日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Conformational Trajectory of the Molecular Chameleon Grazoprevir From Formulation to Target-Bound

分子变色龙格拉佐普韦从制剂到靶点结合的构象轨迹

Wieske, Lianne H E; Bu, Guanhong; Erdélyi, Máté; Kihlberg, Jan; Gonen, Tamir; Danelius, Emma Rova

Ultra-large virtual screening unveils potent agonists of the neuromodulatory orphan receptor GPR139

超大规模虚拟筛选揭示了神经调节孤儿受体 GPR139 的强效激动剂

Cabeza de Vaca, Israel; Trapkov, Boris; Shen, Ling; Vo, Duy Duc; Zhang, Xiaoqun; Yang, Yunting; Pezeshki, Mitra; Zhang, Xuehan; Bällgren, Frida; Saleh, Aljona; Tarnovskiy, Andrii V; Radchenko, Dmytro S; Moroz, Yurii S; Bräuner-Osborne, Hans; Svenningsson, Per; Kihlberg, Jan; Liu, Zhi-Jie; Hauser, Alexander Sebastian; Carlsson, Jens

Virtual fragment screening for DNA repair inhibitors in vast chemical space.

在广阔的化学空间中对DNA修复抑制剂进行虚拟片段筛选

Luttens Andreas, Vo Duc Duy, Scaletti Emma R, Wiita Elisée, Almlöf Ingrid, Wallner Olov, Davies Jonathan, Košenina Sara, Meng Liuzhen, Long Maeve, Mortusewicz Oliver, Masuyer Geoffrey, Ballante Flavio, Michel Maurice, Homan Evert, Scobie Martin, Kalderén Christina, Warpman Berglund Ulrika, Tarnovskiy Andrii V, Radchenko Dmytro S, Moroz Yurii S, Kihlberg Jan, Stenmark Pål, Helleday Thomas, Carlsson Jens

Tolerogenic antigen-specific vaccine induces VISTA-enriched regulatory T cells and protects against arthritis in DRB1∗04:01 mice

耐受性抗原特异性疫苗可诱导富含 VISTA 的调节性 T 细胞,并保护 DRB1∗04:01 小鼠免受关节炎侵害。

Romero-Castillo, Laura; Pandey, Rajan Kumar; Xu, Bingze; Beusch, Christian M; Oliveira-Coelho, Ana; Zeqiraj, Kejsi; Svensson, Carolin; Xu, Zhongwei; Luo, Huqiao; Sareila, Outi; Sabatier, Pierre; Ge, Changrong; Cheng, Lei; Urbonaviciute, Vilma; Krämer, Alexander; Lindgren, Cecilia; Haag, Sabrina; Viljanen, Johan; Zubarev, Roman A; Kihlberg, Jan; Linusson, Anna; Burkhardt, Harald; Holmdahl, Rikard

Structure-based discovery of positive allosteric modulators of the A(1) adenosine receptor

基于结构的A(1)腺苷受体正向变构调节剂的发现

Nguyen, Anh T N; Panel, Nicolas; Vo, Duc Duy; Thai, Bui San; Chia, Ling Yeong; Lu, Cam Sinh; Hellyer, Shane D; Langiu, Monica; Jörg, Manuela; Gregory, Karen J; Kihlberg, Jan; White, Paul J; Scammells, Peter J; Christopoulos, Arthur; Carlsson, Jens; May, Lauren T

A membrane permeability database for nonpeptidic macrocycles

非肽类大环化合物的膜渗透性数据库

Feng, Qiushi; De Chavez, Danjo; Kihlberg, Jan; Poongavanam, Vasanthanathan

Autoantibodies to joint-related peptides as predictive markers in early rheumatoid arthritis

针对关节相关肽的自身抗体作为早期类风湿性关节炎的预测标志物

Leu Agelii, Monica; Sareila, Outi; Lönnblom, Erik; Cheng, Lei; Forslind, Kristina; Hafström, Ingiäld; Andersson, Maria L E; Kastbom, Alf; Sjöwall, Christopher; Jacobsson, Lennart T H; Kihlberg, Jan; Holmdahl, Rikard; Gjertsson, Inger

Linker-Determined Folding and Hydrophobic Interactions Explain a Major Difference in PROTAC Cell Permeability

连接基团决定的折叠和疏水相互作用解释了PROTAC细胞渗透性的主要差异

Poongavanam, Vasanthanathan; Peintner, Stefan; Abeje, Yordanos; Kölling, Florian; Meibom, Daniel; Erdelyi, Mate; Kihlberg, Jan

Correction: Antigen-presenting autoreactive B cells activate regulatory T cells and suppress autoimmune arthritis in mice

更正:抗原呈递自身反应性B细胞激活调节性T细胞并抑制小鼠自身免疫性关节炎。

Aoun, Mike; Coelho, Ana; Krämer, Alexander; Saxena, Amit; Sabatier, Pierre; Beusch, Christian Michel; Lönnblom, Erik; Geng, Manman; Do, Nhu-Nguyen; Xu, Zhongwei; Zhang, Jingdian; He, Yibo; Castillo, Laura Romero; Abolhassani, Hassan; Xu, Bingze; Viljanen, Johan; Rorbach, Joanna; Lahore, Gonzalo Fernandez; Gjertsson, Inger; Kastbom, Alf; Sjöwall, Christopher; Kihlberg, Jan; Zubarev, Roman A; Burkhardt, Harald; Holmdahl, Rikard

Macrocycles in Drug Discovery─Learning from the Past for the Future

药物发现中的大环化合物——从过去汲取经验,展望未来

Garcia Jimenez, Diego; Poongavanam, Vasanthanathan; Kihlberg, Jan