日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Rational Design of CDK12/13 and BRD4 Molecular Glue Degraders

CDK12/13 和 BRD4 分子胶降解剂的合理设计

Zhuang, Zhe; Byun, Woong Sub; Kozicka, Zuzanna; Donovan, Katherine A; Dwyer, Brendan G; Thornhill, Abby M; Jones, Hannah M; Jiang, Zixuan; Zhu, Xijun; Fischer, Eric S; Thomä, Nicolas H; Gray, Nathanael S

Expanding the druggable zinc-finger proteome defines properties of drug-induced degradation.

扩大可成药锌指蛋白组,可以明确药物诱导降解的特性

Słabicki Mikołaj, Park Jiho, Nowak Radosław P, Roy Burman Shourya S, Pellman Jesse, Zou Charles, Razumkov Hlib, Carreiro Jeannie, Rastogi Simran, Goldstein Anna, Nagiec Marek M, Donovan Katherine A, Che Jianwei, Hunkeler Moritz, Geng Qixiang, Hsu Chi-Lin, Lakshminarayan Megha, Shu Chelsea, Zon Rebecca L, Kozicka Zuzanna, Park Paul M C, Tsai Jonathan M, Yoon Hojong, Jones Lyn H, Sperling Adam S, Gray Nathanael S, Fischer Eric S, Ebert Benjamin L

Clues for glues: from serendipity to nature's blueprints in degrader discovery

粘合剂的线索:从偶然发现到降解剂发现中的自然蓝图

Kozicka, Zuzanna

Development of Degraders and 2-pyridinecarboxyaldehyde (2-PCA) as a recruitment Ligand for FBXO22.

开发降解剂和 2-吡啶甲醛 (2-PCA) 作为 FBXO22 的募集配体

Qiu Tian, Zhuang Zhe, Byun Woong Sub, Kozicka Zuzanna, Baek Kheewoong, Zhong Jianing, Thornhill Abby M, Ryan Julia K, Donovan Katherine A, Fischer Eric S, Ebert Benjamin L, Gray Nathanael S