Design, synthesis, and pharmacological characterization of N- and O-substituted 5,6,7,8-tetrahydro-4H-isoxazolo[4,5-d]azepin-3-ol analogues: novel 5-HT(2A)/5-HT(2C) receptor agonists with pro-cognitive properties
和 O 取代的 5,6,7,8-四氢-4H-异恶唑并[4,5-d]氮杂卓-3-醇类似物的设计、合成和药理学表征:具有促认知特性的新型 5-HT(2A)/5-HT(2C) 受体激动剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm301656h
Anders A Jensen, Niels Plath, Martin H F Pedersen, Vignir Isberg, Jacob Krall, Petrine Wellendorph, Tine B Stensbøl, David E Gloriam, Povl Krogsgaard-Larsen, Bente Frølund