日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural basis of the residence time of adenosine A(2A) receptor ligands revealed by NMR

核磁共振揭示腺苷A(2A)受体配体停留时间的结构基础

Ueda, Takumi; Tsuchida, Tomoki; Kurita, Masatoshi; Mizumura, Takuya; Imai, Shunsuke; Shiraishi, Yutaro; Kofuku, Yutaka; Miyakawa, Shuhei; Fukuzawa, Kaori; Takeuchi, Koh; Shimada, Ichio

A Case of Allergic Bronchopulmonary Mycosis Caused by Cordyceps farinosa, a Species of Caterpillar Fungi

由虫草菌(一种冬虫夏草)引起的过敏性支气管肺真菌病病例报告

Sakano, Yuta; Okumura, Taro; Kofuku, Tomomi; Kidaka, Saki; Nakata, Yugo; Katsura, Satoshi; Goto, Kenichi; Shigematsu, Michio

Activation mechanism of the μ-opioid receptor by an allosteric modulator

变构调节剂激活μ-阿片受体的机制

Kaneko, Shun; Imai, Shunsuke; Asao, Nobuaki; Kofuku, Yutaka; Ueda, Takumi; Shimada, Ichio

Biphasic activation of β-arrestin 1 upon interaction with a GPCR revealed by methyl-TROSY NMR

甲基-TROSY NMR 揭示 β-arrestin 1 与 GPCR 相互作用时的双相激活

Yutaro Shiraishi, Yutaka Kofuku, Takumi Ueda, Shubhi Pandey, Hemlata Dwivedi-Agnihotri, Arun K Shukla, Ichio Shimada

Function-Related Dynamics in Multi-Spanning Helical Membrane Proteins Revealed by Solution NMR

溶液核磁共振揭示多跨膜螺旋膜蛋白的功能相关动力学

Takeuchi, Koh; Kofuku, Yutaka; Imai, Shunsuke; Ueda, Takumi; Tokunaga, Yuji; Toyama, Yuki; Shiraishi, Yutaro; Shimada, Ichio

Targeting FROUNT with disulfiram suppresses macrophage accumulation and its tumor-promoting properties

使用双硫仑靶向 FROUNT 可抑制巨噬细胞聚集及其促肿瘤特性。

Yuya Terashima # ,Etsuko Toda # ,Meiji Itakura ,Mikiya Otsuji ,Sosuke Yoshinaga ,Kazuhiro Okumura ,Francis H W Shand ,Yoshihiro Komohara ,Mitsuhiro Takeda ,Kana Kokubo ,Ming-Chen Chen ,Sana Yokoi ,Hirofumi Rokutan ,Yutaka Kofuku ,Koji Ohnishi ,Miki Ohira ,Toshihiko Iizasa ,Hirofumi Nakano ,Takayoshi Okabe ,Hirotatsu Kojima ,Akira Shimizu ,Shiro Kanegasaki ,Ming-Rong Zhang ,Ichio Shimada ,Hiroki Nagase ,Hiroaki Terasawa ,Kouji Matsushima

Activation of adenosine A2A receptor by lipids from docosahexaenoic acid revealed by NMR

NMR 揭示二十二碳六烯酸脂质对腺苷 A2A 受体的激活作用

Takuya Mizumura, Keita Kondo, Masatoshi Kurita, Yutaka Kofuku, Mei Natsume, Shunsuke Imai, Yutaro Shiraishi, Takumi Ueda, Ichio Shimada

GPCR drug discovery: integrating solution NMR data with crystal and cryo-EM structures

GPCR药物发现:整合溶液核磁共振数据与晶体和冷冻电镜结构

Shimada, Ichio; Ueda, Takumi; Kofuku, Yutaka; Eddy, Matthew T; Wüthrich, Kurt

Function-related conformational dynamics of G protein-coupled receptors revealed by NMR

核磁共振揭示G蛋白偶联受体的功能相关构象动力学

Ueda, Takumi; Kofuku, Yutaka; Okude, Junya; Imai, Shunsuke; Shiraishi, Yutaro; Shimada, Ichio

Phosphorylation-induced conformation of β2-adrenoceptor related to arrestin recruitment revealed by NMR

核磁共振揭示与抑制蛋白募集有关的β2-肾上腺素能受体磷酸化诱导构象

Yutaro Shiraishi, Mei Natsume, Yutaka Kofuku, Shunsuke Imai, Kunio Nakata, Toshimi Mizukoshi, Takumi Ueda, Hideo Iwaï, Ichio Shimada