日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Covalent inhibitors of the PI3Kα RAS binding domain impair tumor growth driven by RAS and HER2

PI3Kα RAS结合域的共价抑制剂可抑制RAS和HER2驱动的肿瘤生长。

Klebba, Joseph E; Roy, Nilotpal; Bernard, Steffen M; Grabow, Stephanie; Hoffman, Melissa A; Miao, Hui; Tamiya, Junko; Wang, Jinwei; Berry, Cynthia; Esparza-Oros, Antonio; Lin, Richard; Liu, Yongsheng; Pariollaud, Marie; Parker, Holly; Mochalkin, Igor; Rana, Sareena; Snead, Aaron N; Walton, Eric J; Wyrick, Taylor E; Aitichson, Erick; Bedke, Karl; Brannon, Jacyln C; Chick, Joel M; Hee, Kenneth; Horning, Benjamin D; Ismail, Mohamed; Lamb, Kelsey N; Lin, Wei; Lu, Justine; Pastuszka, Martha K; Pollock, Jonathan; Sigler, John J; Tomaschko, Mona; Tran, Eileen; Yue, Chanyu; Kinsella, Todd M; Molina-Arcas, Miriam; Cook, Brian N; Simon, Gabriel M; Weinstein, David S; Downward, Julian; Patricelli, Matthew P

Covalent inhibitors of the RAS binding domain of PI3Kα impair tumor growth driven by RAS and HER2

PI3Kα RAS结合域的共价抑制剂可抑制RAS和HER2驱动的肿瘤生长。

Klebba, Joseph E; Roy, Nilotpal; Bernard, Steffen M; Grabow, Stephanie; Hoffman, Melissa A; Miao, Hui; Tamiya, Junko; Wang, Jinwei; Berry, Cynthia; Esparza-Oros, Antonio; Lin, Richard; Liu, Yongsheng; Pariollaud, Marie; Parker, Holly; Mochalkin, Igor; Rana, Sareena; Snead, Aaron N; Walton, Eric J; Wyrick, Taylor E; Aitichson, Erick; Bedke, Karl; Brannon, Jacyln C; Chick, Joel M; Hee, Kenneth; Horning, Benjamin D; Ismail, Mohamed; Lamb, Kelsey N; Lin, Wei; Metzger, Justine; Pastuszka, Martha K; Pollock, Jonathan; Sigler, John J; Tomaschko, Mona; Tran, Eileen; Kinsella, Todd M; Molina-Arcas, Miriam; Simon, Gabriel M; Weinstein, David S; Downward, Julian; Patricelli, Matthew P

Polo-like kinase 4 autodestructs by generating its Slimb-binding phosphodegron

Polo样激酶4通过生成其Slimb结合磷酸降解子而发生自毁。

Klebba, Joseph E; Buster, Daniel W; Nguyen, Annie L; Swatkoski, Stephen; Gucek, Marjan; Rusan, Nasser M; Rogers, Gregory C

SCFSlimb ubiquitin ligase suppresses condensin II-mediated nuclear reorganization by degrading Cap-H2.

SCFSlimb 泛素连接酶通过降解 Cap-H2 来抑制凝聚素 II 介导的核重组

Buster Daniel W, Daniel Scott G, Nguyen Huy Q, Windler Sarah L, Skwarek Lara C, Peterson Maureen, Roberts Meredith, Meserve Joy H, Hartl Tom, Klebba Joseph E, Bilder David, Bosco Giovanni, Rogers Gregory C

Preparation of Drosophila S2 cells for light microscopy

制备用于光学显微镜观察的果蝇S2细胞

Buster, Daniel W; Nye, Jonathan; Klebba, Joseph E; Rogers, Gregory C

FepA- and TonB-dependent bacteriophage H8: receptor binding and genomic sequence.

依赖 FepA 和 TonB 的噬菌体 H8:受体结合和基因组序列

Rabsch Wolfgang, Ma Li, Wiley Graham, Najar Fares Z, Kaserer Wallace, Schuerch Daniel W, Klebba Joseph E, Roe Bruce A, Laverde Gomez Jenny A, Schallmey Marcus, Newton Salete M C, Klebba Phillip E