日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of BMS-986365, a First-in-Class Dual Androgen Receptor Ligand-Directed Degrader and Antagonist, for the Treatment of Advanced Prostate Cancer.

发现 BMS-986365,一种首创的双重雄激素受体配体导向降解剂和拮抗剂,用于治疗晚期前列腺癌。

Nayak Surendra, Norris John D, Ammirante Massimo, Rychak Emily, Wardell Suzanne E, Liao Debbie, Toyama Brandon, Kandimalla Raju, Christoforou Andy, Tsuji Toshiya, Liu Ken, Tran Minerva, Meiring Joseph, Reiss Samantha, Piccotti Joseph R, Baughman Joshua M, Fontanillo Celia, Khater Marwa, Mortensen Deborah S, Cathers Brian, Bence Neil, Pierce Daniel W, Plantevin-Krenitsky Veronique, Rathkopf Dana, Hansen Joshua D, Hamann Lawrence G, Narla Rama Krishna, Arora Vivek K, McDonnell Donald P, Rolfe Mark, Xu Shuichan

Elucidating binding hot spots and structural stability in sirtuin family proteins for selective inhibitors: a computational approach

阐明sirtuin家族蛋白的结合热点和结构稳定性,以开发选择性抑制剂:一种计算方法

Rawlins, Lettie E; Maroofian, Reza; Cannon, Stuart J; Daana, Muhannad; Zamani, Mina; Ghani, Shamsul; Leslie, Joseph S; Ubeyratna, Nishanka; Khan, Nasar; Khan, Hamid; Scardamaglia, Annarita; Cloarec, Robin; Khan, Shujaat Ali; Umair, Muhammad; Sadeghian, Saeid; Galehdari, Hamid; Al-Maawali, Almundher; Al-Kindi, Adila; Azizimalamiri, Reza; Shariati, Gholamreza; Ahmad, Faraz; Al-Futaisi, Amna; Rodriguez Cruz, Pedro M; Salazar-Villacorta, Ainara; Ndiaye, Moustapha; Diop, Amadou G; Sedaghat, Alireza; Saberi, Alihossein; Hamid, Mohammad; Zaki, Maha S; Vona, Barbara; Owrang, Daniel; Alhashem, Abdullah M; Obeid, Makram; Khan, Amjad; Beydoun, Ahmad; Najjar, Marwan; Tajsharghi, Homa; Zifarelli, Giovanni; Bauer, Peter; Hakami, Wejdan S; Al Hashem, Amal M; Boustany, Rose-Mary N; Burglen, Lydie; Alavi, Shahryar; Gunning, Adam C; Owens, Martina; Karimiani, Ehsan G; Gleeson, Joseph G; Milh, Mathieu; Salah, Somaya; Khan, Jahangir; Haucke, Volker; Wright, Caroline F; McGavin, Lucy; Elpeleg, Orly; Shabbir, Muhammad I; Houlden, Henry; Ebner, Michael; Baple, Emma L; Crosby, Andrew H; Dhar, Atika; Kitani, Atsushi; Strober, Warren; Bohall, Bradley S; Gorbis, Alexander; Gorbis, Eda; Chopra, Pradeep; Kandeel, Samah; El-Beltagi, Eman M; Wang, Wei-ren; Yan, Lin; Zhao, Chuan-ying; He, Cong-cong; Gao, Xing-Hua; Li, Linhui; Zhang, Shuangxi; Yue, Jianghuan; Wang, Xiuli; Li, Cuiting; Wang, Lulu; Li, Xiaoling; Lin, Aifen; Yan, Wei-Hua; Ouyang, Chaowei; Zhang, Dandan; Lei, Changbin; Morey, Manoviraj Gajendra; Illanad, Gouri H; Rasool, Mahaboobkhan; Chooklin, Serge; Chuklin, Serhii; An, Lina; Han, Yidi; Sun, Xiaohui; Wang, Lili; Guo, Lei; Long, Yu; Li, Dan; Jian, Xuemin; Yang, Zhi; Leng, Ting; Wang, Xilian; Zhang, Wanxue; Ge, Xinyun; Li, Nan; Yin, Yuan; Li, Xiaoan; Wang, Chunying; Zhang, Meihua; Bode, Erik