Structure-Guided Development of a Potent BioA Inhibitor Validates Biotin Synthesis Inhibition as a Therapeutic Strategy for Tuberculosis
结构导向开发高效BioA抑制剂验证了生物素合成抑制作为结核病治疗策略的有效性
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doi:10.1101/2025.09.24.678246
Liu, Qiang; Wallach, Joshua B; Jayasinghe, Yahani P; Sullivan, Mark R; Proietto, Julianna; Rodriguez, Suyapa; Vo, Sang; Boshoff, Helena I M; Jia, Ziyi; Ostrer, Lev; Mehdiratta, Kritee; Shi, Rui; Dartois, Véronique; Baughn, Anthony D; Rubin, Eric J; Ronning, Donald R; Zimmerman, Matthew D; Schnappinger, Dirk; Aldrich, Courtney C