日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Author Correction: Direct and selective pharmacological disruption of the YAP-TEAD interface by IAG933 inhibits Hippo-dependent and RAS-MAPK-altered cancers

作者更正:IAG933 通过直接和选择性地药理学手段破坏 YAP-TEAD 界面,从而抑制 Hippo 依赖性和 RAS-MAPK 改变的癌症。

Chapeau, Emilie A; Sansregret, Laurent; Galli, Giorgio G; Chène, Patrick; Wartmann, Markus; Mourikis, Thanos P; Jaaks, Patricia; Baltschukat, Sabrina; Barbosa, Ines A M; Bauer, Daniel; Brachmann, Saskia M; Delaunay, Clara; Estadieu, Claire; Faris, Jason E; Furet, Pascal; Harlfinger, Stefanie; Hueber, Andreas; Jiménez Núñez, Eloísa; Kodack, David P; Mandon, Emeline; Martin, Typhaine; Mesrouze, Yannick; Romanet, Vincent; Scheufler, Clemens; Sellner, Holger; Stamm, Christelle; Sterker, Dario; Tordella, Luca; Hofmann, Francesco; Soldermann, Nicolas; Schmelzle, Tobias

Direct and selective pharmacological disruption of the YAP-TEAD interface by IAG933 inhibits Hippo-dependent and RAS-MAPK-altered cancers

IAG933通过直接和选择性地药理学手段破坏YAP-TEAD界面,从而抑制Hippo依赖性和RAS-MAPK改变的癌症。

Emilie A Chapeau ,Laurent Sansregret ,Giorgio G Galli ,Patrick Chène ,Markus Wartmann ,Thanos P Mourikis ,Patricia Jaaks ,Sabrina Baltschukat ,Ines A M Barbosa ,Daniel Bauer ,Saskia M Brachmann ,Clara Delaunay ,Claire Estadieu ,Jason E Faris ,Pascal Furet ,Stefanie Harlfinger ,Andreas Hueber ,Eloísa Jiménez Núñez ,David P Kodack ,Emeline Mandon ,Typhaine Martin ,Yannick Mesrouze ,Vincent Romanet ,Clemens Scheufler ,Holger Sellner ,Christelle Stamm ,Dario Sterker ,Luca Tordella ,Francesco Hofmann ,Nicolas Soldermann ,Tobias Schmelzle

A complication of an axillary intra-aortic balloon pump

腋窝主动脉内球囊反搏泵的并发症

Kodack, Eileen; Patel, Riya; Bonner, Carain; Pantin, Enrique

RNF43 mutations predict response to anti-BRAF/EGFR combinatory therapies in BRAFV600E metastatic colorectal cancer

RNF43 突变可预测 BRAFV600E 转移性结直肠癌对抗 BRAF/EGFR 联合疗法的疗效

Elena Elez, Javier Ros, Jose Fernández, Guillermo Villacampa, Ana Belén Moreno-Cárdenas, Carlota Arenillas, Kinga Bernatowicz, Raquel Comas, Shanshan Li, David Philip Kodack, Roberta Fasani, Ariadna Garcia, Javier Gonzalo-Ruiz, Alejandro Piris-Gimenez, Paolo Nuciforo, Grainne Kerr, Rossana Intini, A

FATTY ACID SYNTHESIS IS REQUIRED FOR BREAST CANCER BRAIN METASTASIS

脂肪酸合成是乳腺癌脑转移所必需的

Gino B Ferraro # ,Ahmed Ali # ,Alba Luengo # ,David P Kodack ,Amy Deik ,Keene L Abbott ,Divya Bezwada ,Landry Blanc ,Brendan Prideaux ,Xin Jin ,Jessica M Posada ,Jiang Chen ,Christopher R Chin ,Zohreh Amoozgar ,Raphael Ferreira ,Ivy X Chen ,Kamila Naxerova ,Christopher Ng ,Anna M Westermark ,Mark Duquette ,Sylvie Roberge ,Neal I Lindeman ,Costas A Lyssiotis ,Jens Nielsen ,David E Housman ,Dan G Duda ,Elena Brachtel ,Todd R Golub ,Lewis C Cantley ,John M Asara ,Shawn M Davidson ,Dai Fukumura ,Véronique A Dartois ,Clary B Clish ,Rakesh K Jain ,Matthew G Vander Heiden

Dual endothelin receptor inhibition enhances T-DM1 efficacy in brain metastases from HER2-positive breast cancer

双重内皮素受体抑制可增强 T-DM1 对 HER2 阳性乳腺癌脑转移的疗效

Vasileios Askoxylakis, Gino B Ferraro, Mark Badeaux, David P Kodack, Isabelle Kirst, Ram C Shankaraiah, Christina S F Wong, Dan G Duda, Dai Fukumura, Rakesh K Jain

The brain microenvironment mediates resistance in luminal breast cancer to PI3K inhibition through HER3 activation

脑微环境通过HER3激活介导管腔型乳腺癌对PI3K抑制剂的耐药性。

Kodack, David P; Askoxylakis, Vasileios; Ferraro, Gino B; Sheng, Qing; Badeaux, Mark; Goel, Shom; Qi, Xiaolong; Shankaraiah, Ram; Cao, Z Alexander; Ramjiawan, Rakesh R; Bezwada, Divya; Patel, Bhushankumar; Song, Yongchul; Costa, Carlotta; Naxerova, Kamila; Wong, Christina S F; Kloepper, Jonas; Das, Rita; Tam, Angela; Tanboon, Jantima; Duda, Dan G; Miller, C Ryan; Siegel, Marni B; Anders, Carey K; Sanders, Melinda; Estrada, Monica V; Schlegel, Robert; Arteaga, Carlos L; Brachtel, Elena; Huang, Alan; Fukumura, Dai; Engelman, Jeffrey A; Jain, Rakesh K

Primary Patient-Derived Cancer Cells and Their Potential for Personalized Cancer Patient Care

患者来源的原发性癌细胞及其对癌症患者个性化治疗的潜力

David P Kodack, Anna F Farago, Anahita Dastur, Matthew A Held, Leila Dardaei, Luc Friboulet, Friedrich von Flotow, Leah J Damon, Dana Lee, Melissa Parks, Richard Dicecca, Max Greenberg, Krystina E Kattermann, Amanda K Riley, Florian J Fintelmann, Coleen Rizzo, Zofia Piotrowska, Alice T Shaw, Justin

Preclinical Efficacy of Ado-trastuzumab Emtansine in the Brain Microenvironment

Ado-trastuzumab Emtansine 在脑微环境中的临床前疗效

Vasileios Askoxylakis, Gino B Ferraro, David P Kodack, Mark Badeaux, Ram C Shankaraiah, Giorgio Seano, Jonas Kloepper, Trupti Vardam, John D Martin, Kamila Naxerova, Divya Bezwada, Xiaolong Qi, Martin K Selig, Elena Brachtel, Dan G Duda, Peigen Huang, Dai Fukumura, Jeffrey A Engelman, Rakesh K Jain

Blockade of MMP14 activity in murine breast carcinomas: implications for macrophages, vessels, and radiotherapy

阻断小鼠乳腺癌中的 MMP14 活性:对巨噬细胞、血管和放射治疗的影响

Eleanor I Ager, Sergey V Kozin, Nathaniel D Kirkpatrick, Giorgio Seano, David P Kodack, Vasileios Askoxylakis, Yuhui Huang, Shom Goel, Matija Snuderl, Alona Muzikansky, Dianne M Finkelstein, Daniel T Dransfield, Laetitia Devy, Yves Boucher, Dai Fukumura, Rakesh K Jain