L; Krasniqi, Samanda; Rosenthal, Annika; Friedel, Eva; Schlagenhauf, Florian; Sebold, Miriam; Wei, Hongxia; Li, Zhe; Liu, Zi'ang; Wu, Baofeng; Li, Ru; Xu, Ming; Yang, Xifeng; Yin, Jianhong; Zhang, Yi; Liu, Yunfeng; Kitase, Yukiko; Ji, Jia; Bonewald, Lynda F; Prideaux, Matthew; Roh, Hyun Cheol; Peng, Gang; Lin, Ying; Wen, Deng-tai; Huang, Jianhuang; Wang, Qixiu; Chen, Jianning; Parri, Muralidhar; Singh, Kiratmeet; Xing, Yun; Liu, Jiaxin; Wu, Linrui; Zhang, Ke; Yang, Shengbo; Srisuwan, Tanida; Kornsuthisopon, Chatvadee; Nowwarote, Nunthawan; Zhu, Xiaofei; Dissanayaka, Waruna Lakmal; Osathanon, Thanaphum; Sun, Jingjing; Zhang, Kai; Li, Panpan; Xu, Wenyue; Ding, Kaimo; Zhang, Bidan; Zhao, Bei; Zhang, Danwei; Sirajo, Mujittapha Umar; Obie, Rukevwe; Mukhtar, Abubakar I; Abdullahi, Nasiru M; Taniyohwo, Enaohwo M; Oyem, John C; Badamasi, Ibrahim M; Deb, Vishal Kumar; Mukherjee, Abhishek; Pathak, Surajit; Paul, Sujay; Duttaroy, Asim K; Adhikari, Suman; Gao, Huiquan; Ma, Tao; Jiang, Qinqin; Gao, Lanfang; Li, Jinfang; Wang, Shubo; Liu, Ziyong; Zhang, Zhixin; Wu, Gang; He, Wenxin; Zhou, Fuxin; Xu, XiuRong; Lai, JiuXin; Cheng, Shiming; Shuai, Qi; Tian, Jun; Yang, Wenlong; Huang, Santing; Tutu, Paul; Altamura, Gennaro; Daraban Bocaneti, Florentina; Hritcu, Ozana Maria; Pasca, Aurelian-Sorin; Dascalu, Mihaela Anca; Horodincu, Loredana; Tanase, Oana Irina; Mares, Mihai; Borzacchiello, Giuseppe; Yang, Guanhao; Huang, Xuan; Qiu, Duorun; Wang, Anzhao; Liu, Denghui; Liu, Zhongtang; Nuccio, Daniel A; Grippo, Angela; Singh, Pallavi; Gao, Xiaomeng; Wu, Yihan; Zheng, Ronglian; Kou, Yining; Xing, Huili; Li, Kun; Zhang, Meng; Priyadharshini, Eswaran; Sandhya, Maddi; Anand, Theerthagiri; Angamuthu, Mahalingam; Murugan, Marimuthu; Tharmalingam, Nagendran; Senthilraja, Govindasamy; Meng, Yonghui; He, Jinjun; Yan, An; Che, Bangwei; Tang, Kaifa; Zhang, Tao; Vukić, Dragana; Du, Qiupei; Cherian, Anna; Amoruso, Damiano; Brožinová, Květoslava; Wacheul, Ludivine; Lacovich, Valentina; Zorbas, Christiane; Yadav, Leena; Sedmík, Jiří; Keskitalo, Salla; Hajji, Khadija; Stejskal, Stanislav; Varjosalo, Markku; Lafontaine, Denis L J; Keegan, Liam P; O’Connell, Mary A; Allichon, Marie-Charlotte; Espinosa, Jeanne; Cole, Rebecca H; Ko, Mei-Chuan; Vanhoutte, Peter; Joffe, Max E; Abd El-kader, Marwa; Farrag, Eman A E; El-Gamal, Randa; El Nashar, Eman Mohamed; Alshehri, Areej M; Aldahhan, Rashid A; Al-khater, Khulood M; El-Desouky, Sara; El-Sherbeni, M W; Ebrahim, Neven A; Truitt, Kate; Walsh, McKenna E; Dalton, Michelle R; Cai, Jiali; Zhang, Yaojian; Zhang, Tian; Wu, Mengyi; Wang, Dijun; Yin, Chunyan; Nie, Xueke; Chen, Lan; Sun, Zhihu; Liu, Chanming; Yan, Xiaojing; Kong, Weihao; Wang, Jiawen; Zhang, Kangjie; Wang, Xingyu; Zhang, Jianlin; Sharma, Deepak; Muniyan, Rajiniraja

