日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

CELF1 is a non-canonical eIF4E binding protein that promotes translation of epithelial-mesenchymal transition effector mRNAs

CELF1是一种非经典的eIF4E结合蛋白,可促进上皮-间质转化效应mRNA的翻译。

Chaudhury, Arindam; Kongchan, Natee; Massey, Shebna A; Sharma, Rajesh; Pal, Rituraj; Zhao, Na; Tsoi, Phoebe; Zhu, Yingmin; Olokpa, Emuejevoke; Mao, Sufeng; Del Rincon, Sonia; Reineke, Lucas C; Lloyd, Richard E; Sardiello, Marco; Rosen, Jeffrey M; Kim, Choel; Ferreon, Josephine C; Neilson, Joel R

Fyn-Saracatinib Complex Structure Reveals an Active State-like Conformation

Fyn-Saracatinib复合物结构揭示了一种活性状态样构象

Ta, Hai Minh; Sankaran, Banumathi; Roush, Eric D; Ferreon, Josephine C; Ferreon, Allan Chris M; Kim, Choel

A divergent cyclic nucleotide binding protein promotes Plasmodium ookinete infection of the mosquito.

一种不同的环核苷酸结合蛋白促进疟原虫卵动子感染蚊子

Kwecka Dominika, Wang Zhishuo, Eigminas Edvardas, Liu Lijia, Regan Jennifer C, Kim Choel, Philip Nisha

Reversible male contraception by targeted inhibition of serine/threonine kinase 33

通过靶向抑制丝氨酸/苏氨酸激酶33实现可逆性男性避孕

Ku, Angela F; Sharma, Kiran L; Ta, Hai Minh; Sutton, Courtney M; Bohren, Kurt M; Wang, Yong; Chamakuri, Srinivas; Chen, Ruihong; Hakenjos, John M; Jimmidi, Ravikumar; Kent, Katarzyna; Li, Feng; Li, Jian-Yuan; Ma, Lang; Madasu, Chandrashekhar; Palaniappan, Murugesan; Palmer, Stephen S; Qin, Xuan; Robers, Matthew B; Sankaran, Banumathi; Tan, Zhi; Vasquez, Yasmin M; Wang, Jian; Wilkinson, Jennifer; Yu, Zhifeng; Ye, Qiuji; Young, Damian W; Teng, Mingxing; Kim, Choel; Matzuk, Martin M

Discovery of highly potent and ALK2/ALK1 selective kinase inhibitors using DNA-encoded chemistry technology.

利用DNA编码化学技术发现高效且对ALK2/ALK1具有选择性的激酶抑制剂

Jimmidi Ravikumar, Monsivais Diana, Ta Hai Minh, Sharma Kiran L, Bohren Kurt M, Chamakuri Srinivas, Liao Zian, Li Feng, Hakenjos John M, Li Jian-Yuan, Mishina Yuji, Pan Haichun, Qin Xuan, Robers Matthew B, Sankaran Banumathi, Tan Zhi, Tang Suni, Vasquez Yasmin M, Wilkinson Jennifer, Young Damian W, Palmer Stephen S, MacKenzie Kevin R, Kim Choel, Matzuk Martin M

Stereospecific NANOG PEST Stabilization by Pin1

Pin1 的立体特异性 NANOG PEST 稳定化

Ferreon, Josephine C; Ta, Hai Minh; Yun, Hyosuk; Choi, Kyoung-Jae; Quan, My Diem; Tsoi, Phoebe S; Kim, Choel; Lee, Chul Won; Ferreon, Allan Chris M

Discovery of potent BET bromodomain 1 stereoselective inhibitors using DNA-encoded chemical library selections

利用DNA编码化学库筛选发现强效BET溴结构域1立体选择性抑制剂

Modukuri, Ram K; Yu, Zhifeng; Tan, Zhi; Ta, Hai Minh; Ucisik, Melek Nihan; Jin, Zhuang; Anglin, Justin L; Sharma, Kiran L; Nyshadham, Pranavanand; Li, Feng; Riehle, Kevin; Faver, John C; Duong, Kevin; Nagarajan, Sureshbabu; Simmons, Nicholas; Palmer, Stephen S; Teng, Mingxing; Young, Damian W; Yi, Joanna S; Kim, Choel; Matzuk, Martin M

Discovery and characterization of bromodomain 2-specific inhibitors of BRDT

BRDT溴结构域2特异性抑制剂的发现与表征

Yu, Zhifeng; Ku, Angela F; Anglin, Justin L; Sharma, Rajesh; Ucisik, Melek Nihan; Faver, John C; Li, Feng; Nyshadham, Pranavanand; Simmons, Nicholas; Sharma, Kiran L; Nagarajan, Sureshbabu; Riehle, Kevin; Kaur, Gundeep; Sankaran, Banumathi; Storl-Desmond, Marta; Palmer, Stephen S; Young, Damian W; Kim, Choel; Matzuk, Martin M

Cyclic nucleotide selectivity of protein kinase G isozymes

蛋白激酶G同工酶对环核苷酸的选择性

Kim, Choel; Sharma, Rajesh

Correction to: Crystal structure of PKG Iβ holoenzyme reveals a trans‑inhibiting dimer assembly

更正:PKG Iβ 全酶的晶体结构揭示了一种反式抑制二聚体组装体

Kim, Choel; Sharma, Rajesh; Casteel, Darren E