日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Engineering a Coiled-Coil Protein for DARPin Presentation as a Potent SARS-CoV-2 Therapeutic

构建用于DARPin呈递的卷曲螺旋蛋白作为一种有效的SARS-CoV-2治疗药物

Mai, Linh D; Cheedarla, Narayanaiah; Krishnathas, Siamalan; Sadab, Ishmamul H; Gray, Mikaela A; Lv, Wei; Dhankher, Anshul; Roback, John D; Neish, Andrew S; Champion, Julie A

Structure-Based Rational Design of a Selective Hydrolase Inhibitor of the Severe Acute Respiratory Syndrome Coronavirus-2 Nsp3 Macrodomain

基于结构的严重急性呼吸综合征冠状病毒2 Nsp3宏结构域选择性水解酶抑制剂的合理设计

Krishnathas, Robin; Mineev, Konstantin S; Fourkiotis, Nikolaos K; Touret, Franck; Sideras-Bisdekis, Christos; Tsika, Aikaterini C; Gande, Santosh Lakshmi; Linhard, Verena; Sreeramulu, Sridhar; Lennartz, Frank; Weiss, Manfred S; Coutard, Bruno; Spyroulias, Georgios A; Schwalbe, Harald

2-Desaza-annomontine (C81) impedes angiogenesis through reduced VEGFR2 expression derived from inhibition of CDC2-like kinases

2-Desaza-annomontine (C81) 通过抑制 CDC2 样激酶来降低 VEGFR2 表达,从而阻碍血管生成

T J Zech, A Wolf, M Hector, I Bischoff-Kont, G M Krishnathas, S Kuntschar, T Schmid, F Bracher, T Langmann, R Fürst

Knock-out of 5-lipoxygenase in overexpressing tumor cells-consequences on gene expression and cellular function

5-脂氧合酶在过度表达的肿瘤细胞中的敲除——对基因表达和细胞功能的影响

Hannah Weisser, Tamara Göbel, G Melissa Krishnathas, Marius Kreiß, Carlo Angioni, Duran Sürün, Dominique Thomas, Tobias Schmid, Ann-Kathrin Häfner, Astrid S Kahnt

Comprehensive Fragment Screening of the SARS-CoV-2 Proteome Explores Novel Chemical Space for Drug Development

对SARS-CoV-2蛋白质组的全面片段筛选探索了药物研发的新化学空间

Berg, Hannes; Wirtz Martin, Maria A; Altincekic, Nadide; Alshamleh, Islam; Kaur Bains, Jasleen; Blechar, Julius; Ceylan, Betül; de Jesus, Vanessa; Dhamotharan, Karthikeyan; Fuks, Christin; Gande, Santosh L; Hargittay, Bruno; Hohmann, Katharina F; Hutchison, Marie T; Marianne Korn, Sophie; Krishnathas, Robin; Kutz, Felicitas; Linhard, Verena; Matzel, Tobias; Meiser, Nathalie; Niesteruk, Anna; Pyper, Dennis J; Schulte, Linda; Trucks, Sven; Azzaoui, Kamal; Blommers, Marcel J J; Gadiya, Yojana; Karki, Reagon; Zaliani, Andrea; Gribbon, Philip; da Silva Almeida, Marcius; Dinis Anobom, Cristiane; Bula, Anna L; Bütikofer, Matthias; Putinhon Caruso, Ícaro; Caterina Felli, Isabella; Da Poian, Andrea T; Cardoso de Amorim, Gisele; Fourkiotis, Nikolaos K; Gallo, Angelo; Ghosh, Dhiman; Gomes-Neto, Francisco; Gorbatyuk, Oksana; Hao, Bing; Kurauskas, Vilius; Lecoq, Lauriane; Li, Yunfeng; Cunha Mebus-Antunes, Nathane; Mompeán, Miguel; Cristtina Neves-Martins, Thais; Ninot-Pedrosa, Martí; Pinheiro, Anderson S; Pontoriero, Letizia; Pustovalova, Yulia; Riek, Roland; Robertson, Angus J; Jose Abi Saad, Marie; Treviño, Miguel Á; Tsika, Aikaterini C; Almeida, Fabio C L; Bax, Ad; Henzler-Wildman, Katherine; Hoch, Jeffrey C; Jaudzems, Kristaps; Laurents, Douglas V; Orts, Julien; Pierattelli, Roberta; Spyroulias, Georgios A; Duchardt-Ferner, Elke; Ferner, Jan; Fürtig, Boris; Hengesbach, Martin; Löhr, Frank; Qureshi, Nusrat; Richter, Christian; Saxena, Krishna; Schlundt, Andreas; Sreeramulu, Sridhar; Wacker, Anna; Weigand, Julia E; Wirmer-Bartoschek, Julia; Wöhnert, Jens; Schwalbe, Harald

Binding Adaptation of GS-441524 Diversifies Macro Domains and Downregulates SARS-CoV-2 de-MARylation Capacity