Rescue Therapy With Pegcetacoplan in a Patient With Proliferative Glomerulonephritis With Monoclonal Immunoglobulin Deposits

使用培塞他考普兰对伴有单克隆免疫球蛋白沉积的增生性肾小球肾炎患者进行挽救治疗

Dastoor, Hormaz; Khater, Emad; Al Salam, Suhail; Holt, Stephen G

Rapid dissolving microneedle patch integrated with benidipine-loaded nanotransfersomes for transdermal drug delivery: optimization, characterizations, and preclinical bioavailability assessment

用于透皮给药的快速溶解微针贴片与载有贝尼地平的纳米转运体相结合:优化、表征和临床前生物利用度评估

Al-Japairai, Khater; Almurisi, Samah Hamed; Alheibshy, Fawaz; Abdul-Halim, Nadiya; Mahmood, Syed

Harnessing faba bean MAGIC populations for enhanced protein content, yield, and agronomic performance in diverse environments

利用蚕豆MAGIC种群提高不同环境下的蛋白质含量、产量和农艺性状

Abou Khater, Lynn; Maalouf, Fouad; Walker, Cassandra; Bouhlal, Outmane; Aloui, Khawla; Balech, Rind; Mahmoudi, Kaoutar El; Ibriz, Mohammed; Ogbonnaya, Francis Chuks; Kumar, Shiv

The oral maternal microbiome plays a role in the development of cleft lip and palate condition in children

母体口腔微生物群在儿童唇腭裂的发生发展中起着一定作用

Khater, Safaa I; Hussein, Mohamed M A; Abdel-Magied, Saydat S; Lotfy, Marwa M; Khamis, Tarek; Abdelaziz, Sahar; Mostafa, Mahmoud; El-Shaer, Noha Osama; El-Emam, Mahran Mohamed Abd; Guima, Suzana Eiko Sato; Bischain, Bárbara; Morais Gama, Lívia C; Faria, Agatha Cristhina; Lourenço, Talita; Bueno, Daniela Franco; Heller, Debora; Passos-Bueno, Maria Rita; Setubal, João C

Whole-genome sequencing-based characterization of resistome and virulome in Klebsiella pneumoniae isolated from ready-to-eat foods

基于全基因组测序的即食食品中分离的肺炎克雷伯菌耐药组和毒力组特征分析

Anajirih, Nuha; Anagreyyah, Sulaiman A; Brangsch, Hanka; Moustafa, Shawky; Khater, Dalia F; Gesraha, Ahmed S; Rizk, Amira M; Neubauer, Heinrich; Wareth, Gamal

Unlocking the Diagnostic Challenge of Tuberculosis and Sarcoidosis Intrathoracic Lymphadenopathy: Potential Role of HMGB1 and miRNA-221 as Diagnostic Tools

破解结核病和结节病胸内淋巴结肿大的诊断难题:HMGB1 和 miRNA-221 作为诊断工具的潜在作用

Kamel, Fatma Z; Ismail, Nagwan Adel; Khater, Asmaa Z; El Shahawy, Alia A; Almadani, Noura; Sankarapandian, Chandrakala; Hammad, Noha M

Exploring the Association of Interleukin 13 Polymorphism (rs20541) and Serum Lipocalin 2 with Risk and Disability in Multiple Sclerosis

探讨白细胞介素 13 多态性 (rs20541) 和血清脂质运载蛋白 2 与多发性硬化症风险和残疾的关联

Kamel, Fatma Z; El Shahawy, Alia A; Abdelaziz, Eman Ahmed; Mohamed, Eman Atef; El Shahawy, Aya A; Hassaneen, Ahmad M; Khater, Asmaa Z; Mokhtar, Ghada A; Boghdady, Wesam Abdelmoniem Hafez

KM-DBSCAN: an enhanced density and centroid based border detection framework for data reduction towards green AI

KM-DBSCAN:一种基于密度和质心的增强型边界检测框架,用于数据降维,以实现绿色人工智能

AboElsaad, Mohamed Yasser; Farouk, Mohamed; Khater, Hatem A