日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of VU6083859, a TAOK1 Selective Inhibitor, and VU6080195, a pan-TAOK Activator

发现 VU6083859(一种 TAOK1 选择性抑制剂)和 VU6080195(一种泛 TAOK 激活剂)

Schultz, Daniel C; Parr, Lauren C; Sweet, Hunter; Lamb, Sean; Engers, Julie L; Napier, Nathaniel C; McKinnie, Hallie G; Whomble, David; Kramlinger, Valerie; Boutaud, Olivier; Lindsley, Craig W

Discovery of a Novel sp(3)‑Rich M(1) Positive Allosteric Modulators (PAMs) Chemotype via Scaffold Hopping

通过骨架跃迁发现一种新型富含sp(3)杂环的M(1)正变构调节剂(PAM)化学类型

Bungard, Joseph D; Spearing, Paul; Nishio, Yu; Rathnayake, Upendra; Presley, Chris C; Chang, Sichen; Kling, Haley E; Thompson, Analisa D; Cho, Hyekyung P; Peng, Li; Rodriguez, Alice L; Niswender, Colleen M; Boutaud, Olivier; Kramlinger, Valerie; Jones, Carrie K; Conn, P Jeffrey; Engers, Julie L; Engers, Darren W; Lindsley, Craig W; Han, Changho

Discovery of VU6052254: A Novel, Potent M(1) Positive Allosteric Modulator

VU6052254 的发现:一种新型、强效的 M(1) 正向变构调节剂

Engers, Julie L; Bungard, Joseph D; Presley, Christopher C; Zagol-Ikapitte, Irene; Watson, Katherine J; Chang, Sichen; O'Carroll, Colin; Dey, P Markus; Burstein, Ethan S; Dickerson, Jonathan W; Thompson Gray, Analisa; Bubser, Michael; Rook, Jerri M; Cho, Hyekyung P; Kramlinger, Valerie M; Boutaud, Olivier; Jones, Carrie K; Conn, P Jeffrey; Engers, Darren W; Lindsley, Craig W

Highly Potent and Subtype-Selective Sperm-Specific Potassium Channel SLO3 Inhibitors Display High Tissue Exposure in the Murine Female Reproductive Tract

高效且具有亚型选择性的精子特异性钾通道SLO3抑制剂在小鼠雌性生殖道中表现出高组织暴露量

Temple, Kayla J; Li, Ping; McKinnie, Hallie G; Thompson Gray, Analisa; Bertron, Jeanette L; Ringuette, Anna E; de Andrade Horn, Pedro; Lyon, Maximilian D; Bhagwat, Shweta; Asadi, Leila; Li, Sophia; Lazarenko, Roman M; McCarthy, Ronald; Chang, Sichen; Turkett, Jeremy A; Kramlinger, Valerie; Watson, Katherine J; Zagol-Ikapitte, Irene A; Denton, Jerod S; Santi, Celia M; Jones, Carrie K; Lindsley, Craig W; Boutaud, Olivier

Computer-Aided Design and Biological Evaluation of Diazaspirocyclic D(4)R Antagonists

二氮杂螺环D(4)R拮抗剂的计算机辅助设计和生物学评价

Jones, Caleb A H; Brown, Benjamin P; Schultz, Daniel C; Engers, Julie; Kramlinger, Valerie M; Meiler, Jens; Lindsley, Craig W

Interviewer biases in medical survey data: The example of blood pressure measurements

医疗调查数据中的访谈者偏差:以血压测量为例

Geldsetzer, Pascal; Chang, Andrew Young; Meijer, Erik; Sudharsanan, Nikkil; Charu, Vivek; Kramlinger, Peter; Haarburger, Richard

Novel advances in biotransformation and bioactivation research - 2020 year in review

生物转化和生物活化研究的新进展——2020年回顾

Khojasteh, S Cyrus; Argikar, Upendra A; Driscoll, James P; Heck, Carley J S; King, Lloyd; Jackson, Klarissa D; Jian, Wenying; Kalgutkar, Amit S; Miller, Grover P; Kramlinger, Valerie; Rietjens, Ivonne M C M; Teitelbaum, Aaron M; Wang, Kai; Wei, Cong

Human cytochrome P450 27C1 catalyzes 3,4-desaturation of retinoids

人细胞色素P450 27C1催化类视黄醇的3,4-去饱和作用

Kramlinger, Valerie M; Nagy, Leslie D; Fujiwara, Rina; Johnson, Kevin M; Phan, Thanh T N; Xiao, Yi; Enright, Jennifer M; Toomey, Matthew B; Corbo, Joseph C; Guengerich, Frederick Peter

Oxidation of pyrene, 1-hydroxypyrene, 1-nitropyrene and 1-acetylpyrene by human cytochrome P450 2A13

人细胞色素P450 2A13对芘、1-羟基芘、1-硝基芘和1-乙酰基芘的氧化作用

Shimada, Tsutomu; Takenaka, Shigeo; Murayama, Norie; Kramlinger, Valerie M; Kim, Joo-Hwan; Kim, Donghak; Liu, Jiawang; Foroozesh, Maryam K; Yamazaki, Hiroshi; Guengerich, F Peter; Komori, Masayuki

Cyp27c1 Red-Shifts the Spectral Sensitivity of Photoreceptors by Converting Vitamin A1 into A2.

Cyp27c1 通过将维生素 A1 转化为 A2 来红移光感受器的光谱敏感性

Enright Jennifer M, Toomey Matthew B, Sato Shin-ya, Temple Shelby E, Allen James R, Fujiwara Rina, Kramlinger Valerie M, Nagy Leslie D, Johnson Kevin M, Xiao Yi, How Martin J, Johnson Stephen L, Roberts Nicholas W, Kefalov Vladimir J, Guengerich F Peter, Corbo Joseph C