Discovery of a Druggable, Cryptic Pocket in SARS-CoV-2 nsp16 Using Allosteric Inhibitors
利用变构抑制剂发现SARS-CoV-2 nsp16中一个可成药的隐蔽口袋
期刊:ACS Infectious Diseases
影响因子:3.8
doi:10.1021/acsinfecdis.3c00203
Inniss, Nicole L; Kozic, Ján; Li, Fengling; Rosas-Lemus, Monica; Minasov, George; Rybáček, Jiří; Zhu, Yingjie; Pohl, Radek; Shuvalova, Ludmilla; Rulíšek, Lubomír; Brunzelle, Joseph S; Bednárová, Lucie; Štefek, Milan; Kormaník, Ján Michael; Andris, Erik; Šebestík, Jaroslav; Li, Alice Shi Ming; Brown, Peter J; Schmitz, Uli; Saikatendu, Kumar; Chang, Edcon; Nencka, Radim; Vedadi, Masoud; Satchell, Karla J F