日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, Synthesis, and Anti-RNA Virus Activity of 6'-Fluorinated-Aristeromycin Analogues

6'-氟代阿利司霉素类似物的设计、合成及抗RNA病毒活性

Yoon, Ji-Seong; Kim, Gyudong; Jarhad, Dnyandev B; Kim, Hong-Rae; Shin, Young-Sup; Qu, Shuhao; Sahu, Pramod K; Kim, Hea Ok; Lee, Hyuk Woo; Wang, Su Bin; Kong, Yun Jeong; Chang, Tong-Shin; Ogando, Natacha S; Kovacikova, Kristina; Snijder, Eric J; Posthuma, Clara C; van Hemert, Martijn J; Jeong, Lak Shin

Synthesis and anti-renal fibrosis activity of conformationally locked truncated 2-hexynyl-N(6)-substituted-(N)-methanocarba-nucleosides as A3 adenosine receptor antagonists and partial agonists.

构象锁定截短的 2-己炔基-N(6)-取代-(N)-甲氧基碳核苷作为 A3 腺苷受体拮抗剂和部分激动剂的合成及其抗肾纤维化活性

Nayak Akshata, Chandra Girish, Hwang Inah, Kim Kyunglim, Hou Xiyan, Kim Hea Ok, Sahu Pramod K, Roy Kuldeep K, Yoo Jakyung, Lee Yoonji, Cui Minghua, Choi Sun, Moss Steven M, Phan Khai, Gao Zhan-Guo, Ha Hunjoo, Jacobson Kenneth A, Jeong Lak Shin

Structure-activity relationships of 2-chloro-N6-substituted-4'-thioadenosine-5'-N,N-dialkyluronamides as human A3 adenosine receptor antagonists

2-氯-N6-取代-4'-硫代腺苷-5'-N,N-二烷基糖醛酸酰胺作为人A3腺苷受体拮抗剂的构效关系

Jeong, Lak Shin; Lee, Hyuk Woo; Kim, Hea Ok; Tosh, Dilip K; Pal, Shantanu; Choi, Won Jun; Gao, Zhan-Guo; Patel, Amit R; Williams, Wanda; Jacobson, Kenneth A; Kim, Hee-Doo

Probing the binding site of the A1 adenosine receptor reengineered for orthogonal recognition by tailored nucleosides

利用定制核苷探测经改造以实现正交识别的A1腺苷受体的结合位点

Palaniappan, Krishnan K; Gao, Zhan-Guo; Ivanov, Andrei A; Greaves, Rebecca; Adachi, Hayamitsu; Besada, Pedro; Kim, Hea Ok; Kim, Ae Yil; Choe, Seung Ah; Jeong, Lak Shin; Jacobson, Kenneth A

Conversion of A3 adenosine receptor agonists into selective antagonists by modification of the 5'-ribofuran-uronamide moiety

通过修饰 5'-核糖呋喃-尿酰胺部分将 A3 腺苷受体激动剂转化为选择性拮抗剂

Gao, Zhan-Guo; Joshi, Bhalchandra V; Klutz, Athena M; Kim, Soo-Kyung; Lee, Hyuk Woo; Kim, Hea Ok; Jeong, Lak Shin; Jacobson, Kenneth A

Design and synthesis of 3'-ureidoadenosine-5'-uronamides: effects of the 3'-ureido group on binding to the A3 adenosine receptor

3'-脲基腺苷-5'-尿酰胺的设计与合成:3'-脲基对与A3腺苷受体结合的影响

Jeong, Lak Shin; Kim, Myong Jung; Kim, Hea Ok; Gao, Zhan-Guo; Kim, Soo-Kyung; Jacobson, Kenneth A; Chun, Moon Woo

Design, synthesis and binding affinity of 3'-fluoro analogues of Cl-IB-MECA as adenosine A3 receptor ligands

Cl-IB-MECA 的 3'-氟类似物作为腺苷 A3 受体配体的设计、合成和结合亲和力

Lim, Moo Hong; Kim, Hea Ok; Moon, Hyung Ryong; Lee, Seung Jin; Chun, Moon Woo; Gao, Zhan-Guo; Melman, Neli; Jacobson, Kenneth A; Kim, Joong Hyup; Jeong, Lak Shin

Activation and Desensitization of Rat A(3)-Adenosine Receptors by Selective Adenosine Derivatives and Xanthine-7-Ribosides

选择性腺苷衍生物和黄嘌呤-7-核苷对大鼠A(3)-腺苷受体的激活和脱敏作用

Park, Kyung-Sun; Hoffmann, Carsten; Kim, Hea Ok; Padgett, William L; Daly, John W; Brambilla, Roberta; Motta, Cristina; Abbracchio, Maria P; Jacobson, Kenneth A