日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, Synthesis, and In Vitro and In Silico Study of New Hybrid 1-(2-(4-Arylthiazol-2-yl)hydrazineylidene)-5,6-dihydro-4H-pyrrolo[3,2,1-ij]quinolin-2-ones as Factor Xa and Factor XIa Inhibitors

新型杂合1-(2-(4-芳基噻唑-2-基)肼基亚甲基)-5,6-二氢-4H-吡咯并[3,2,1-ij]喹啉-2-酮作为因子Xa和因子XIa抑制剂的设计、合成及体外和计算机模拟研究

Skoptsova, Anna A; Geronikaki, Athina; Petrou, Anthi; Novichikhina, Nadezhda P; Podoplelova, Nadezhda A; Bykov, Georgii A; Anis'kov, Aleksandr A; Soloveva, Svetlana A; Shikhaliev, Khidmet S

Design, Synthesis, and Evaluation of New Hybrid Derivatives of 5,6-Dihydro-4H-pyrrolo[3,2,1-ij]quinolin-2(1H)-one as Potential Dual Inhibitors of Blood Coagulation Factors Xa and XIa

设计、合成和评价5,6-二氢-4H-吡咯并[3,2,1-ij]喹啉-2(1H)-酮的新型杂合衍生物作为血液凝固因子Xa和XIa的潜在双重抑制剂

Skoptsova, Anna A; Geronikaki, Athina; Novichikhina, Nadezhda P; Sulimov, Alexey V; Ilin, Ivan S; Sulimov, Vladimir B; Bykov, Georgii A; Podoplelova, Nadezhda A; Pyankov, Oleg V; Shikhaliev, Khidmet S

Synthesis and PASS-assisted evaluation of new heterocyclic compounds containing hydroquinoline scaffolds

含有氢化喹啉骨架的新型杂环化合物的合成及 PASS 辅助评估

Gizachew Mulugeta Manahelohe, Khidmet Safarovich Shikhaliev

Rapid Deposition of the Biomimetic Hydroxyapatite-Polydopamine-Amino Acid Composite Layers onto the Natural Enamel

快速将仿生羟基磷灰石-聚多巴胺-氨基酸复合层沉积到天然牙釉质上

Seredin, Pavel; Goloshchapov, Dmitry; Emelyanova, Anna; Eremeev, Konstantin; Peshkov, Yaroslav; Shikhaliev, Khidmet; Potapov, Andrey; Ippolitov, Yury; Kashkarov, Vladimir; Nesterov, Dmitry; Shapiro, Kirill; Freitas, Raul O; Mahdy, Iman A

Fabrication and Characterization of Thin Metal Films Deposited by Electroless Plating with Organic Additives for Electrical Circuits Applications

采用含有机添加剂的化学镀法制备和表征用于电路应用的金属薄膜

Buylov, Nikita S; Sotskaya, Nadezhda V; Kozaderov, Oleg A; Shikhaliev, Khidmet S; Potapov, Andrey Yu; Polikarchuk, Vladimir A; Rodivilov, Sergey V; Pobedinskiy, Vitaly V; Grechkina, Margaryta V; Seredin, Pavel V

6-Hydroxy-2,2,4-trimethyl-1,2,3,4-tetrahydroquinoline Alleviates Oxidative Stress and NF-κB-Mediated Inflammation in Rats with Experimental Parkinson's Disease

6-羟基-2,2,4-三甲基-1,2,3,4-四氢喹啉可减轻实验性帕金森病大鼠的氧化应激和NF-κB介导的炎症

Kryl'skii, Evgenii D; Razuvaev, Grigorii A; Popova, Tatyana N; Medvedeva, Svetlana M; Shikhaliev, Khidmet S

6-Hydroxy-2,2,4-trimethyl-1,2-dihydroquinoline Demonstrates Anti-Inflammatory Properties and Reduces Oxidative Stress in Acetaminophen-Induced Liver Injury in Rats

6-羟基-2,2,4-三甲基-1,2-二氢喹啉具有抗炎特性,并能减轻对乙酰氨基酚诱导的大鼠肝损伤中的氧化应激。

Kryl'skii, Evgenii D; Kravtsova, Svetlana E; Popova, Tatyana N; Matasova, Larisa V; Shikhaliev, Khidmet S; Medvedeva, Svetlana M

Synthesis of 4,5-Dihydro-1 H-[1,2]dithiolo[3,4- c]quinoline-1-thione Derivatives and Their Application as Protein Kinase Inhibitors

4,5-二氢-1H-[1,2]二硫代[3,4-c]喹啉-1-硫酮衍生物的合成及其作为蛋白激酶抑制剂的应用

Svetlana M Medvedeva, Khidmet S Shikhaliev

A novel synthetic approach to hydroimidazo[1,5-b]pyridazines by the recyclization of itaconimides and HPLC-HRMS monitoring of the reaction pathway

一种通过衣康酰亚胺的重环化反应合成氢化咪唑并[1,5-b]哒嗪的新方法,并利用高效液相色谱-高分辨率质谱监测反应路径。

Vandyshev, Dmitry Yu; Shikhaliev, Khidmet S; Potapov, Andrey Yu; Krysin, Michael Yu; Zubkov, Fedor I; Sapronova, Lyudmila V