日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The cellular prion protein mediates Tau oligomer‐induced memory impairment in mice

细胞朊病毒蛋白介导小鼠Tau寡聚体诱导的记忆障碍

Lalucque, Hervé; Malagnac, Fabienne; Brun, Sylvain; Kicka, Sébastien; Silar, Philippe; Forloni, Gianluigi; Balducci, Claudia; Orsini, Franca; Cerovic, Milica; Masone, Antonio; Raimondi, Ilaria; Lavigna, Giada; Zucchelli, Chiara; Beeg, Marten; Colombo, Laura; Musco, Giovanna; Gobbi, Marco; Chiesa, Roberto; Fioriti, Luana

Regulation of transforming growth factor-β signaling as a therapeutic approach to treating colorectal cancer

调控转化生长因子-β信号通路作为治疗结直肠癌的一种治疗方法

Maslankova, Jana; Vecurkovska, Ivana; Rabajdova, Miroslava; Katuchova, Jana; Kicka, Milos; Gayova, Michala; Katuch, Vladimir

5-ethyl-2'-deoxyuridine fragilizes Klebsiella pneumoniae outer wall and facilitates intracellular killing by phagocytic cells

5-乙基-2'-脱氧尿苷使肺炎克雷伯菌外壁脆弱化并促进吞噬细胞在细胞内杀死细菌

Estelle Ifrid, Hajer Ouertatani-Sakouhi, Tania Jauslin, Sebastien Kicka, Gianpaolo Chiriano, Christopher F Harrison, Hubert Hilbi, Leonardo Scapozza, Thierry Soldati, Pierre Cosson

Identification of Anti- Mycobacterium and Anti- Legionella Compounds With Potential Distinctive Structural Scaffolds From an HD-PBL Using Phenotypic Screens in Amoebae Host Models

使用变形虫宿主模型中的表型筛选从 HD-PBL 中鉴定具有潜在独特结构支架的抗分枝杆菌和抗军团菌化合物

Nabil Hanna, Sébastien Kicka, Gianpaolo Chiriano, Christopher Harrison, Hajer Ouertatani Sakouhi, Valentin Trofimov, Agata Kranjc, Jahn Nitschke, Marco Pagni, Pierre Cosson, Hubert Hilbi, Leonardo Scapozza, Thierry Soldati

Antimycobacterial drug discovery using Mycobacteria-infected amoebae identifies anti-infectives and new molecular targets

利用感染分枝杆菌的变形虫进行抗分枝杆菌药物发现可确定抗感染药物和新的分子靶点

Valentin Trofimov, Sébastien Kicka, Sabrina Mucaria, Nabil Hanna, Fernando Ramon-Olayo, Laura Vela-Gonzalez Del Peral, Joël Lelièvre, Lluís Ballell, Leonardo Scapozza, Gurdyal S Besra, Jonathan A G Cox, Thierry Soldati

Mycobacterium marinum antagonistically induces an autophagic response while repressing the autophagic flux in a TORC1- and ESX-1-dependent manner

海分枝杆菌以TORC1和ESX-1依赖的方式拮抗性地诱导自噬反应,同时抑制自噬通量。

Cardenal-Muñoz, Elena; Arafah, Sonia; López-Jiménez, Ana Teresa; Kicka, Sébastien; Falaise, Alexandra; Bach, Frauke; Schaad, Olivier; King, Jason S; Hagedorn, Monica; Soldati, Thierry

Open Source Drug Discovery with the Malaria Box Compound Collection for Neglected Diseases and Beyond

