日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

SuFEx-based antitubercular compound irreversibly inhibits Pks13

基于 SuFEx 的抗结核化合物不可逆地抑制 Pks13

Krieger, Inna V; Sukheja, Paridhi; Yang, Baiyuan; Tang, Su; Selle, Daniel; Woods, Ashley; Engelhart, Curtis; Kumar, Pradeep; Harbut, Michael B; Liu, Dongdong; Tsuda, Brendan; Qin, Bo; Bare, Grant A L; Li, Gencheng; Chi, Victor; Gambacurta, Julian; Hvizdos, Janine; Reagan, Matthew; Jones, Isabelle L; Massoudi, Lisa M; Woolhiser, Lisa K; Cascioferro, Alessandro; Kundrick, Erica; Singh, Parul; Reiley, William; Ioerger, Thomas R; Kandula, Dilipkumar Reddy; McCabe, Jacob W; Guo, Taijie; Alland, David; Boshoff, Helena I; Schnappinger, Dirk; Robertson, Gregory T; Mdluli, Khisi; Lee, Kyoung-Jin; Dong, Jiajia; Li, Shuangwei; Schultz, Peter G; Joseph, Sean B; Love, Melissa S; Sharpless, K Barry; Petrassi, H Michael; Chatterjee, Arnab K; Sacchettini, James C; McNamara, Case W

Thioquinazolinones as Antituberculosis Agents Targeting Phosphopantetheinyl Transferase

硫代喹唑啉酮类化合物作为靶向磷酸泛酰巯基转移酶的抗结核药物

Singh, Amrita; Zwerneman, Logan T; Planck, Kyle; Kaneko, Takushi; Perkowski, Andrew J; Suh, Christine M; Alex, Alexander; Bean, James; Burns-Huang, Kristin; Zhang, David; Boshoff, Helena I M; Roubert, Christine; Krieger, Inna; Gardner, Mark; Cautain, Bastien; Cooper, Christopher B; Tanvir, Zaid; Sacchettini, James; Gold, Ben S; Rhee, Kyu Y; Fotouhi, Nader; Nathan, Carl F; Aubé, Jeffrey

Redirecting raltitrexed from cancer cell thymidylate synthase to Mycobacterium tuberculosis phosphopantetheinyl transferase.

将 raltitrexed 从癌细胞胸苷酸合成酶重定向到结核分枝杆菌磷酸泛酰巯基转移酶

Singh Amrita, Ottavi Samantha, Krieger Inna, Planck Kyle, Perkowski Andrew, Kaneko Takushi, Davis Andrew M, Suh Christine, Zhang David, Goullieux Laurent, Alex Alexander, Roubert Christine, Gardner Mark, Preston Marian, Smith Dave M, Ling Yan, Roberts Julia, Cautain Bastien, Upton Anna, Cooper Christopher B, Serbina Natalya, Tanvir Zaid, Mosior John, Ouerfelli Ouathek, Yang Guangli, Gold Ben S, Rhee Kyu Y, Sacchettini James C, Fotouhi Nader, Aubé Jeffrey, Nathan Carl

An oral non-covalent non-peptidic inhibitor of SARS-CoV-2 Mpro ameliorates viral replication and pathogenesis in vivo.

SARS-CoV-2 Mpro 的口服非共价非肽抑制剂可改善体内病毒复制和致病性

Zhou Nian E, Tang Su, Bian Xuelin, Parai Maloy K, Krieger Inna V, Flores Armando, Jaiswal Pradeep K, Bam Radha, Wood Jeremy L, Shi Zhe, Stevens Laura J, Scobey Trevor, Diefenbacher Meghan V, Moreira Fernando R, Baric Thomas J, Acharya Arjun, Shin Joonyoung, Rathi Manish M, Wolff Karen C, Riva Laura, Bakowski Malina A, McNamara Case W, Catanzaro Nicholas J, Graham Rachel L, Schultz David C, Cherry Sara, Kawaoka Yoshihiro, Halfmann Peter J, Baric Ralph S, Denison Mark R, Sheahan Timothy P, Sacchettini James C

Structural anatomy of Protein Kinase C C1 domain interactions with diacylglycerol and other agonists

蛋白激酶C C1结构域与二酰甘油和其他激动剂相互作用的结构解剖

Katti, Sachin S; Krieger, Inna V; Ann, Jihyae; Lee, Jeewoo; Sacchettini, James C; Igumenova, Tatyana I

Bedaquiline reprograms central metabolism to reveal glycolytic vulnerability in Mycobacterium tuberculosis

贝达喹啉通过重编程中心代谢来揭示结核分枝杆菌的糖酵解脆弱性

Mackenzie, Jared S; Lamprecht, Dirk A; Asmal, Rukaya; Adamson, John H; Borah, Khushboo; Beste, Dany J V; Lee, Bei Shi; Pethe, Kevin; Rousseau, Simon; Krieger, Inna; Sacchettini, James C; Glasgow, Joel N; Steyn, Adrie J C

The Structural Basis of T4 Phage Lysis Control: DNA as the Signal for Lysis Inhibition.

T4噬菌体裂解控制的结构基础:DNA作为裂解抑制的信号

Krieger Inna V, Kuznetsov Vladimir, Chang Jeng-Yih, Zhang Junjie, Moussa Samir H, Young Ryland F, Sacchettini James C

Correction: TnSeq of Mycobacterium tuberculosis clinical isolates reveals strain-specific antibiotic liabilities

更正:结核分枝杆菌临床分离株的TnSeq分析揭示了菌株特异性的抗生素敏感性。

Carey, Allison F; Rock, Jeremy M; Krieger, Inna V; Chase, Michael R; Fernandez-Suarez, Marta; Gagneux, Sebastien; Sacchettini, James C; Ioerger, Thomas R; Fortune, Sarah M

Structural destabilization of tropomyosin induced by the cardiomyopathy-linked mutation R21H

心肌病相关突变R21H诱导的原肌球蛋白结构不稳定

Ly, Thu; Krieger, Inna; Tolkatchev, Dmitri; Krone, Cheyenna; Moural, Timothy; Samatey, Fadel A; Kang, ChulHee; Kostyukova, Alla S

TnSeq of Mycobacterium tuberculosis clinical isolates reveals strain-specific antibiotic liabilities

对结核分枝杆菌临床分离株进行TnSeq测序,揭示了菌株特异性的抗生素敏感性。

Carey, Allison F; Rock, Jeremy M; Krieger, Inna V; Chase, Michael R; Fernandez-Suarez, Marta; Gagneux, Sebastien; Sacchettini, James C; Ioerger, Thomas R; Fortune, Sarah M