Anti-tumor activity of new orally bioavailable 2-amino-5-(thiophen-2-yl)benzamide-series histone deacetylase inhibitors, possessing an aqueous soluble functional group as a surface recognition domain
具有水溶性官能团作为表面识别域的新型口服生物可利用 2-氨基-5-(噻吩-2-基)苯甲酰胺系列组蛋白去乙酰化酶抑制剂的抗肿瘤活性
期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.5
doi:10.1016/j.bmcl.2012.01.053
Yoshiyuki Hirata, Masahiko Hirata, Yasuyuki Kawaratani, Makio Shibano, Masahiko Taniguchi, Masahide Yasuda, Yoshiro Ohmomo, Yasuo Nagaoka, Kimiye Baba, Shinichi Uesato