日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Rapid Affinity and Microsomal Stability Ranking of Crude Mixture Libraries of Histone Deacetylase Inhibitors

组蛋白去乙酰化酶抑制剂粗提物库的快速亲和力和微粒体稳定性排序

Tyagarajan, Sriram; Andrews, Christine L; Beshore, Douglas C; Buevich, Alexei V; Curran, Patrick J; Dandliker, Peter; Greshock, Thomas J; Hoar, Jason; Kim, Alex; Karnachi, Prabha; Knemeyer, Ian; Kozlowski, Joseph; Liu, Jian; Maletic, Milana; Myers, Robert; Rada, Vanessa; Sha, Deyou; Sauvagnat, Berengere; Vachal, Petr; Wolkenberg, Scott; Yu, Wensheng; Yu, Younong; Krska, Shane W

In vivo bioluminescence imaging of labile iron in xenograft models and liver using FeAL-1, an iron-activatable form of D-luciferin.

利用 FeAL-1(一种铁激活形式的 D-荧光素)对异种移植模型和肝脏中的不稳定铁进行体内生物发光成像

Gonciarz Ryan L, Jiang Honglin, Tram Linh, Hugelshofer Cedric L, Ekpenyong Oscar, Knemeyer Ian, Aron Allegra T, Chang Christopher J, Flygare John A, Collisson Eric A, Renslo Adam R

Diminishing GSH-Adduct Formation of Tricyclic Diazepine-based Mutant IDH1 Inhibitors

降低三环二氮杂卓类突变型IDH1抑制剂的GSH加合物形成

Huang, Chunhui; Fischer, Christian; Machacek, Michelle R; Bogen, Stephane; Biftu, Tesfaye; Huang, Xianhai; Reutershan, Michael H; Otte, Ryan; Hong, Qingmei; Wu, Zhicai; Yu, Yang; Park, Min; Chen, Lei; Biju, Purakkattle; Knemeyer, Ian; Lu, Ping; Kochansky, Christopher J; Hicks, Michael Brendan; Liu, Yong; Helmy, Roy; Fradera, Xavier; Donofrio, Anthony; Close, Josh; Maddess, Matthew L; White, Catherine; Sloman, David L; Sciammetta, Nunzio; Lu, Jun; Gibeau, Craig; Simov, Vladimir; Zhang, Hongjun; Fuller, Peter; Witter, David

Utilization of Metabolite Identification and Structural Data to Guide Design of Low-Dose IDO1 Inhibitors

利用代谢物鉴定和结构数据指导低剂量IDO1抑制剂的设计

Hopkins, Brett; Zhang, Hongjun; Bharathan, Indu; Li, Derun; Pu, Qinglin; Zhou, Hua; Martinot, Theodore A; Fradera, Xavier; Lammens, Alfred; Lesburg, Charles A; Cohen, Ryan D; Ballard, Jeanine; Knemeyer, Ian; Otte, Karin; Vincent, Stella; Miller, J Richard; Solban, Nicolas; Cheng, Mangeng; Geda, Prasanthi; Smotrov, Nadya; Song, Xuelei; Bennett, David Jonathan; Han, Yongxin

Carbamate and N-Pyrimidine Mitigate Amide Hydrolysis: Structure-Based Drug Design of Tetrahydroquinoline IDO1 Inhibitors

氨基甲酸酯和N-嘧啶可减轻酰胺水解:基于结构的四氢喹啉IDO1抑制剂药物设计

Li, Derun; Deng, Yongqi; Achab, Abdelghani; Bharathan, Indu; Hopkins, Brett Andrew; Yu, Wensheng; Zhang, Hongjun; Sanyal, Sulagna; Pu, Qinglin; Zhou, Hua; Liu, Kun; Lim, Jongwon; Fradera, Xavier; Lesburg, Charles A; Lammens, Alfred; Martinot, Theodore A; Cohen, Ryan D; Doty, Amy C; Ferguson, Heidi; Nickbarg, Elliott B; Cheng, Mangeng; Spacciapoli, Peter; Geda, Prasanthi; Song, Xuelei; Smotrov, Nadya; Abeywickrema, Pravien; Andrews, Christine; Chamberlin, Chad; Mabrouk, Omar; Curran, Patrick; Richards, Matthew; Saradjian, Peter; Miller, J Richard; Knemeyer, Ian; Otte, Karin M; Vincent, Stella; Sciammetta, Nunzio; Pasternak, Alexander; Bennett, David Jonathan; Han, Yongxin

Strategic Incorporation of Polarity in Heme-Displacing Inhibitors of Indoleamine-2,3-dioxygenase-1 (IDO1)

策略性地将极性引入血红素置换抑制剂中,以抑制吲哚胺-2,3-双加氧酶-1 (IDO1)

White, Catherine; McGowan, Meredeth A; Zhou, Hua; Sciammetta, Nunzio; Fradera, Xavier; Lim, Jongwon; Joshi, Elizabeth M; Andrews, Christine; Nickbarg, Elliott B; Cowley, Phillip; Trewick, Sarah; Augustin, Martin; von Köenig, Konstanze; Lesburg, Charles A; Otte, Karin; Knemeyer, Ian; Woo, Hyun; Yu, Wensheng; Cheng, Mangeng; Spacciapoli, Peter; Geda, Prasanthi; Song, Xuelei; Smotrov, Nadya; Curran, Patrick; Heo, Mee Ra; Abeywickrema, Pravien; Miller, J Richard; Bennett, David Jonathan; Han, Yongxin

Discovery of Amino-cyclobutarene-derived Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitors for Cancer Immunotherapy

发现氨基环丁烯衍生的吲哚胺-2,3-双加氧酶1 (IDO1) 抑制剂用于癌症免疫治疗

Zhang, Hongjun; Liu, Kun; Pu, Qinglin; Achab, Abdelghani; Ardolino, Michael J; Cheng, Mangeng; Deng, Yongqi; Doty, Amy C; Ferguson, Heidi; Fradera, Xavier; Knemeyer, Ian; Kurukulasuriya, Ravi; Lam, Yu-Hong; Lesburg, Charles A; Martinot, Theodore A; McGowan, Meredeth A; Miller, J Richard; Otte, Karin; Biju, Purakattle J; Sciammetta, Nunzio; Solban, Nicolas; Yu, Wensheng; Zhou, Hua; Wang, Xiao; Bennett, David Jonathan; Han, Yongxin

Intestinal lymphatic transport for drug delivery

肠道淋巴转运用于药物递送

Yáñez, Jaime A; Wang, Stephen W J; Knemeyer, Ian W; Wirth, Mark A; Alton, Kevin B