Metabolism-driven in vitro/in vivo disconnect of an oral ERɑ VHL-PROTAC
代谢驱动的口服ERα VHL-PROTAC体外/体内分离
期刊:Communications Biology
影响因子:5.2
doi:10.1038/s42003-024-06238-x
Thomas G Hayhow ,Beth Williamson ,Mandy Lawson ,Natalie Cureton ,Erin L Braybrooke ,Andrew Campbell ,Rodrigo J Carbajo ,Azadeh Cheraghchi-Bashi ,Elisabetta Chiarparin ,Coura R Diène ,Charlene Fallan ,David I Fisher ,Frederick W Goldberg ,Lorna Hopcroft ,Philip Hopcroft ,Anne Jackson ,Jason G Kettle ,Teresa Klinowska ,Ulrike Künzel ,Gillian Lamont ,Hilary J Lewis ,Gareth Maglennon ,Scott Martin ,Pablo Morentin Gutierrez ,Christopher J Morrow ,Myria Nikolaou ,J Willem M Nissink ,Patrick O'Shea ,Radoslaw Polanski ,Markus Schade ,James S Scott ,Aaron Smith ,Judith Weber ,Joanne Wilson ,Bin Yang ,Claire Crafter