日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

SuFEx-based antitubercular compound irreversibly inhibits Pks13

基于 SuFEx 的抗结核化合物不可逆地抑制 Pks13

Krieger, Inna V; Sukheja, Paridhi; Yang, Baiyuan; Tang, Su; Selle, Daniel; Woods, Ashley; Engelhart, Curtis; Kumar, Pradeep; Harbut, Michael B; Liu, Dongdong; Tsuda, Brendan; Qin, Bo; Bare, Grant A L; Li, Gencheng; Chi, Victor; Gambacurta, Julian; Hvizdos, Janine; Reagan, Matthew; Jones, Isabelle L; Massoudi, Lisa M; Woolhiser, Lisa K; Cascioferro, Alessandro; Kundrick, Erica; Singh, Parul; Reiley, William; Ioerger, Thomas R; Kandula, Dilipkumar Reddy; McCabe, Jacob W; Guo, Taijie; Alland, David; Boshoff, Helena I; Schnappinger, Dirk; Robertson, Gregory T; Mdluli, Khisi; Lee, Kyoung-Jin; Dong, Jiajia; Li, Shuangwei; Schultz, Peter G; Joseph, Sean B; Love, Melissa S; Sharpless, K Barry; Petrassi, H Michael; Chatterjee, Arnab K; Sacchettini, James C; McNamara, Case W

An oral non-covalent non-peptidic inhibitor of SARS-CoV-2 Mpro ameliorates viral replication and pathogenesis in vivo.

SARS-CoV-2 Mpro 的口服非共价非肽抑制剂可改善体内病毒复制和致病性

Zhou Nian E, Tang Su, Bian Xuelin, Parai Maloy K, Krieger Inna V, Flores Armando, Jaiswal Pradeep K, Bam Radha, Wood Jeremy L, Shi Zhe, Stevens Laura J, Scobey Trevor, Diefenbacher Meghan V, Moreira Fernando R, Baric Thomas J, Acharya Arjun, Shin Joonyoung, Rathi Manish M, Wolff Karen C, Riva Laura, Bakowski Malina A, McNamara Case W, Catanzaro Nicholas J, Graham Rachel L, Schultz David C, Cherry Sara, Kawaoka Yoshihiro, Halfmann Peter J, Baric Ralph S, Denison Mark R, Sheahan Timothy P, Sacchettini James C

Structural anatomy of Protein Kinase C C1 domain interactions with diacylglycerol and other agonists

蛋白激酶C C1结构域与二酰甘油和其他激动剂相互作用的结构解剖

Katti, Sachin S; Krieger, Inna V; Ann, Jihyae; Lee, Jeewoo; Sacchettini, James C; Igumenova, Tatyana I

The Structural Basis of T4 Phage Lysis Control: DNA as the Signal for Lysis Inhibition.

T4噬菌体裂解控制的结构基础:DNA作为裂解抑制的信号

Krieger Inna V, Kuznetsov Vladimir, Chang Jeng-Yih, Zhang Junjie, Moussa Samir H, Young Ryland F, Sacchettini James C

Correction: TnSeq of Mycobacterium tuberculosis clinical isolates reveals strain-specific antibiotic liabilities

更正:结核分枝杆菌临床分离株的TnSeq分析揭示了菌株特异性的抗生素敏感性。

Carey, Allison F; Rock, Jeremy M; Krieger, Inna V; Chase, Michael R; Fernandez-Suarez, Marta; Gagneux, Sebastien; Sacchettini, James C; Ioerger, Thomas R; Fortune, Sarah M

TnSeq of Mycobacterium tuberculosis clinical isolates reveals strain-specific antibiotic liabilities

对结核分枝杆菌临床分离株进行TnSeq测序,揭示了菌株特异性的抗生素敏感性。

Carey, Allison F; Rock, Jeremy M; Krieger, Inna V; Chase, Michael R; Fernandez-Suarez, Marta; Gagneux, Sebastien; Sacchettini, James C; Ioerger, Thomas R; Fortune, Sarah M

Mycobacterium tuberculosis Malate Synthase Structures with Fragments Reveal a Portal for Substrate/Product Exchange

结核分枝杆菌苹果酸合酶的结构片段揭示了底物/产物交换的通道

Huang, Hsiao-Ling; Krieger, Inna V; Parai, Maloy K; Gawandi, Vijay B; Sacchettini, James C

Structure-guided discovery of phenyl-diketo acids as potent inhibitors of M. tuberculosis malate synthase

结构导向发现苯基二酮酸是结核分枝杆菌苹果酸合酶的强效抑制剂

Krieger, Inna V; Freundlich, Joel S; Gawandi, Vijay B; Roberts, Justin P; Gawandi, Vidyadhar B; Sun, Qingan; Owen, Joshua L; Fraile, Maria T; Huss, Sofia I; Lavandera, Jose-Luis; Ioerger, Thomas R; Sacchettini, James C