Discovery of Five SOS2 Fragment Hits with Binding Modes Determined by SOS2 X-Ray Cocrystallography
利用SOS2 X射线共晶体学方法发现了五个SOS2片段结合位点及其结合模式。
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.3c02140
Smith, Christopher R; Chen, Dan; Christensen, James G; Coulombe, René; Féthière, James; Gunn, Robin J; Hollander, Johan; Jones, Benjamin; Ketcham, John M; Khare, Shilpi; Kuehler, Jon; Lawson, J David; Marx, Matthew A; Olson, Peter; Pearson, Kelly E; Ren, Cynthia; Tsagris, Denise; Ulaganathan, Thirumalaiselvi; Van't Veer, Inge; Wang, Xiaolun; Ivetac, Anthony