日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Another Kid on the Block: Long-acting FGF21 Analogue to Treat Dyslipidemia and Fatty Liver

又一款新药问世:长效FGF21类似物用于治疗血脂异常和脂肪肝

Yang, Ranyao; Xu, Aimin; Kharitonenkov, Alexei

FGF19 and FGF21: In NASH we trust

FGF19 和 FGF21:在 NASH 中,我们信赖它们

Talukdar, Saswata; Kharitonenkov, Alexei

Glucagon receptor signaling regulates weight loss via central KLB receptor complexes

胰高血糖素受体信号通过中枢 KLB 受体复合物调节减肥

Shelly R Nason, Jessica Antipenko, Natalie Presedo, Stephen E Cunningham, Tanya H Pierre, Teayoun Kim, Jodi R Paul, Cassie Holleman, Martin E Young, Karen L Gamble, Brian Finan, Richard DiMarchi, Chad S Hunter, Alexei Kharitonenkov, Kirk M Habegger

Withdrawal: Increased expression of fibroblast growth factor 21 (FGF21) during chronic undernutrition causes growth hormone insensitivity in chondrocytes by inducing leptin receptor overlapping transcript (LEPROT) and leptin receptor overlapping transcript-like 1 (LEPROTL1) expression

撤退:慢性营养不良期间成纤维细胞生长因子21 (FGF21) 表达增加,通过诱导瘦素受体重叠转录物 (LEPROT) 和瘦素受体重叠转录物样1 (LEPROTL1) 的表达,导致软骨细胞对生长激素不敏感。

Wu, Shufang; Grunwald, Tal; Kharitonenkov, Alexei; Dam, Julie; Jockers, Ralf; Luca, Francesco De

Molecular elements in FGF19 and FGF21 defining KLB/FGFR activity and specificity

FGF19 和 FGF21 中的分子元素决定了 KLB/FGFR 活性和特异性

Archita Agrawal, Sebastian Parlee, Diego Perez-Tilve, Pengyun Li, Jia Pan, Piotr A Mroz, Ann Maria Kruse Hansen, Birgitte Andersen, Brian Finan, Alexei Kharitonenkov, Richard D DiMarchi

Fibroblast activation protein (FAP) as a novel metabolic target

成纤维细胞活化蛋白(FAP)作为新型代谢靶点

Miguel Angel Sánchez-Garrido, Kirk M Habegger, Christoffer Clemmensen, Cassie Holleman, Timo D Müller, Diego Perez-Tilve, Pengyun Li, Archita S Agrawal, Brian Finan, Daniel J Drucker, Matthias H Tschöp, Richard D DiMarchi, Alexei Kharitonenkov

The Nuclear Receptor Rev-erbα Regulates Adipose Tissue-specific FGF21 Signaling

核受体 Rev-erbα 调节脂肪组织特异性 FGF21 信号传导

Jennifer Jager, Fenfen Wang, Bin Fang, Hee-Woong Lim, Lindsey C Peed, David J Steger, Kyoung-Jae Won, Alexei Kharitonenkov, Andrew C Adams, Mitchell A Lazar

Interplay between FGF21 and insulin action in the liver regulates metabolism

FGF21与胰岛素在肝脏中的相互作用调节代谢

Emanuelli, Brice; Vienberg, Sara G; Smyth, Graham; Cheng, Christine; Stanford, Kristin I; Arumugam, Manimozhiyan; Michael, Mervyn D; Adams, Andrew C; Kharitonenkov, Alexei; Kahn, C Ronald

Genetic disruption of uncoupling protein 1 in mice renders brown adipose tissue a significant source of FGF21 secretion

小鼠体内解偶联蛋白1基因的遗传破坏使得棕色脂肪组织成为FGF21分泌的重要来源。

Keipert, Susanne; Kutschke, Maria; Lamp, Daniel; Brachthäuser, Laura; Neff, Frauke; Meyer, Carola W; Oelkrug, Rebecca; Kharitonenkov, Alexei; Jastroch, Martin

Central Fibroblast Growth Factor 21 Browns White Fat via Sympathetic Action in Male Mice

中枢成纤维细胞生长因子 21 通过雄性小鼠的交感神经作用使白色脂肪变成棕色

Nicholas Douris, Darko M Stevanovic, Ffolliott M Fisher, Theodore I Cisu, Melissa J Chee, Ngoc L Nguyen, Eleen Zarebidaki, Andrew C Adams, Alexei Kharitonenkov, Jeffrey S Flier, Timothy J Bartness, Eleftheria Maratos-Flier