日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Highly specific Immunoproteasome inhibitor M3258 induces proteotoxic stress and apoptosis in KMT2A::AFF1 driven acute lymphoblastic leukemia.

高特异性免疫蛋白酶体抑制剂 M3258 可诱导 KMT2A::AFF1 驱动的急性淋巴细胞白血病中的蛋白毒性应激和细胞凋亡

Jenkins Tyler W, Fitzgerald Jacquelyn Elise, Park Jieun, Wilson Addison M, Berry Kristy L, Wong Keith S, Houry Walid A, Lee Irene, Maksimenko Andrey V, Panizzi Peter R, Maxuitenko Yulia Y, Loop Matthew Shane, Mitra Amit K, Kisselev Alexei F

Early recovery of proteasome activity in cells pulse-treated with proteasome inhibitors is independent of DDI2

用蛋白酶体抑制剂脉冲处理的细胞中蛋白酶体活性的早期恢复与DDI2无关。

Ibtisam, Ibtisam; Kisselev, Alexei F

Site-Specific Proteasome Inhibitors

位点特异性蛋白酶体抑制剂

Kisselev, Alexei F

DNA-Histone Cross-Links: Formation and Repair

DNA-组蛋白交联:形成与修复

Pachva, Manideep C; Kisselev, Alexei F; Matkarimov, Bakhyt T; Saparbaev, Murat; Groisman, Regina

Structure-Based Design of Fluorogenic Substrates Selective for Human Proteasome Subunits

基于结构的、对人蛋白酶体亚基具有选择性的荧光底物设计

Maurits, Elmer; Degeling, Christian G; Kisselev, Alexei F; Florea, Bogdan I; Overkleeft, Herman S

Structure-Based Design of Inhibitors Selective for Human Proteasome β2c or β2i Subunits

基于结构的、选择性抑制人蛋白酶体β2c或β2i亚基的抑制剂设计

Xin, Bo-Tao; Huber, Eva M; de Bruin, Gerjan; Heinemeyer, Wolfgang; Maurits, Elmer; Espinal, Christofer; Du, Yimeng; Janssens, Marissa; Weyburne, Emily S; Kisselev, Alexei F; Florea, Bogdan I; Driessen, Christoph; van der Marel, Gijsbert A; Groll, Michael; Overkleeft, Herman S

The novel β2-selective proteasome inhibitor LU-102 synergizes with bortezomib and carfilzomib to overcome proteasome inhibitor resistance of myeloma cells

新型β2选择性蛋白酶体抑制剂LU-102与硼替佐米和卡非佐米协同作用,可克服骨髓瘤细胞对蛋白酶体抑制剂的耐药性。

Kraus, Marianne; Bader, Juergen; Geurink, Paul P; Weyburne, Emily S; Mirabella, Anne C; Silzle, Tobias; Shabaneh, Tamer B; van der Linden, Wouter A; de Bruin, Gerjan; Haile, Sarah R; van Rooden, Eva; Appenzeller, Christina; Li, Nan; Kisselev, Alexei F; Overkleeft, Herman; Driessen, Christoph

The novel β2-selective proteasome inhibitor LU-102 decreases phosphorylation of I kappa B and induces highly synergistic cytotoxicity in combination with ibrutinib in multiple myeloma cells

新型β2选择性蛋白酶体抑制剂LU-102可降低IκB的磷酸化水平,并与伊布替尼联合使用时在多发性骨髓瘤细胞中产生高度协同的细胞毒性。

Kraus, Johannes; Kraus, Marianne; Liu, Nora; Besse, Lenka; Bader, Jürgen; Geurink, Paul P; de Bruin, Gerjan; Kisselev, Alexei F; Overkleeft, Herman; Driessen, Christoph

Proteasome inhibitors: an expanding army attacking a unique target

蛋白酶体抑制剂:一支不断壮大的军队,攻击一个独特的靶点

Kisselev, Alexei F; van der Linden, Wouter A; Overkleeft, Herman S

Specific cell-permeable inhibitor of proteasome trypsin-like sites selectively sensitizes myeloma cells to bortezomib and carfilzomib

特异性细胞渗透性蛋白酶体胰蛋白酶样位点抑制剂可选择性地增强骨髓瘤细胞对硼替佐米和卡非佐米的敏感性。

Mirabella, Anne C; Pletnev, Alexandre A; Downey, Sondra L; Florea, Bogdan I; Shabaneh, Tamer B; Britton, Matthew; Verdoes, Martijn; Filippov, Dmitri V; Overkleeft, Herman S; Kisselev, Alexei F