GS-441524 的结合适应性使大结构域多样化并下调 SARS-CoV-2 去甲基化能力

Aikaterini C Tsika, Angelo Gallo, Nikolaos K Fourkiotis, Aikaterini I Argyriou, Sridhar Sreeramulu, Frank Löhr, Vladimir V Rogov, Christian Richter, Verena Linhard, Santosh L Gande, Nadide Altincekic, Robin Krishnathas, Isam Elamri, Harald Schwalbe, Jan Wollenhaupt, Manfred S Weiss, Georgios A Spyro

Large-Scale Recombinant Production of the SARS-CoV-2 Proteome for High-Throughput and Structural Biology Applications

用于高通量和结构生物学应用的SARS-CoV-2蛋白质组的大规模重组生产

Altincekic, Nadide; Korn, Sophie Marianne; Qureshi, Nusrat Shahin; Dujardin, Marie; Ninot-Pedrosa, Martí; Abele, Rupert; Abi Saad, Marie Jose; Alfano, Caterina; Almeida, Fabio C L; Alshamleh, Islam; de Amorim, Gisele Cardoso; Anderson, Thomas K; Anobom, Cristiane D; Anorma, Chelsea; Bains, Jasleen Kaur; Bax, Adriaan; Blackledge, Martin; Blechar, Julius; Böckmann, Anja; Brigandat, Louis; Bula, Anna; Bütikofer, Matthias; Camacho-Zarco, Aldo R; Carlomagno, Teresa; Caruso, Icaro Putinhon; Ceylan, Betül; Chaikuad, Apirat; Chu, Feixia; Cole, Laura; Crosby, Marquise G; de Jesus, Vanessa; Dhamotharan, Karthikeyan; Felli, Isabella C; Ferner, Jan; Fleischmann, Yanick; Fogeron, Marie-Laure; Fourkiotis, Nikolaos K; Fuks, Christin; Fürtig, Boris; Gallo, Angelo; Gande, Santosh L; Gerez, Juan Atilio; Ghosh, Dhiman; Gomes-Neto, Francisco; Gorbatyuk, Oksana; Guseva, Serafima; Hacker, Carolin; Häfner, Sabine; Hao, Bing; Hargittay, Bruno; Henzler-Wildman, K; Hoch, Jeffrey C; Hohmann, Katharina F; Hutchison, Marie T; Jaudzems, Kristaps; Jović, Katarina; Kaderli, Janina; Kalniņš, Gints; Kaņepe, Iveta; Kirchdoerfer, Robert N; Kirkpatrick, John; Knapp, Stefan; Krishnathas, Robin; Kutz, Felicitas; Zur Lage, Susanne; Lambertz, Roderick; Lang, Andras; Laurents, Douglas; Lecoq, Lauriane; Linhard, Verena; Löhr, Frank; Malki, Anas; Bessa, Luiza Mamigonian; Martin, Rachel W; Matzel, Tobias; Maurin, Damien; McNutt, Seth W; Mebus-Antunes, Nathane Cunha; Meier, Beat H; Meiser, Nathalie; Mompeán, Miguel; Monaca, Elisa; Montserret, Roland; Mariño Perez, Laura; Moser, Celine; Muhle-Goll, Claudia; Neves-Martins, Thais Cristtina; Ni, Xiamonin; Norton-Baker, Brenna; Pierattelli, Roberta; Pontoriero, Letizia; Pustovalova, Yulia; Ohlenschläger, Oliver; Orts, Julien; Da Poian, Andrea T; Pyper, Dennis J; Richter, Christian; Riek, Roland; Rienstra, Chad M; Robertson, Angus; Pinheiro, Anderson S; Sabbatella, Raffaele; Salvi, Nicola; Saxena, Krishna; Schulte, Linda; Schiavina, Marco; Schwalbe, Harald; Silber, Mara; Almeida, Marcius da Silva; Sprague-Piercy, Marc A; Spyroulias, Georgios A; Sreeramulu, Sridhar; Tants, Jan-Niklas; Tārs, Kaspars; Torres, Felix; Töws, Sabrina; Treviño, Miguel Á; Trucks, Sven; Tsika, Aikaterini C; Varga, Krisztina; Wang, Ying; Weber, Marco E; Weigand, Julia E; Wiedemann, Christoph; Wirmer-Bartoschek, Julia; Wirtz Martin, Maria Alexandra; Zehnder, Johannes; Hengesbach, Martin; Schlundt, Andreas

Identification of 4-N-[2-(4-phenoxyphenyl)ethyl]quinazoline-4,6-diamine as a novel, highly potent and specific inhibitor of mitochondrial complex I

鉴定出 4-N-[2-(4-苯氧基苯基)乙基]喹唑啉-4,6-二胺是一种新型、高效且特异性的线粒体复合物 I 抑制剂。

Krishnathas, Robin; Bonke, Erik; Dröse, Stefan; Zickermann, Volker; Nasiri, Hamid R