日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

In vitro evaluation of the immunogenic potential of gramicidin S and its photocontrolled analogues.

体外评价革兰氏菌素 S 及其光控类似物的免疫原性

Horbatok Kateryna, Semchuk Iryna, Horbach Oleksandr, Khranovska Natalia, Kosach Viktoriia, Borysko Petro, Koniev Serhii, Ulrich Anne S, Afonin Sergii, Komarov Igor V

Neural Network Models for Prediction of Biological Activity using Molecular Dynamics Data: A Case of Photoswitchable Peptides

利用分子动力学数据预测生物活性的神经网络模型:以光开关肽为例

Cherednichenko, Anton; Afonin, Sergii; Babii, Oleg; Voitsitskyi, Taras; Stratiichuk, Roman; Koleiev, Ihor; Vozniak, Volodymyr; Shevchuk, Nazar; Ostrovsky, Zakhar; Yesylevskyy, Semen; Nafiiev, Alan; Starosyla, Serhii; Ulrich, Anne S; Jirgensons, Aigars; Komarov, Igor V

Structure-Activity Assessment and In-Depth Analysis of Biased Agonism in a Set of Phenylalkylamine 5-HT(2A) Receptor Agonists

苯烷基胺类5-HT(2A)受体激动剂的结构-活性评价及偏向性激动作用的深入分析

Pottie, Eline; Poulie, Christian B M; Simon, Icaro A; Harpsøe, Kasper; D'Andrea, Laura; Komarov, Igor V; Gloriam, David E; Jensen, Anders A; Kristensen, Jesper L; Stove, Christophe P

Challenges for chemistry in Ukraine after the war: Ukrainian science requires rebuilding and support

战后乌克兰化学面临的挑战:乌克兰科学需要重建和支持

Kondratov, Ivan S; Moroz, Yurii S; Gorgulla, Christoph; Grygorenko, Oleksandr O; Komarov, Igor V; Wagner, Gerhard; Tolmachev, Andrey A

Discovery of β-Arrestin-Biased 25CN-NBOH-Derived 5-HT(2A) Receptor Agonists

发现β-arrestin偏向性25CN-NBOH衍生的5-HT(2A)受体激动剂

Poulie, Christian B M; Pottie, Eline; Simon, Icaro A; Harpsøe, Kasper; D'Andrea, Laura; Komarov, Igor V; Gloriam, David E; Jensen, Anders A; Stove, Christophe P; Kristensen, Jesper L

Diarylethene-Based Photoswitchable Inhibitors of Serine Proteases

基于二芳基乙烯的光开关丝氨酸蛋白酶抑制剂

Babii, Oleg; Afonin, Sergii; Diel, Christian; Huhn, Marcel; Dommermuth, Jennifer; Schober, Tim; Koniev, Serhii; Hrebonkin, Andrii; Nesterov-Mueller, Alexander; Komarov, Igor V; Ulrich, Anne S

Nature of Fast Relaxation Processes and Spectroscopy of a Membrane-Active Peptide Modified with Fluorescent Amino Acid Exhibiting Excited State Intramolecular Proton Transfer and Efficient Stimulated Emission

快速弛豫过程的性质及荧光氨基酸修饰的膜活性肽的光谱学研究,该肽表现出激发态分子内质子转移和高效受激发射

Shaydyuk, Yevgeniy O; Bashmakova, Nataliia V; Dmytruk, Andriy M; Kachkovsky, Olexiy D; Koniev, Serhii; Strizhak, Alexander V; Komarov, Igor V; Belfield, Kevin D; Bondar, Mykhailo V; Babii, Oleg

In Vivo Behavior of the Antibacterial Peptide Cyclo[RRRWFW], Explored Using a 3-Hydroxychromone-Derived Fluorescent Amino Acid

利用3-羟基色酮衍生的荧光氨基酸研究抗菌肽环[RRRWFW]的体内行为

Afonin, Sergii; Koniev, Serhii; Préau, Laetitia; Takamiya, Masanari; Strizhak, Alexander V; Babii, Oleg; Hrebonkin, Andrii; Pivovarenko, Vasyl G; Dathe, Margitta; le Noble, Ferdinand; Rastegar, Sepand; Strähle, Uwe; Ulrich, Anne S; Komarov, Igor V

Light-controllable dithienylethene-modified cyclic peptides: photoswitching the in vivo toxicity in zebrafish embryos

光控二噻吩乙烯修饰环肽:光开关斑马鱼胚胎体内毒性

Afonin, Sergii; Babii, Oleg; Reuter, Aline; Middel, Volker; Takamiya, Masanari; Strähle, Uwe; Komarov, Igor V; Ulrich, Anne S

Orientation and Location of the Cyclotide Kalata B1 in Lipid Bilayers Revealed by Solid-State NMR

固态核磁共振揭示环肽Kalata B1在脂质双层中的取向和位置

Grage, Stephan L; Sani, Marc-Antoine; Cheneval, Olivier; Henriques, Sónia Troeira; Schalck, Constantin; Heinzmann, Ralf; Mylne, Joshua S; Mykhailiuk, Pavel K; Afonin, Sergii; Komarov, Igor V; Separovic, Frances; Craik, David J; Ulrich, Anne S