利用疟疾化合物库进行开源药物发现,以应对被忽视的热带病及其他疾病

Van Voorhis, Wesley C; Adams, John H; Adelfio, Roberto; Ahyong, Vida; Akabas, Myles H; Alano, Pietro; Alday, Aintzane; Alemán Resto, Yesmalie; Alsibaee, Aishah; Alzualde, Ainhoa; Andrews, Katherine T; Avery, Simon V; Avery, Vicky M; Ayong, Lawrence; Baker, Mark; Baker, Stephen; Ben Mamoun, Choukri; Bhatia, Sangeeta; Bickle, Quentin; Bounaadja, Lotfi; Bowling, Tana; Bosch, Jürgen; Boucher, Lauren E; Boyom, Fabrice F; Brea, Jose; Brennan, Marian; Burton, Audrey; Caffrey, Conor R; Camarda, Grazia; Carrasquilla, Manuela; Carter, Dee; Belen Cassera, Maria; Chih-Chien Cheng, Ken; Chindaudomsate, Worathad; Chubb, Anthony; Colon, Beatrice L; Colón-López, Daisy D; Corbett, Yolanda; Crowther, Gregory J; Cowan, Noemi; D'Alessandro, Sarah; Le Dang, Na; Delves, Michael; DeRisi, Joseph L; Du, Alan Y; Duffy, Sandra; Abd El-Salam El-Sayed, Shimaa; Ferdig, Michael T; Fernández Robledo, José A; Fidock, David A; Florent, Isabelle; Fokou, Patrick V T; Galstian, Ani; Gamo, Francisco Javier; Gokool, Suzanne; Gold, Ben; Golub, Todd; Goldgof, Gregory M; Guha, Rajarshi; Guiguemde, W Armand; Gural, Nil; Guy, R Kiplin; Hansen, Michael A E; Hanson, Kirsten K; Hemphill, Andrew; Hooft van Huijsduijnen, Rob; Horii, Takaaki; Horrocks, Paul; Hughes, Tyler B; Huston, Christopher; Igarashi, Ikuo; Ingram-Sieber, Katrin; Itoe, Maurice A; Jadhav, Ajit; Naranuntarat Jensen, Amornrat; Jensen, Laran T; Jiang, Rays H Y; Kaiser, Annette; Keiser, Jennifer; Ketas, Thomas; Kicka, Sebastien; Kim, Sunyoung; Kirk, Kiaran; Kumar, Vidya P; Kyle, Dennis E; Lafuente, Maria Jose; Landfear, Scott; Lee, Nathan; Lee, Sukjun; Lehane, Adele M; Li, Fengwu; Little, David; Liu, Liqiong; Llinás, Manuel; Loza, Maria I; Lubar, Aristea; Lucantoni, Leonardo; Lucet, Isabelle; Maes, Louis; Mancama, Dalu; Mansour, Nuha R; March, Sandra; McGowan, Sheena; Medina Vera, Iset; Meister, Stephan; Mercer, Luke; Mestres, Jordi; Mfopa, Alvine N; Misra, Raj N; Moon, Seunghyun; Moore, John P; Morais Rodrigues da Costa, Francielly; Müller, Joachim; Muriana, Arantza; Nakazawa Hewitt, Stephen; Nare, Bakela; Nathan, Carl; Narraidoo, Nathalie; Nawaratna, Sujeevi; Ojo, Kayode K; Ortiz, Diana; Panic, Gordana; Papadatos, George; Parapini, Silvia; Patra, Kailash; Pham, Ngoc; Prats, Sarah; Plouffe, David M; Poulsen, Sally-Ann; Pradhan, Anupam; Quevedo, Celia; Quinn, Ronald J; Rice, Christopher A; Abdo Rizk, Mohamed; Ruecker, Andrea; St Onge, Robert; Salgado Ferreira, Rafaela; Samra, Jasmeet; Robinett, Natalie G; Schlecht, Ulrich; Schmitt, Marjorie; Silva Villela, Filipe; Silvestrini, Francesco; Sinden, Robert; Smith, Dennis A; Soldati, Thierry; Spitzmüller, Andreas; Stamm, Serge Maximilian; Sullivan, David J; Sullivan, William; Suresh, Sundari; Suzuki, Brian M; Suzuki, Yo; Swamidass, S Joshua; Taramelli, Donatella; Tchokouaha, Lauve R Y; Theron, Anjo; Thomas, David; Tonissen, Kathryn F; Townson, Simon; Tripathi, Abhai K; Trofimov, Valentin; Udenze, Kenneth O; Ullah, Imran; Vallieres, Cindy; Vigil, Edgar; Vinetz, Joseph M; Voong Vinh, Phat; Vu, Hoan; Watanabe, Nao-Aki; Weatherby, Kate; White, Pamela M; Wilks, Andrew F; Winzeler, Elizabeth A; Wojcik, Edward; Wree, Melanie; Wu, Wesley; Yokoyama, Naoaki; Zollo, Paul H A; Abla, Nada; Blasco, Benjamin; Burrows, Jeremy; Laleu, Benoît; Leroy, Didier; Spangenberg, Thomas; Wells, Timothy; Willis, Paul A

Amoebae-Based Screening Reveals a Novel Family of Compounds Restricting Intracellular Legionella pneumophila

基于变形虫的筛选揭示出一类限制细胞内嗜肺军团菌的新型化合物

Christopher F Harrison, Gianpaolo Chiriano, Ivo Finsel, Christian Manske, Christine Hoffmann, Bernhard Steiner, Agata Kranjc, Ophelie Patthey-Vuadens, Sébastien Kicka, Valentin Trofimov, Hajer Ouertatani-Sakouhi, Thierry Soldati, Leonardo Scapozza, Hubert Hilbi

Establishment and validation of whole-cell based fluorescence assays to identify anti-mycobacterial compounds using the Acanthamoeba castellanii-Mycobacterium marinum host-pathogen system

建立并验证基于全细胞的荧光检测方法,利用卡氏棘阿米巴-海洋分枝杆菌宿主-病原体系统鉴定抗分枝杆菌化合物

Sébastien Kicka, Valentin Trofimov, Christopher Harrison, Hajer Ouertatani-Sakouhi, John McKinney, Leonardo Scapozza, Hubert Hilbi, Pierre Cosson, Thierry Soldati

Exploring anti-bacterial compounds against intracellular Legionella

探索针对细胞内军团菌的抗菌化合物

Christopher F Harrison, Sébastien Kicka, Valentin Trofimov, Kathrin Berschl, Hajer Ouertatani-Sakouhi, Nikolaus Ackermann, Christian Hedberg, Pierre Cosson, Thierry Soldati, Hubert Hilbi