日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A clinical-stage oncology compound selectively targets drug-resistant cancers

一种处于临床阶段的肿瘤化合物可选择性地靶向耐药性癌症。

Long, Kaitlin; Bhattacharjee, Debanjan; Newman-Stonebraker, Samuel H; Suhr, Simon; Mercado, Brandon Q; Scheib, Emily; Tighe, Anthony; Romero, Luciano; Thompson, Sarah L; Sausville, Erin L; John, Kristen M; Julian, Linda; Mishra, Sanat; Klingbeil, Olaf; Gupta, Punya; Bhatt, Uditi; Gao, Allen C; Ricardo, Sara; Vakoc, Christopher R; Bornhauser, Beat C; Corsello, Steven M; Taylor, Stephen S; Chen, Jue; Holland, Patrick L; Sheltzer, Jason M

KLF5 enables dichotomous lineage programs in pancreatic cancer via the AAA+ ATPase coactivators RUVBL1 and RUVBL2

KLF5 通过 AAA+ ATPase 共激活因子 RUVBL1 和 RUVBL2 激活胰腺癌中的二分谱系程序。

Cunniff, Patrick J; Sivetz, Nicole; Skopelitis, Damianos; Klingbeil, Olaf; Toobian, Daniel; Maia-Silva, Diogo; Egeblad, Mikala; Vakoc, Christopher R

Dietary pro-oxidant therapy by a vitamin K precursor targets PI 3-kinase VPS34 function.

通过维生素 K 前体进行膳食促氧化疗法,可靶向 PI 3-激酶 VPS34 的功能

Swamynathan Manojit M, Kuang Shan, Watrud Kaitlin E, Doherty Mary R, Gineste Charlotte, Mathew Grinu, Gong Grace Q, Cox Hilary, Cheng Eileen, Reiss David, Kendall Jude, Ghosh Diya, Reczek Colleen R, Zhao Xiang, Herzka Tali, Špokaitė Saulė, Dessus Antoine N, Kim Seung Tea, Klingbeil Olaf, Liu Juan, Nowak Dawid G, Alsudani Habeeb, Wee Tse-Luen, Park Youngkyu, Minicozzi Francesca, Rivera Keith, Almeida Ana S, Chang Kenneth, Chakrabarty Ram P, Wilkinson John E, Gimotty Phyllis A, Diermeier Sarah D, Egeblad Mikala, Vakoc Christopher R, Locasale Jason W, Chandel Navdeep S, Janowitz Tobias, Hicks James B, Wigler Michael, Pappin Darryl J, Williams Roger L, Cifani Paolo, Tuveson David A, Laporte Jocelyn, Trotman Lloyd C

Targeting the mSWI/SNF complex in POU2F-POU2AF transcription factor-driven malignancies.

靶向 POU2F-POU2AF 转录因子驱动的恶性肿瘤中的 mSWI/SNF 复合物

He Tongchen, Xiao Lanbo, Qiao Yuanyuan, Klingbeil Olaf, Young Eleanor, Wu Xiaoli S, Mannan Rahul, Mahapatra Somnath, Redin Esther, Cho Hanbyul, Bao Yi, Kandarpa Malathi, Ching-Yi Tien Jean, Wang Xiaoju, Eyunni Sanjana, Zheng Yang, Kim NamHoon, Zheng Heng, Hou Siyu, Su Fengyun, Miner Stephanie J, Mehra Rohit, Cao Xuhong, Abbineni Chandrasekhar, Samajdar Susanta, Ramachandra Murali, Dhanasekaran Saravana M, Talpaz Moshe, Parolia Abhijit, Rudin Charles M, Vakoc Christopher R, Chinnaiyan Arul M