Discovery of a Potent and Selective Protein Arginine Methyltransferase 5 (PRMT5) PROTAC Degrader.
发现一种高效且选择性的蛋白质精氨酸甲基转移酶 5 (PRMT5) PROTAC 降解剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c00198
Zhong Yue, Kim Huensuk, Qian Chao, Xie Ling, Chen Xian, Xiong Yan, Hu Jacqueline, Chen Matthew, Guccione Ernesto, Shen Yudao, Jin Jian