日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Target-Directed Approaches for Screening Small Molecules against RNA Targets

针对RNA靶点筛选小分子靶标的靶向方法

Haniff, Hafeez S; Knerr, Laurent; Chen, Jonathan L; Disney, Matthew D; Lightfoot, Helen L

IA-Lab: A MATLAB framework for efficient microscopy image analysis development, applied to quantifying intracellular transport of internalized peptide-drug conjugate

IA-Lab:一个用于高效开发显微图像分析程序的MATLAB框架,应用于量化胞内肽-药物偶联物的转运

Corrigan, Adam M; Karlsson, Johan; Wildenhain, Jan; Knerr, Laurent; Ölwegård-Halvarsson, Maria; Karlsson, Maria; Lünse, Svenja; Wang, Yinhai

Development of Novel Melanocortin Receptor Agonists Based on the Cyclic Peptide Framework of Sunflower Trypsin Inhibitor-1.

基于向日葵胰蛋白酶抑制剂-1的环肽骨架开发新型黑皮质素受体激动剂

Durek Thomas, Cromm Philipp M, White Andrew M, Schroeder Christina I, Kaas Quentin, Weidmann Joachim, Ahmad Fuaad Abdullah, Cheneval Olivier, Harvey Peta J, Daly Norelle L, Zhou Yang, Dellsén Anita, Österlund Torben, Larsson Niklas, Knerr Laurent, Bauer Udo, Kessler Horst, Cai Minying, Hruby Victor J, Plowright Alleyn T, Craik David J

Design of Selective sPLA(2)-X Inhibitor (-)-2-{2-[Carbamoyl-6-(trifluoromethoxy)-1H-indol-1-yl]pyridine-2-yl}propanoic Acid

选择性 sPLA(2)-X 抑制剂 (-)-2-{2-[氨基甲酰基-6-(三氟甲氧基)-1H-吲哚-1-基]吡啶-2-基}丙酸的设计

Giordanetto, Fabrizio; Knerr, Laurent; Nordberg, Peter; Pettersen, Daniel; Selmi, Nidhal; Beisel, Hans-Georg; de la Motte, Hannah; Månsson, Åsa; Dahlström, Mikael; Broddefalk, Johan; Saarinen, Gabrielle; Klingegård, Fredrik; Hurt-Camejo, Eva; Rosengren, Birgitta; Wikström, Johannes; Wågberg, Maria; Brengdahl, Johan; Rohman, Mattias; Sandmark, Jenny; Åkerud, Tomas; Roth, Robert G; Jansen, Frank; Ahlqvist, Marie

Discovery of a Series of Indole-2 Carboxamides as Selective Secreted Phospholipase A(2) Type X (sPLA(2)-X) Inhibitors.

发现一系列吲哚-2 甲酰胺类化合物作为选择性分泌型磷脂酶 A(2) X 型 (sPLA(2)-X) 抑制剂

Knerr Laurent, Giordanetto Fabrizio, Nordberg Peter, Pettersen Daniel, Selmi Nidhal, Beisel Hans-Georg, de la Motte Hannah, Olsson Thomas, Perkins Tim D J, Herslöf Margareta, Månsson à sa, Dahlström Mikael, Starke Ingemar, Broddefalk Johan, Saarinen Gabrielle, Klingegård Fredrik, Hurt-Camejo Eva, Rosengren Birgitta, Brengdahl Johan, Jansen Frank, Rohman Mattias, Sandmark Jenny, Hallberg Kenth, à kerud Tomas, Roth Robert G, Ahlqvist Marie