日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Enhancing the therapeutic window for Spectinamide anti-tuberculosis Agents: Synthesis, Evaluation, and activation of phosphate prodrug 3408

扩大Spectinamide抗结核药物的治疗窗口:磷酸前药3408的合成、评价和活化

Liu, Jiuyu; Lukka, Pradeep B; Ektnitphong, Victoria A; Parmar, Keyur R; Wagh, Santosh; Lu, Yan; Lee, Robin B; Scherbakov, Dimitri; Wang, Han; Zimmerman, Matthew D; Meibohm, Bernd; Robertson, Gregory T; Dartois, Vêronique; Böttger, Erik C; Lenaerts, Anne J; Lee, Richard E

Efficacy of a brain-penetrant antiviral in lethal Venezuelan and eastern equine encephalitis mouse models

脑穿透性抗病毒药物在致命性委内瑞拉脑炎和东部马脑炎小鼠模型中的疗效

Cao, Xufeng; Yang, Dong; Parvathareddy, Jyothi; Chu, Yong-Kyu; Kim, Eun Jung; Fitz-Henley, Jhewelle N; Li, Xiaoyu; Lukka, Pradeep B; Parmar, Keyur R; Temrikar, Zaid H; Dhole, Priya; Adcock, Robert Scott; Gabbard, Jon; Bansal, Shruti; Lee, Jasper; Zalduondo, Lillian; Hayes, Ernestine; Stabenow, Jennifer; Meibohm, Bernd; Fitzpatrick, Elizabeth A; Bailey, Kevin; Campos, Rafael K; Julander, Justin G; Rossi, Shannan L; Chung, Donghoon; Jonsson, Colleen B; Golden, Jennifer E

Development of a Minimalistic Physiologically Based Pharmacokinetic (mPBPK) Model for the Preclinical Development of Spectinamide Antibiotics

开发用于Spectinamide类抗生素临床前开发的极简生理药代动力学(mPBPK)模型

Parmar, Keyur R; Lukka, Pradeep B; Wagh, Santosh; Temrikar, Zaid H; Liu, Jiuyu; Lee, Richard E; Braunstein, Miriam; Hickey, Anthony J; Robertson, Gregory T; Gonzalez-Juarrero, Mercedes; Edginton, Andrea; Meibohm, Bernd