日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Corrigendum to "A novel FGFR1 inhibitor CYY292 suppresses tumor progression, invasion, and metastasis of glioblastoma by inhibiting the Akt/GSK3β/snail signaling axis" [Genes & Diseases 11 (2024) 479-494]

对“一种新型 FGFR1 抑制剂 CYY292 通过抑制 Akt/GSK3β/snail 信号轴抑制胶质母细胞瘤的肿瘤进展、侵袭和转移”的更正 [Genes & Diseases 11 (2024) 479-494]

Bi, Yanran; Zheng, Ruiling; Hu, Jiahao; Shi, Ruiqing; Shi, Junfeng; Wang, Yutao; Wang, Peng; Jiang, Wenyi; Kim, Gyudong; Liu, Zhiguo; Li, Xiaokun; Lin, Li

In Silico Discovery of 5'-Modified 7-Deoxy-7-ethynyl-4'-thioadenosine as a HASPIN Inhibitor and Its Synergistic Anticancer Effect with the PLK1 Inhibitor

利用计算机模拟发现 5'-修饰的 7-脱氧-7-乙炔基-4'-硫代腺苷作为 HASPIN 抑制剂及其与 PLK1 抑制剂的协同抗癌作用

Kwon, Eun-Ji; Mashelkar, Karishma K; Seo, Juhee; Shin, Yoon-Ze; Sung, Kisu; Jang, Sung Chul; Cheon, Sang Won; Lee, Haeseung; Lee, Hyuk Woo; Kim, Gyudong; Han, Byung Woo; Lee, Sang Kook; Jeong, Lak Shin; Cha, Hyuk-Jin

Structure-Activity Relationship of Truncated 2,8-Disubstituted-Adenosine Derivatives as Dual A(2A)/A(3) Adenosine Receptor Antagonists and Their Cancer Immunotherapeutic Activity.

截短的 2,8-二取代腺苷衍生物作为双重 A(2A)/A(3) 腺苷受体拮抗剂的构效关系及其癌症免疫治疗活性

Kim Gibae, Hou Xiyan, Byun Woong Sub, Kim Gyudong, Jarhad Dnyandev B, Lee Grim, Hyun Young Eum, Yu Jinha, Lee Chang Soo, Qu Shuhao, Warnick Eugene, Gao Zhan-Guo, Kim Ji Yong, Ji Seunghee, Shin Hyunwoo, Choi Jong-Ryoul, Jacobson Kenneth A, Lee Hyuk Woo, Lee Sang Kook, Jeong Lak Shin

Synthesis of 9-Cinnamyl-9H-purine Derivatives as Novel TLR4/MyD88/NF-κB Pathway Inhibitors for Anti-inflammatory Effects

合成9-肉桂基-9H-嘌呤衍生物作为新型TLR4/MyD88/NF-κB通路抑制剂用于抗炎作用

Pham, Linh; Jiang, Rui; Liu, Zijing; Nguyen, Mai; Nguyen, Yen; Gong, Yue; Bi, Yanran; Kim, Hong-Rae; Kim, Young Ran; Kim, Gyudong

Novel innovative computer-based test (Inno-CBT) item types for national licensing examinations for health care professionals

针对医疗保健专业人员国家执照考试的新型创新型计算机辅助测试 (Inno-CBT) 题型

Chun, Kwang-Hoon; Jin, Hye Kyung; Yoon, Jeong-Hyun; Kim, Myeong Gyu; Choi, Kyung Hee; Kim, Eunyoung; Kim, Hyunah; Kim, Jin-Ki; Kim, Gyudong; Kim, Kyungim; Lee, Ju-Yeun; Chung, Eun Kyoung; Lee, Young Sook; Rhie, Sandy Jeong

Design, Synthesis, and Biological Activity of l-1'-Homologated Adenosine Derivatives

l-1'-同系腺苷衍生物的设计、合成及生物活性

Nguyen, Mai; An, Seungchan; Nguyen, Yen; Hyun, Young Eum; Choi, Hongseok; Pham, Linh; Kim, Jung-Ae; Noh, Minsoo; Kim, Gyudong; Jeong, Lak Shin

Discovery and Structure-Activity Relationships of Novel Template, Truncated 1'-Homologated Adenosine Derivatives as Pure Dual PPARγ/δ Modulators.

新型模板截短的 1'-同系腺苷衍生物作为纯粹的双重 PPARα/α 调节剂的发现和构效关系

An Seungchan, Kim Gyudong, Kim Hyun Jin, Ahn Sungjin, Kim Hyun Young, Ko Hyejin, Hyun Young Eum, Nguyen Mai, Jeong Juri, Liu Zijing, Han Jinhe, Choi Hongseok, Yu Jinha, Kim Ji Won, Lee Hyuk Woo, Jacobson Kenneth A, Cho Won Jea, Kim Young-Mi, Kang Keon Wook, Noh Minsoo, Jeong Lak Shin

6'-β-Fluoro-Homoaristeromycin and 6'-Fluoro-Homoneplanocin A Are Potent Inhibitors of Chikungunya Virus Replication through Their Direct Effect on Viral Nonstructural Protein 1

6'-β-氟-高阿利斯特霉素和6'-氟-高诺霉素A通过直接作用于病毒非结构蛋白1,成为基孔肯雅病毒复制的强效抑制剂。

Kovacikova, Kristina; Morren, Bas M; Tas, Ali; Albulescu, Irina C; van Rijswijk, Robin; Jarhad, Dnyandev B; Shin, Young Sup; Jang, Min Hwan; Kim, Gyudong; Lee, Hyuk Woo; Jeong, Lak Shin; Snijder, Eric J; van Hemert, Martijn J

Development of a Potent Brain-Penetrant EGFR Tyrosine Kinase Inhibitor against Malignant Brain Tumors

开发一种强效的、可穿透血脑屏障的EGFR酪氨酸激酶抑制剂,用于治疗恶性脑肿瘤

Tsang, Jonathan E; Urner, Lorenz M; Kim, Gyudong; Chow, Kingsley; Baufeld, Lynn; Faull, Kym; Cloughesy, Timothy F; Clark, Peter M; Jung, Michael E; Nathanson, David A

Design, Synthesis, and Anti-RNA Virus Activity of 6'-Fluorinated-Aristeromycin Analogues

6'-氟代阿利司霉素类似物的设计、合成及抗RNA病毒活性

Yoon, Ji-Seong; Kim, Gyudong; Jarhad, Dnyandev B; Kim, Hong-Rae; Shin, Young-Sup; Qu, Shuhao; Sahu, Pramod K; Kim, Hea Ok; Lee, Hyuk Woo; Wang, Su Bin; Kong, Yun Jeong; Chang, Tong-Shin; Ogando, Natacha S; Kovacikova, Kristina; Snijder, Eric J; Posthuma, Clara C; van Hemert, Martijn J; Jeong, Lak Shin