日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of KLHL12 Ligands Using Fragment-Based Methods

利用基于片段的方法鉴定KLHL12配体

Waterson, Alex G; Vadukoot, Anish; Jana, Somnath; Cui, Jianwen; Luong, Kelvin; Rietz, Tyson A; Madrigal-Carrillo, Ezequiel Alejandro; Lehmann, Brian D; Sensintaffar, John L; Zhao, Bin; Amporndanai, Kangsa; Petros, Zoe A; Scaggs, William Rush; Chacon Simon, Selena; Vekariya, Rakesh H; Kim, Kwangho; Thangaraj, Manikandan; Christov, Plamen P; South, Taylor M; Sai, Jiqing; Thiruvaipati, Anusha; Schmidt, Charles R; Eells, Rebecca; Moore, William J; Olejniczak, Edward T; Phan, Jason; Fesik, Stephen W

Discovery of Macrocyclic Myeloid Cell Leukemia 1 (Mcl-1) Inhibitors that Demonstrate Potent Cellular Efficacy and In Vivo Activity in a Mouse Solid Tumor Xenograft Model

发现具有强效细胞活性和在小鼠实体瘤异种移植模型中体内活性的巨环髓系细胞白血病1 (Mcl-1) 抑制剂

Tarr, James C; Jeon, Kyuok; Veerasamy, Nagarathanam; Aichinger, Martin; Salovich, James M; Zhao, Bin; Sensintaffar, John L; Arnhof, Heribert; Wunberg, Tobias; Sgubin, Danielle; Arnold, Allison; Vekariya, Rakesh H; Christov, Plamen P; Kim, Kwangho; Fuchs, Julian Emanuel; Karier, Pol; Betzemeier, Bodo; Van Meveren, Mayme; Miriyala, Nagaraju; Olejniczak, Edward T; Engelhardt, Harald; Lee, Taekyu; McConnell, Darryl; Fesik, Stephen W

Time-Resolved Analysis of Protein-Protein Ensembles Using a Destabilizing Domain to Map Dynamic Interactions of SARS-CoV-2 nsp15

利用去稳定结构域对蛋白质-蛋白质复合物进行时间分辨分析,以绘制SARS-CoV-2 nsp15的动态相互作用图谱

Cameron, Crissey; Clark, R Mason; Metts, Adam M; Jiang, Runze M; Scaggs, Toya D; Kim, Kwangho; Sulikowski, Gary A; Plate, Lars

Photoaffinity Ligand of Cystic Fibrosis Corrector VX-445 Identifies SCCPDH as an Off-Target.

囊性纤维化矫正剂 VX-445 的光亲和配体鉴定出 SCCPDH 为脱靶靶点

Kim Minsoo, Kim Kwangho, Lee Jesun, Barny Lea A, Scaggs Toya D, Romaine Ian M, Jeon KyuOk, Codreanu Simona G, Sherrod Stacy D, McLean John A, Naren Anjaparavanda P, Sulikowski Gary A, Plate Lars

Ultrasound-Guided vs Non-Guided Pharmacopuncture for Cervical Myofascial Pain Syndrome: A Multi-Center Prospective Comparative Study Protocol

超声引导与非引导下药针治疗颈椎肌筋膜疼痛综合征:一项多中心前瞻性比较研究方案

Kim, Kwangho; Song, Juhwan; Chu, Hongmin; Kwon, Robin; Park, Seongjun; Kwon, Junhui; Hong, Hyeon Joon; Lee, Youngyun; Kwon, Sanghyuk; Kang, Kyungho; Leem, Jungtae; Kim, Cheol-Hyun

Effectiveness and Safety of Portable Ultrasound-Guided Pharmacopuncture for Cervical Myofascial Pain Syndrome: A Prospective Observational Multi-Center Study

便携式超声引导药针疗法治疗颈椎肌筋膜疼痛综合征的有效性和安全性:一项前瞻性观察性多中心研究

Kwon, Robin; Kim, Kwangho; Lee, Young-Ung; Kwon, Sanghyuk; Song, Juhwan; Park, Seongjun; Kwon, Junhui; Hong, Hyeon Joon; Lee, Youngyun; Leem, Jungtae; Chu, Hongmin; Kim, Cheol-Hyun

Response to Korean medicine with acupotomy in patients with cognitive impairment in primary care: A multicenter registry protocol

基层医疗中认知障碍患者接受针灸治疗的疗效:一项多中心注册研究方案

Jun, Hyungsun; Ryu, Myungseok; Chae, Hyocheong; Chu, Hongmin; Kim, Kwangho; Lee, Do-Eun; Jin, Hanbit; Joo, Sungjun; Park, Dasol; Leem, Jungtae; Kang, Hyung Won

Positive regulation of cell proliferation by the miR-1290-EHHADH axis in hepatocellular carcinoma

miR-1290-EHHADH轴在肝细胞癌中对细胞增殖的正向调控

Lee, Jinkwon; Kim, Gyeonghwa; Han, Tae-Su; Jung, Eunsun; Son, Taesang; Kim, Kwangho; Kwon, Kiyoon; Roh, Yuna; Ryu, Tae Young; Tae, In Hwan; Kang, Yunsang; Lee, Byungheon; Lee, Yu Rim; Park, Soo Young; Tak, Won Young; Kim, Dae-Soo; Son, Mi-Young; Hur, Keun; Cho, Hyun-Soo

Epigenetic alterations of TP53INP1 by EHMT2 regulate the cell cycle in gastric cancer

EHMT2介导的TP53INP1表观遗传修饰调控胃癌细胞周期

Ryu, Tae Young; Tae, In Hwan; Han, Tae-Su; Lee, Jinkwon; Kim, Kwangho; Kang, Yunsang; Kim, Solbi; Lee, Hyo Jin; Jung, Cho-Rok; Lim, Jung Hwa; Kim, Dae-Soo; Son, Mi-Young; Cho, Hyun-Soo

The cannabinoid CB(2) receptor positive allosteric modulator EC21a exhibits complicated pharmacology in vitro

大麻素CB(2)受体正向变构调节剂EC21a在体外表现出复杂的药理学特性。

Qi, Aidong; Han, Xueqing; Quitalig, Marc; Wu, Jessica; Christov, Plamen P; Jeon, KyuOk; Jana, Somnath; Kim, Kwangho; Engers, Darren W; Lindsley, Craig W; Rodriguez, Alice L; Niswender, Colleen M