against MCF-7 human breast cancer cell line

菟丝子(Cuscuta epithymum (L.))粗草药产品对 MCF-7 人乳腺癌细胞系的蛋白质组学表征和细胞毒性潜力

Umaima Akhtar, Yamna Khurshid, Bishoy El-Aarag, Basir Syed, Ishtiaq A Khan, Keykavous Parang, Aftab Ahmed

Design, Synthesis, and Evaluation of Oleyl-WRH Peptides for siRNA Delivery

用于 siRNA 递送的油酰-WRH 肽的设计、合成和评估

Mrigank Shekhar Rai, Muhammad Imran Sajid, Jonathan Moreno, Keykavous Parang, Rakesh Kumar Tiwari

Structure-Based Rational Design of Small α-Helical Peptides with Broad-Spectrum Activity against Multidrug-Resistant Pathogens

基于结构的合理设计具有广谱抗多药耐药病原体活性的小α-螺旋肽

Sandeep Lohan, Anastasia G Konshina, Roman G Efremov, Innokentiy Maslennikov, Keykavous Parang

Modified Linear Peptides Effectively Silence STAT-3 in Breast Cancer and Ovarian Cancer Cell Lines

修饰的线性肽可有效抑制乳腺癌和卵巢癌细胞系中的 STAT-3

Dindyal Mandal, Sandeep Lohan, Muhammad Imran Sajid, Abdulelah Alhazza, Rakesh Kumar Tiwari, Keykavous Parang, Hamidreza Montazeri Aliabadi

Structural Analysis and Activity Correlation of Amphiphilic Cyclic Antimicrobial Peptides Derived from the [W4R4] Scaffold

基于[W4R4]骨架的两亲性环状抗菌肽的结构分析及活性关联

Shaima A El-Mowafi, Anastasia G Konshina, Eman H M Mohammed, Nikolay A Krylov, Roman G Efremov, Keykavous Parang

Design, Synthesis, and Antiproliferative Activity of Benzopyran-4-One-Isoxazole Hybrid Compounds

苯并吡喃-4-酮-异噁唑杂化化合物的设计、合成及抗增殖活性

Shilpi Gupta, Shang Eun Park, Saghar Mozaffari, Bishoy El-Aarag, Keykavous Parang, Rakesh Kumar Tiwari

Tolfenamic Acid Derivatives: A New Class of Transcriptional Modulators with Potential Therapeutic Applications for Alzheimer's Disease and Related Disorders

托芬那酸衍生物:一类具有治疗阿尔茨海默病及相关疾病潜力的新型转录调节剂

Jaunetta Hill, Karim E Shalaby, Syed W Bihaqi, Bothaina H Alansi, Benjamin Barlock, Keykavous Parang, Richard Thompson, Khalid Ouararhni, Nasser H Zawia

Structure-Activity Relationship Study of Subtype-Selective Positive Modulators of KCa2 Channels

KCa2通道亚型选择性正调节剂的构效关系研究

Naglaa Salem El-Sayed, Young-Woo Nam, Polina A Egorova, Hai Minh Nguyen, Razan Orfali, Mohammad Asikur Rahman, Grace Yang, Heike Wulff, Ilya Bezprozvanny, Keykavous Parang, Miao Zhang

Membrane-Active Cyclic Amphiphilic Peptides: Broad-Spectrum Antibacterial Activity Alone and in Combination with Antibiotics

膜活性环状两亲肽:单独及与抗生素联合使用时具有广谱抗菌活性

Eman H M Mohammed, Sandeep Lohan, Tarra Ghaffari, Shilpi Gupta, Rakesh K Tiwari, Keykavous Parang

Bis-Cinnamamide Derivatives as APE/Ref-1 Inhibitors for the Treatment of Human Melanoma

双肉桂酰胺衍生物作为 APE/Ref-1 抑制剂用于治疗人类黑色素瘤

Razan Alhazmi, Shirley Tong, Shaban Darwish, Elina Khanjani, Bharti Khungar, Swati Chawla, Zhonghui Zheng, Richard Chamberlin, Keykavous Parang, Sun Yang