日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Guided Optimization of 4-Chloro-Pyrazolopyridine Analogs for Covalent PREP Inhibition

基于结构的4-氯吡唑并吡啶类似物优化用于共价PREP抑制

Thakur, Kalyani; Fucci, Ian; Pandian, Joshua; Suazo, Kiall F; Monteiro, Diana C F; Yoo, Euna

Chemical tools to define and manipulate interferon-inducible Ubl protease USP18

定义和操纵干扰素诱导的 Ubl 蛋白酶 USP18 的化学工具

Griffin J Davis #, Anthony O Omole #, Yejin Jung #, Wioletta Rut, Ronald Holewinski, Kiall F Suazo, Hong-Rae Kim, Mo Yang, Thorkell Andresson, Marcin Drag, Euna Yoo

Potent β-lactam-based tyrosyl-DNA phosphodiesterase 1 inhibitors identified by a virtual screen.

通过虚拟筛选鉴定出强效β-内酰胺类酪氨酰-DNA磷酸二酯酶1抑制剂

Zhao Xue Zhi, Wang Wenjie, Suazo Kiall F, Al Mahmud Md Rasel, Agama Keli, Lountos George T, Andresson Thorkell, Pommier Yves, Burke Terrence R Jr

Hierarchical small molecule inhibition of MYST acetyltransferases

MYST乙酰转移酶的分级小分子抑制

Chen, Xuemin; Castroverde, Alexandra; Perez, Minervo; Holewinski, Ronald; Suazo, Kiall F; Karki, Rashmi; Andressen, Thorkell; Garcia, Benjamin A; Meier, Jordan L

Paralogue-Selective Degradation of the Lysine Acetyltransferase EP300

赖氨酸乙酰转移酶EP300的旁系同源选择性降解

Chen, Xuemin; Crawford, McKenna C; Xiong, Ying; Shaik, Anver Basha; Suazo, Kiall F; Bauer, Ludwig G; Penikalapati, Manini S; Williams, Joycelyn H; Huber, Kilian V M; Andressen, Thorkell; Swenson, Rolf E; Meier, Jordan L

Targeted sulfur(VI) fluoride exchange-mediated covalent modification of a tyrosine residue in the catalytic pocket of tyrosyl-DNA phosphodiesterase 1

靶向硫(VI)氟化物交换介导的酪氨酰-DNA磷酸二酯酶1催化口袋中酪氨酸残基的共价修饰

Xue Zhi Zhao, Idris A Barakat, George T Lountos, Wenjie Wang, Keli Agama, Md Rasel Al Mahmud, Kiall F Suazo, Thorkell Andresson, Yves Pommier, Terrence R Burke Jr

Improved synthesis and application of an alkyne-functionalized isoprenoid analogue to study the prenylomes of motor neurons, astrocytes and their stem cell progenitors.

改进炔烃官能化异戊二烯类似物的合成和应用,以研究运动神经元、星形胶质细胞及其干细胞祖细胞的异戊二烯体

Suazo Kiall F, Mishra Vartika, Maity Sanjay, Auger Shelby A, Justyna Katarzyna, Petre Alexandru M, Ottoboni Linda, Ongaro Jessica, Corti Stefania P, Lotti Francesco, Przedborski Serge, Distefano Mark D

Broadening the Utility of Farnesyltransferase-Catalyzed Protein Labeling Using Norbornene-Tetrazine Click Chemistry

利用降冰片烯-四嗪点击化学拓展法尼基转移酶催化蛋白质标记的应用范围

Auger, Shelby A; Venkatachalapathy, Sneha; Suazo, Kiall Francis G; Wang, Yiao; Sarkis, Alexander W; Bernhagen, Kaitlyn; Justyna, Katarzyna; Schaefer, Jonas V; Wollack, James W; Plückthun, Andreas; Li, Ling; Distefano, Mark D

Discovery of a Tunable Heterocyclic Electrophile 4-Chloro-pyrazolopyridine That Defines a Unique Subset of Ligandable Cysteines

发现一种可调控的杂环亲电试剂 4-氯吡唑并吡啶,它定义了可配位半胱氨酸的一个独特子集

Kim, Hong-Rae; Byun, David P; Thakur, Kalyani; Ritchie, Jennifer; Xie, Yixin; Holewinski, Ronald; Suazo, Kiall F; Stevens, Mckayla; Liechty, Hope; Tagirasa, Ravichandra; Jing, Yihang; Andresson, Thorkell; Johnson, Steven M; Yoo, Euna

Strategic career behaviours among hybrid workers: testing a general European model

混合型员工的战略性职业行为:检验一个通用的欧洲模型

Hildred, Kiall; Piteira, Margarida; Cervai, Sara; Pinto, Joana Carneiro