日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Periphery Exploration around 2,6-Diazaspiro[3.4]octane Core Identifies a Potent Nitrofuran Antitubercular Lead.

围绕 2,6-二氮杂螺[3.4]辛烷核心的外围探索发现了一种强效的硝基呋喃抗结核先导化合物

Lukin Alexei, Komarova Kristina, Vinogradova Lyubov, Dogonadze Marine, Vinogradova Tatiana, Yablonsky Piotr, Kazantsev Alexander, Krasavin Mikhail

5-(Sulfamoyl)thien-2-yl 1,3-oxazole inhibitors of carbonic anhydrase II with hydrophilic periphery

具有亲水性外围结构的 5-(磺酰基)噻吩-2-基 1,3-噁唑类碳酸酐酶 II 抑制剂

Kalinin, Stanislav; Kovalenko, Alexander; Valtari, Annika; Nocentini, Alessio; Gureev, Maxim; Urtti, Arto; Korsakov, Mikhail; Supuran, Claudiu T; Krasavin, Mikhail

Diversely substituted sulfamides for fragment-based drug discovery of carbonic anhydrase inhibitors: synthesis and inhibitory profile

用于基于片段的碳酸酐酶抑制剂药物发现的多种取代磺酰胺:合成及抑制谱

Sharonova, Tatiana; Zhmurov, Petr; Kalinin, Stanislav; Nocentini, Alessio; Angeli, Andrea; Ferraroni, Marta; Korsakov, Mikhail; Supuran, Claudiu T; Krasavin, Mikhail

The Use of Aryl-Substituted Homophthalic Anhydrides in the Castagnoli-Cushman Reaction Provides Access to Novel Tetrahydroisoquinolone Carboxylic Acid Bearing an All-Carbon Quaternary Stereogenic Center

在 Castagnoli-Cushman 反应中使用芳基取代的邻苯二甲酸酐可合成具有全碳季碳立体中心的新型四氢异喹啉酮羧酸。

Moshnenko, Nazar; Kazantsev, Alexander; Bakulina, Olga; Dar'in, Dmitry; Krasavin, Mikhail

Preparation and Synthetic Applications of Five-to-Seven-Membered Cyclic α-Diazo Monocarbonyl Compounds

五元至七元环状α-重氮单羰基化合物的制备及其合成应用

Zhukovsky, Daniil; Dar'in, Dmitry; Bakulina, Olga; Krasavin, Mikhail

The Role of the Thioredoxin Detoxification System in Cancer Progression and Resistance

硫氧还蛋白解毒系统在癌症进展和耐药性中的作用

Jovanović, Mirna; Podolski-Renić, Ana; Krasavin, Mikhail; Pešić, Milica

Novel 5-Nitrofuran-Tagged Imidazo-Fused Azines and Azoles Amenable by the Groebke-Blackburn-Bienaymé Multicomponent Reaction: Activity Profile against ESKAPE Pathogens and Mycobacteria

新型5-硝基呋喃标记的咪唑稠合嗪和唑类化合物可通过Groebke-Blackburn-Bienaymé多组分反应合成:针对ESKAPE病原体和分枝杆菌的活性分析

Sapegin, Alexander; Rogacheva, Elizaveta; Kraeva, Lyudmila; Gureev, Maxim; Dogonadze, Marine; Vinogradova, Tatiana; Yablonsky, Petr; Balalaie, Saeed; Baykov, Sergey V; Krasavin, Mikhail

Synthesis, Structure, and Antiproliferative Action of 2-Pyridyl Urea-Based Cu(II) Complexes

2-吡啶基脲基Cu(II)配合物的合成、结构及抗增殖作用

Geyl, Kirill K; Baykov, Sergey V; Kalinin, Stanislav A; Bunev, Alexandr S; Troshina, Marina A; Sharonova, Tatiana V; Skripkin, Mikhail Yu; Kasatkina, Svetlana O; Presnukhina, Sofia I; Shetnev, Anton A; Krasavin, Mikhail Yu; Boyarskiy, Vadim P

Multicomponent Reactions Involving Diazo Reagents: A 5-Year Update

涉及重氮试剂的多组分反应:五年最新进展

Bakulina, Olga; Inyutina, Anna; Dar'in, Dmitry; Krasavin, Mikhail

Diazocarbonyl and Related Compounds in the Synthesis of Azoles

重氮羰基化合物及相关化合物在唑类化合物合成中的应用

Budeev, Anton; Kantin, Grigory; Dar'in, Dmitry; Krasavin, Mikhail