日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Based Design of Covalent SARS-CoV‑2 Main Protease Inhibitors Targeting the Nirmatrelvir-Resistant E166 Mutants

基于结构的共价SARS-CoV-2主蛋白酶抑制剂设计,靶向耐尼马替利韦的E166突变体

Cai, Zhengjun; Kohaal, Navita; Georgiou, Kyriakos; Liang, Xueying; Chi, Xiang; Tan, Haozhou; Tan, Bin; Li, Kan; Fan, Guangjin; Lambrinidis, George; Kolocouris, Antonios; Deng, Xufang; Chen, Yu; Wang, Jun

Distal protein-protein interactions contribute to nirmatrelvir resistance

远端蛋白质-蛋白质相互作用导致尼尔马特雷韦耐药性

Eric M Lewandowski # ,Xiujun Zhang # ,Haozhou Tan # ,Aiden Jaskolka-Brown ,Navita Kohaal ,Aliaksandra Frazier ,Jesper J Madsen ,Lian M C Jacobs ,Jun Wang ,Yu Chen